Lista de obras - Greta Varchi - Dominio Público Uruguay

1,4-Substituted Triazoles as Nonsteroidal Anti-Androgens for Prostate Cancer Treatment

artículo científico publicado en 2017

2-Hydroxypropyl-β-cyclodextrin-enhanced pharmacokinetics of cabotegravir from a nanofluidic implant for HIV pre-exposure prophylaxis

artículo científico publicado en 2019

A SMYD3 Small-Molecule Inhibitor Impairing Cancer Cell Growth

artículo científico publicado en 2015

A new avenue toward androgen receptor pan-antagonists: C2 sterically hindered substitution of hydroxy-propanamides

artículo científico publicado en 2014

A photodynamic bifunctional conjugate for prostate cancer: an in vitro mechanistic study

artículo científico publicado en 2016

A small-molecule targeting the microRNA binding domain of argonaute 2 improves the retinoic acid differentiation response of the acute promyelocytic leukemia cell line NB4.

artículo científico publicado en 2014

Androgen Receptor Targeted Conjugate for Bimodal Photodynamic Therapy of Prostate Cancer in Vitro.

artículo científico publicado en 2015

Anticancer activity of paclitaxel-loaded keratin nanoparticles in two-dimensional and perfused three-dimensional breast cancer models

Camptothecin and thiocamptothecin: the role of sulfur in shifting the hydrolysis equilibrium towards the closed lactone form

artículo científico publicado en 2011

Complex Nanostructures Based on Oligonucleotide Optical Switches and Nanoparticles for Intracellular mRNA Sensing and Silencing

Concise and stereocontrolled synthesis of pseudo-C2-symmetric diamino alcohols and triamines for use in HIV protease inhibitors.

artículo científico publicado en 2003

Copper Catalyzed Conjugate Addition of Highly Functionalized Arylmagnesium Compounds to Enones

article

Core-shell poly-methyl methacrylate nanoparticles covalently functionalized with a non-symmetric porphyrin for anticancer photodynamic therapy

Core-shell poly-methylmethacrylate nanoparticles as effective carriers of electrostatically loaded anionic porphyrin

article published in 2013

Development of near-infrared photoactivable phthalocyanine-loaded nanoparticles to kill tumor cells: An improved tool for photodynamic therapy of solid cancers.

artículo científico publicado en 2016

Direct preparation of polyfunctional amino-substituted arylmagnesium reagents via an iodine-magnesium exchange reaction

artículo científico publicado en 2003

Effect of small molecules modulating androgen receptor (SARMs) in human prostate cancer models

artículo científico publicado en 2013

Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors

Enantiomeric HPLC resolution and absolute stereochemistry assignment of a new poligamain derivative

artículo científico publicado en 2012

Engineered porphyrin loaded core-shell nanoparticles for selective sonodynamic anticancer treatment

artículo científico publicado en 2015

Extremely facile formation and high reactivity of new thioacylsilanes containing the ferrocene moiety

Functionalized Keratin as Nanotechnology-Based Drug Delivery System for the Pharmacological Treatment of Osteosarcoma ⬇️

artículo científico publicado en 2018

Highlights of the Fifth International Workshop on Nitric Oxide and Cancer

artículo científico publicado en 2016

Intracellular Nanosensing and Nanodelivery by PMMA Nanoparticles

Intracellular delivery of molecular beacons by PMMA nanoparticles and carbon nanotubes for mRNA sensing

Keratin nanoparticles co-delivering Docetaxel and Chlorin e6 promote synergic interaction between chemo- and photo-dynamic therapies

artículo científico publicado en 2019

Keratin-hydrotalcites hybrid films for drug delivery applications

Light-Induced Therapies for Prostate Cancer Treatment

scientific article published on 29 October 2019

Mesenchymal stem cells as delivery vehicle of porphyrin loaded nanoparticles: effective photoinduced in vitro killing of osteosarcoma

artículo científico publicado en 2013

Methylene Blue Doped Films of Wool Keratin with Antimicrobial Photodynamic Activity

