Lista de obras - François Marceau - Dominio Público Uruguay

A fluorescent version of the bradykinin B2 receptor antagonist B-9430: pharmacological characterization and use in live cell imaging

artículo científico publicado en 2008

A ligand-based approach to investigate the expression and function of angiotensin converting enzyme in intact human umbilical vein endothelial cells

artículo científico publicado en 2010

A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor

artículo científico publicado en 2003

A nonpeptide antagonist reveals a highly glycosylated state of the rabbit kinin B1 receptor.

artículo científico publicado en 2006

A novel nonpeptide antagonist of the kinin B1 receptor: effects at the rabbit receptor

artículo científico publicado en 2004

A possible common pharmacophore in the non-peptide antagonists of the bradykinin B1 receptor

scientific article published on 01 March 2005

A tagged parathyroid hormone derivative as a carrier of antibody cargoes transported by the G protein coupled PTH1 receptor.

artículo científico publicado en 2014

Absence of ligand-induced regulation of kinin receptor expression in the rabbit

artículo científico publicado en 2001

Abstracts from the 10th C1-inhibitor deficiency workshop.

artículo científico publicado en 2017

Advances in the development of bradykinin receptor ligands

artículo científico publicado en 2006

Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.

artículo científico publicado en 2002

Altered cardiac bradykinin metabolism in experimental diabetes caused by the variations of angiotensin-converting enzyme and other peptidases.

artículo científico publicado en 2010

Altered frequency of a promoter polymorphic allele of the kinin B1 receptor gene in inflammatory bowel disease

artículo científico publicado en 1998

Altered frequency of a promoter polymorphism of the kinin B2 receptor gene in hypertensive African-Americans.

artículo científico publicado en 2000

Aminopeptidase modulation of the pharmacological responses to synthetic thrombin receptor agonists

artículo científico publicado en 1994

An in vitro reconstitution system to address the mechanism of the vascular expression of the bradykinin B₁ receptor in response to angiotensin converting enzyme inhibition

scientific article published on 02 October 2011

Anaphylatoxin C5a fails to promote prostacyclin release in cultured endothelial cells from human umbilical veins

artículo científico publicado en 1986

Angiotensin converting enzyme inhibitor induced angio-oedema: a review of the pathophysiology and risk factors.

scientific article published on 29 July 2009

Antagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptors

artículo científico publicado en 2006

Assessment of cation trapping by cellular acidic compartments.

artículo científico publicado en 2014

Autophagic flux inhibition and lysosomogenesis ensuing cellular capture and retention of the cationic drug quinacrine in murine models

artículo científico publicado en 2015

B-9972 (D-Arg-[Hyp3,Igl5,Oic7,Igl8]-bradykinin) is an inactivation-resistant agonist of the bradykinin B2 receptor derived from the peptide antagonist B-9430 (D-Arg-[Hyp3,Igl5,D-Igl7,Oic8]-bradykinin): pharmacologic profile and effective induction o

artículo científico publicado en 2007

Bacitracin U.S.P. contains a factor that stimulates receptors for 5-hydroxytryptamine on rabbit aortic strips

artículo científico publicado en 1990

Bifunctional epitope-agonist ligands of the bradykinin B(2) receptor

artículo científico publicado en 2013

Bifunctional fusion proteins containing the sequence of the bradykinin homologue maximakinin: activities at the rat bradykinin B₂ receptor

artículo científico publicado en 2018

Bifunctional ligands of the bradykinin B2 and B1 receptors: An exercise in peptide hormone plasticity

artículo científico publicado en 2018

Biotechnological Fluorescent Ligands of the Bradykinin B1 Receptor: Protein Ligands for a Peptide Receptor

artículo científico publicado en 2016

Bradykinin B2 receptor gene polymorphism is associated with altered urinary albumin/creatinine values in diabetic patients.

artículo científico publicado en 2002

Bradykinin B₂ receptor-mediated transport into intact cells: anti-receptor antibody-based cargoes

artículo científico publicado en 2011

Bradykinin forming capacity of oversulfated chondroitin sulfate contaminated heparin in vitro

artículo científico publicado en 2010

Bradykinin receptor ligands: therapeutic perspectives

artículo científico publicado en 2004

Bradykinin receptors: Agonists, antagonists, expression, signaling, and adaptation to sustained stimulation

artículo científico publicado en 2020

C-C chemokine receptor-7 mediated endocytosis of antibody cargoes into intact cells

artículo científico publicado en 2013

Carboxypeptidase N (kininase I) activity in blood and synovial fluid from patients with arthritis

artículo científico publicado en 1987

Cardiovascular expression of inflammatory signaling molecules, the kinin B1 receptor and COX2, in the rabbit: effects of LPS, anti-inflammatory and anti-hypertensive drugs

artículo científico publicado en 2007

Cation trapping by cellular acidic compartments: beyond the concept of lysosomotropic drugs

artículo científico publicado en 2011

Characterization of a fluorescent conjugate of the rabbit angiotensin AT(1) receptor.

