Lista de obras - Thierry Billard - Dominio Público Uruguay

18F-F13640 preclinical evaluation in rodent, cat and primate as a 5-HT1A receptor agonist for PET neuroimaging

scientific article published on 05 May 2018

A Metal-Free Route to Heterocyclic Trifluoromethyl- and Fluoroalkylselenolated Molecules

artículo científico publicado en 2017

A postmortem study to compare agonist and antagonist 5-HT1A receptor-binding sites in Alzheimer's disease.

artículo científico publicado en 2014

Agonist and antagonist bind differently to 5-HT1A receptors during Alzheimer's disease: A post-mortem study with PET radiopharmaceuticals

artículo científico publicado en 2016

Amyloid-Beta Radiotracer [18F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue.

artículo científico publicado en 2018

Base-catalyzed electrophilic trifluoromethylthiolation of terminal alkynes.

artículo científico publicado en 2013

Benzyltrifluoromethyl (or Fluoroalkyl) Selenide: Reagent for Electrophilic Trifluoromethyl (or Fluoroalkyl) Selenolation

artículo científico publicado en 2016

Binding of the PET radiotracer [¹⁸F]BF227 does not reflect the presence of alpha-synuclein aggregates in transgenic mice

artículo científico publicado en 2014

Characterization and Reliability of [18F]2FNQ1P in Cynomolgus Monkeys as a PET Radiotracer for Serotonin 5-HT6 Receptors.

artículo científico publicado en 2017

Comparison of 4 radiolabeled antagonists for serotonin 5-HT(7) receptor neuroimaging: toward the first PET radiotracer

artículo científico publicado en 2011

Copper-Catalyzed Perfluoroalkylthiolation of Alkynes with Perfluoroalkanesulfenamides

artículo científico publicado en 2016

Difluoro(aryl)(perfluoroalkyl)-λ4 -sulfanes and Selanes: Missing Links of Trichloroisocyanuric Acid/Potassium Fluoride Chemistry

artículo científico publicado en 2019

Direct Electrophilic (Benzenesulfonyl)Difluoromethylthiolation with a Shelf-Stable Reagent

artículo científico publicado en 2016

Direct electrophilic N-trifluoromethylthiolation of amines with trifluoromethanesulfenamide.

artículo científico publicado en 2013

Electrophilic trifluoromethanesulfanylation of organometallic species with trifluoromethanesulfanamides

artículo científico publicado en 2012

Electrophilic trifluoromethylselenolation of terminal alkynes with Se-(trifluoromethyl) 4-methylbenzenesulfonoselenoate

artículo científico publicado en 2017

Electrophilic trifluoromethylthiolation of carbonyl compounds

scientific article published on 30 May 2014

Evaluation of Myelin Radiotracers in the Lysolecithin Rat Model of Focal Demyelination: Beware of Pitfalls!

scientific article published on 29 May 2019

Evaluation of [ F]2FP3 in pigs and non-human primates

artículo científico publicado en 2018

Exploring the Reactivity of Trifluoromethyl Tolueneselenosulfonate with Alkynes under Copper Catalysis

artículo científico publicado en 2017

Fluorous l-Carbidopa Precursors: Highly Enantioselective Synthesis and Computational Prediction of Bioactivity

artículo científico publicado en 2017

Formation of C-SCF3 bonds through direct trifluoromethylthiolation.

artículo científico publicado en 2013

Generation of the SCF3 Radical by Photoredox Catalysis: Intra- and Intermolecular Carbotrifluoromethylthiolation of Alkenes

artículo científico publicado en 2017

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α-Synuclein PET Imaging

artículo científico publicado en 2018

Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate

artículo científico publicado en 2020

Mild and Soft Catalyzed Trifluoromethylthiolation of Boronic Acids: The Crucial Role of Water

artículo científico publicado en 2015

Molecular imaging of the serotonin 5-HT7 receptors: from autoradiography to positron emission tomography

artículo científico publicado en 2014

Preclinical evaluation of [18F]2FNQ1P as the first fluorinated serotonin 5-HT6 radioligand for PET imaging.

artículo científico publicado en 2014

Radiosynthesis and preclinical evaluation of 18F-F13714 as a fluorinated 5-HT1A receptor agonist radioligand for PET neuroimaging

artículo científico publicado en 2012

Superacid-Catalyzed Trifluoromethylthiolation of Aromatic Amines

artículo científico publicado en 2016

Syntheses, radiolabelings, and in vitro evaluations of fluorinated PET radioligands of 5-HT6 serotoninergic receptors.

artículo científico publicado en 2014

Synthesis and pharmacological evaluation of a new series of radiolabeled ligands for 5-HT7 receptor PET neuroimaging.