artículo científico publicado en 2015

Molecular beacon-decorated polymethylmethacrylate core-shell fluorescent nanoparticles for the detection of survivin mRNA in human cancer cells

artículo científico publicado en 2016

New Polyfunctional Magnesium Reagents for Organic Synthesis

artículo científico publicado en 2000

New chiral allylaminosilanes and their use in asymmetric Sakurai reactions

Non-Steroidal Androgen Receptor Antagonists and Prostate Cancer: a Survey on Chemical Structures Binding this Fast-Mutating Target

artículo científico publicado en 2019

Nonsteroidal androgen receptor ligands: versatile syntheses and biological data

artículo científico publicado en 2012

Novel 20(S)-sulfonylamidine derivatives of camptothecin and the use thereof as a potent antitumor agent: a patent evaluation of WO2015048365 (A1).

artículo científico publicado en 2016

Oligonucleotide switches and nanomaterials for intracellular mRNA sensing

article published in 2013

Optical biosensor analysis in studying new synthesized bicalutamide analogs binding to androgen receptor

artículo científico publicado en 2014

Organic solvent-free preparation of keratin nanoparticles as doxorubicin carriers for antitumour activity

article

Polyenylcyclopropane carboxylic esters with high insecticidal activity

artículo científico publicado en 2014

Polymer nanoparticles with electrostatically loaded multicargo for combined cancer phototherapy

artículo científico publicado en 2015

Polymeric nanoparticles enhance the sonodynamic activity of meso-tetrakis (4-sulfonatophenyl) porphyrin in an in vitro neuroblastoma model

artículo científico publicado en 2013

Polymethylmethacrylate nanoparticles as carrier of an oligodeoxynucleotide molecular beacon specific for survivin mRNA in A549 human lung adenocarcinoma epithelial cells

Quinazolinedione SIRT6 inhibitors sensitize cancer cells to chemotherapeutics

Rapid microwave-assisted deprotection of N-Cbz and N-Bn derivatives

SILK.IT project: Silk Italian Technology for industrial biomanufacturing

article

Selective sensitiveness of mesenchymal stem cells to shock waves leads to anticancer effect in human cancer cell co-cultures.

artículo científico publicado en 2017

Semisynthesis, biological activity, and molecular modeling studies of C-ring-modified camptothecins.

artículo científico publicado en 2009

Silk fibroin film from golden-yellow Bombyx mori is a biocomposite that contains lutein and promotes axonal growth of primary neurons

artículo científico publicado en 2016

Silylcupration of acylimidazolides: a new synthesis of α-aminoacylsilanes and their synthetic applications

Species-dependent binding of new synthesized bicalutamide analogues to albumin by optical biosensor analysis

artículo científico publicado en 2015

Stereoselective Three-Carbon and Two-Carbon Elongation of the Carbon Chain inN-Boc-Protected α-Aminoacylsilanes: An Entry to Functionalized β-Amino Alcohols and to Statine Analogues

Stereoselective one-pot synthesis of constrained N,O-orthogonally protected C-glycosyl norstatines [C(1')-aminoglycosyl-1,3-dioxolan-4-ones]

artículo científico publicado en 2006

Structure-activity relationship study of 16 a-thiocamptothecins: an integrated in vitro and in silico approach

artículo científico publicado en 2010

Sulfonates-PMMA nanoparticles conjugates: a versatile system for multimodal application

artículo científico publicado en 2012

Synthesis and reactivity of achiral and of a novel planar chiral thioferrocenoylsilanes

Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs

Synthesis of Heterocycles Through Hydrosilylation, Silylformylation, Silylcarbocyclization and Cyclohydrocarbonylation Reactions

article published in 2006

Synthesis of chiral β2,2,3-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-β-lactams by double asymmetric induction

Synthesis of deserpidine from reserpine

artículo científico publicado en 2005

Synthesis of α2,2,β3-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates toN-(tert-Butylsulfinyl) Imines

article

TPPS supported on core–shell PMMA nanoparticles: the development of continuous-flow membrane-mediated electrocoagulation as a photocatalyst processing method in aqueous media

article

The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin−Polyamine Conjugates

scholarly article by Cristian Samorì et al published 18 March 2009 in Bioconjugate Chemistry