artículo científico publicado en 2014

Synthetic Approaches to Trifluoromethoxy-Substituted Compounds

artículo científico publicado en 2016

Synthetic Approaches to Trifluoromethylselenolated Compounds

artículo científico publicado en 2017

Trifluoromethyl- and Fluoroalkylselenolations of Alkynyl Copper(I) Compounds.

artículo científico publicado en 2017

Visible-Light-Mediated Metal-Free Synthesis of Trifluoromethylselenolated Arenes

artículo científico publicado en 2018

Visible-light promoted fluoroalkylselenolation: toward the reactivity of unsaturated compounds

artículo científico publicado en 2018

[11C]PF-3274167 as a PET radiotracer of oxytocin receptors: Radiosynthesis and evaluation in rat brain

artículo científico publicado en 2017

Lista de obras de Thierry Billard

18F-F13640 preclinical evaluation in rodent, cat and primate as a 5-HT1A receptor agonist for PET neuroimaging

A Metal-Free Route to Heterocyclic Trifluoromethyl- and Fluoroalkylselenolated Molecules

A postmortem study to compare agonist and antagonist 5-HT1A receptor-binding sites in Alzheimer's disease.

Agonist and antagonist bind differently to 5-HT1A receptors during Alzheimer's disease: A post-mortem study with PET radiopharmaceuticals

Amyloid-Beta Radiotracer [18F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue.

Base-catalyzed electrophilic trifluoromethylthiolation of terminal alkynes.

Benzyltrifluoromethyl (or Fluoroalkyl) Selenide: Reagent for Electrophilic Trifluoromethyl (or Fluoroalkyl) Selenolation

Binding of the PET radiotracer [¹⁸F]BF227 does not reflect the presence of alpha-synuclein aggregates in transgenic mice

Characterization and Reliability of [18F]2FNQ1P in Cynomolgus Monkeys as a PET Radiotracer for Serotonin 5-HT6 Receptors.

Comparison of 4 radiolabeled antagonists for serotonin 5-HT(7) receptor neuroimaging: toward the first PET radiotracer

Copper-Catalyzed Perfluoroalkylthiolation of Alkynes with Perfluoroalkanesulfenamides

Difluoro(aryl)(perfluoroalkyl)-λ4 -sulfanes and Selanes: Missing Links of Trichloroisocyanuric Acid/Potassium Fluoride Chemistry

Direct Electrophilic (Benzenesulfonyl)Difluoromethylthiolation with a Shelf-Stable Reagent

Direct electrophilic N-trifluoromethylthiolation of amines with trifluoromethanesulfenamide.

Electrophilic trifluoromethanesulfanylation of organometallic species with trifluoromethanesulfanamides

Electrophilic trifluoromethylselenolation of terminal alkynes with Se-(trifluoromethyl) 4-methylbenzenesulfonoselenoate

Electrophilic trifluoromethylthiolation of carbonyl compounds

Evaluation of Myelin Radiotracers in the Lysolecithin Rat Model of Focal Demyelination: Beware of Pitfalls!

Evaluation of [ F]2FP3 in pigs and non-human primates

Exploring the Reactivity of Trifluoromethyl Tolueneselenosulfonate with Alkynes under Copper Catalysis

Fluorous l-Carbidopa Precursors: Highly Enantioselective Synthesis and Computational Prediction of Bioactivity

Formation of C-SCF3 bonds through direct trifluoromethylthiolation.

Generation of the SCF3 Radical by Photoredox Catalysis: Intra- and Intermolecular Carbotrifluoromethylthiolation of Alkenes

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α-Synuclein PET Imaging

Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate

Mild and Soft Catalyzed Trifluoromethylthiolation of Boronic Acids: The Crucial Role of Water

Molecular imaging of the serotonin 5-HT7 receptors: from autoradiography to positron emission tomography

Preclinical evaluation of [18F]2FNQ1P as the first fluorinated serotonin 5-HT6 radioligand for PET imaging.

Radiosynthesis and preclinical evaluation of 18F-F13714 as a fluorinated 5-HT1A receptor agonist radioligand for PET neuroimaging

Superacid-Catalyzed Trifluoromethylthiolation of Aromatic Amines

Syntheses, radiolabelings, and in vitro evaluations of fluorinated PET radioligands of 5-HT6 serotoninergic receptors.

Synthesis and pharmacological evaluation of a new series of radiolabeled ligands for 5-HT7 receptor PET neuroimaging.

Synthetic Approaches to Trifluoromethoxy-Substituted Compounds

Synthetic Approaches to Trifluoromethylselenolated Compounds

Trifluoromethyl- and Fluoroalkylselenolations of Alkynyl Copper(I) Compounds.

Visible-Light-Mediated Metal-Free Synthesis of Trifluoromethylselenolated Arenes

Visible-light promoted fluoroalkylselenolation: toward the reactivity of unsaturated compounds

[11C]PF-3274167 as a PET radiotracer of oxytocin receptors: Radiosynthesis and evaluation in rat brain