The first synthesis of N,O-protected β2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding β-lactams

The role of polyamine architecture on the pharmacological activity of open lactone camptothecin-polyamine conjugates

artículo científico publicado en 2008

Thiocamptothecin

artículo científico publicado en 2008

Thiophene-based compounds as fluorescent tags to study mesenchymal stem cell uptake and release of taxanes.

artículo científico publicado en 2014

Unprecedented Behavior of (9 R)-9-Hydroxystearic Acid-Loaded Keratin Nanoparticles on Cancer Cell Cycle

artículo científico publicado en 2019

Wool Keratin 3D Scaffolds with Light-Triggered Antimicrobial Activity.

artículo científico publicado en 2016

Lista de obras de Greta Varchi

1,4-Substituted Triazoles as Nonsteroidal Anti-Androgens for Prostate Cancer Treatment

2-Hydroxypropyl-β-cyclodextrin-enhanced pharmacokinetics of cabotegravir from a nanofluidic implant for HIV pre-exposure prophylaxis

A SMYD3 Small-Molecule Inhibitor Impairing Cancer Cell Growth

A new avenue toward androgen receptor pan-antagonists: C2 sterically hindered substitution of hydroxy-propanamides

A photodynamic bifunctional conjugate for prostate cancer: an in vitro mechanistic study

A small-molecule targeting the microRNA binding domain of argonaute 2 improves the retinoic acid differentiation response of the acute promyelocytic leukemia cell line NB4.

Androgen Receptor Targeted Conjugate for Bimodal Photodynamic Therapy of Prostate Cancer in Vitro.

Anticancer activity of paclitaxel-loaded keratin nanoparticles in two-dimensional and perfused three-dimensional breast cancer models

Camptothecin and thiocamptothecin: the role of sulfur in shifting the hydrolysis equilibrium towards the closed lactone form

Complex Nanostructures Based on Oligonucleotide Optical Switches and Nanoparticles for Intracellular mRNA Sensing and Silencing

Concise and stereocontrolled synthesis of pseudo-C2-symmetric diamino alcohols and triamines for use in HIV protease inhibitors.

Copper Catalyzed Conjugate Addition of Highly Functionalized Arylmagnesium Compounds to Enones

Core-shell poly-methyl methacrylate nanoparticles covalently functionalized with a non-symmetric porphyrin for anticancer photodynamic therapy

Core-shell poly-methylmethacrylate nanoparticles as effective carriers of electrostatically loaded anionic porphyrin

Development of near-infrared photoactivable phthalocyanine-loaded nanoparticles to kill tumor cells: An improved tool for photodynamic therapy of solid cancers.

Direct preparation of polyfunctional amino-substituted arylmagnesium reagents via an iodine-magnesium exchange reaction

Effect of small molecules modulating androgen receptor (SARMs) in human prostate cancer models

Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors

Enantiomeric HPLC resolution and absolute stereochemistry assignment of a new poligamain derivative

Engineered porphyrin loaded core-shell nanoparticles for selective sonodynamic anticancer treatment

Extremely facile formation and high reactivity of new thioacylsilanes containing the ferrocene moiety

Functionalized Keratin as Nanotechnology-Based Drug Delivery System for the Pharmacological Treatment of Osteosarcoma ⬇️

Highlights of the Fifth International Workshop on Nitric Oxide and Cancer

Intracellular Nanosensing and Nanodelivery by PMMA Nanoparticles

Intracellular delivery of molecular beacons by PMMA nanoparticles and carbon nanotubes for mRNA sensing

Keratin nanoparticles co-delivering Docetaxel and Chlorin e6 promote synergic interaction between chemo- and photo-dynamic therapies

Keratin-hydrotalcites hybrid films for drug delivery applications

Light-Induced Therapies for Prostate Cancer Treatment

Mesenchymal stem cells as delivery vehicle of porphyrin loaded nanoparticles: effective photoinduced in vitro killing of osteosarcoma

Methylene Blue Doped Films of Wool Keratin with Antimicrobial Photodynamic Activity

Molecular beacon-decorated polymethylmethacrylate core-shell fluorescent nanoparticles for the detection of survivin mRNA in human cancer cells

New Polyfunctional Magnesium Reagents for Organic Synthesis

New chiral allylaminosilanes and their use in asymmetric Sakurai reactions

Non-Steroidal Androgen Receptor Antagonists and Prostate Cancer: a Survey on Chemical Structures Binding this Fast-Mutating Target

Nonsteroidal androgen receptor ligands: versatile syntheses and biological data

Novel 20(S)-sulfonylamidine derivatives of camptothecin and the use thereof as a potent antitumor agent: a patent evaluation of WO2015048365 (A1).

Oligonucleotide switches and nanomaterials for intracellular mRNA sensing

Optical biosensor analysis in studying new synthesized bicalutamide analogs binding to androgen receptor

Organic solvent-free preparation of keratin nanoparticles as doxorubicin carriers for antitumour activity

Polyenylcyclopropane carboxylic esters with high insecticidal activity

Polymer nanoparticles with electrostatically loaded multicargo for combined cancer phototherapy

Polymeric nanoparticles enhance the sonodynamic activity of meso-tetrakis (4-sulfonatophenyl) porphyrin in an in vitro neuroblastoma model

Polymethylmethacrylate nanoparticles as carrier of an oligodeoxynucleotide molecular beacon specific for survivin mRNA in A549 human lung adenocarcinoma epithelial cells

Quinazolinedione SIRT6 inhibitors sensitize cancer cells to chemotherapeutics

Rapid microwave-assisted deprotection of N-Cbz and N-Bn derivatives

SILK.IT project: Silk Italian Technology for industrial biomanufacturing

Selective sensitiveness of mesenchymal stem cells to shock waves leads to anticancer effect in human cancer cell co-cultures.

Semisynthesis, biological activity, and molecular modeling studies of C-ring-modified camptothecins.

Silk fibroin film from golden-yellow Bombyx mori is a biocomposite that contains lutein and promotes axonal growth of primary neurons

Silylcupration of acylimidazolides: a new synthesis of α-aminoacylsilanes and their synthetic applications

Species-dependent binding of new synthesized bicalutamide analogues to albumin by optical biosensor analysis

Stereoselective Three-Carbon and Two-Carbon Elongation of the Carbon Chain inN-Boc-Protected α-Aminoacylsilanes: An Entry to Functionalized β-Amino Alcohols and to Statine Analogues

Stereoselective one-pot synthesis of constrained N,O-orthogonally protected C-glycosyl norstatines [C(1')-aminoglycosyl-1,3-dioxolan-4-ones]

Structure-activity relationship study of 16 a-thiocamptothecins: an integrated in vitro and in silico approach

Sulfonates-PMMA nanoparticles conjugates: a versatile system for multimodal application

Synthesis and reactivity of achiral and of a novel planar chiral thioferrocenoylsilanes

Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs

Synthesis of Heterocycles Through Hydrosilylation, Silylformylation, Silylcarbocyclization and Cyclohydrocarbonylation Reactions

Synthesis of chiral β2,2,3-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-β-lactams by double asymmetric induction

Synthesis of deserpidine from reserpine

Synthesis of α2,2,β3-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates toN-(tert-Butylsulfinyl) Imines

TPPS supported on core–shell PMMA nanoparticles: the development of continuous-flow membrane-mediated electrocoagulation as a photocatalyst processing method in aqueous media

The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin−Polyamine Conjugates

The first synthesis of N,O-protected β2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding β-lactams

The role of polyamine architecture on the pharmacological activity of open lactone camptothecin-polyamine conjugates

Thiocamptothecin

Thiophene-based compounds as fluorescent tags to study mesenchymal stem cell uptake and release of taxanes.

Unprecedented Behavior of (9 R)-9-Hydroxystearic Acid-Loaded Keratin Nanoparticles on Cancer Cell Cycle

Wool Keratin 3D Scaffolds with Light-Triggered Antimicrobial Activity.