artículo científico publicado en 2003

Characterization of a polymorphism in the coding region of the human C5a anaphylatoxin receptor

artículo científico publicado en 1999

Cloning and preliminary pharmacological characterization of the anaphylatoxin C5a receptor in the rabbit.

artículo científico publicado en 1999

Comparing Pathways of Bradykinin Formation in Whole Blood From Healthy Volunteers and Patients With Hereditary Angioedema Due to C1 Inhibitor Deficiency

Comparison of two classes of non-peptide drugs as antagonists of neutrophil receptors for f-Met-Leu-Phe. Pyrazolons and iodinated radiographic contrast agents

artículo científico publicado el 4 de febrero de 1992

Contractile effect of anaphylatoxin C5a and of a mimetic peptide on the human umbilical artery: further evidence for leukocyte-dependent vasomotion

artículo científico publicado en 2002

D-Arg0-Bradykinin-Arg-Arg, a Latent Vasoactive Bradykinin B2 Receptor Agonist Metabolically Activated by Carboxypeptidases

artículo científico publicado en 2018

Design of fluorescent bradykinin analogs: application to imaging of B2 receptor-mediated agonist endocytosis and trafficking and angiotensin-converting enzyme

artículo científico publicado en 2011

Development of a binding assay for the B1 receptors for kinins

artículo científico publicado en 1995

Discovery of a dual-function peptide that combines aminopeptidase N inhibition and kinin B1 receptor antagonism

artículo científico publicado en 2005

Dissociation of the vacuolar and macroautophagic cytopathology from the cytotoxicity induced by the lipophilic local anesthetic bupivacaine

artículo científico publicado en 2011

Do angiotensin-converting enzyme inhibitors directly stimulate the kinin B1 receptor?

artículo científico publicado en 2003

Does zaltoprofen antagonize the bradykinin receptors?

artículo científico publicado en 2007

Down-regulation of interleukin-1beta production and PGE2 accumulation by an indomethacin-phenylalanine derivative in human monocytes

artículo científico publicado en 1998

Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists

artículo científico publicado en 2006

Editorial: Correspondence from Chirumbolo and Bjorklund.

artículo científico publicado en 2018

Editorial: Improving the data reproducibility and general interest of natural product submissions

artículo científico publicado en 2015

Effect of interferon-γ on inflammatory cytokine-induced bradykinin B1 receptor expression in human vascular cells.

artículo científico publicado en 2010

Effects of experimental conditions on the production of interleukin-1 alpha and -1 beta by human endothelial cells cultured in vitro

artículo científico publicado el 1 de mayo de 1992

Effects of inactivation-resistant agonists on the signalling, desensitization and down-regulation of bradykinin B(2) receptors.

artículo científico publicado en 2009

Effects of low molecular weight fibrin degradation products 6A and 6D on rabbit aorta strips

artículo científico publicado en 1987

Endogenous aminopeptidase N decreases the potency of peptide agonists and antagonists of the kinin B1 receptors in the rabbit aorta

artículo científico publicado en 2005

Epidermal growth factor-induced rapid relaxation of the isolated rabbit mesenteric artery

artículo científico publicado en 1994

Evidence for vascular tone regulation by resident or infiltrating leukocytes.

artículo científico publicado en 1996

Expression of kinin B(1) receptor in fresh or cultured rabbit aortic smooth muscle: role of NF-kappa B.

artículo científico publicado en 2002

Expression of metallopeptidases and kinin receptors in swine oropharyngeal tissues: effects of angiotensin I-converting enzyme inhibition and inflammation.

artículo científico publicado en 2005

Fluorescent ligands of the bradykinin B1 receptors: pharmacologic characterization and application to the study of agonist-induced receptor translocation and cell surface receptor expression.

artículo científico publicado en 2009

Further analysis of the upregulation of bradykinin B1 receptors in isolated rabbit aorta by using metabolic inhibitors

artículo científico publicado en 1994

Generation of kinins during preparation and storage of whole blood-derived platelet concentrates

artículo científico publicado en 2007

Green fluorescent protein fused to peptide agonists of two dissimilar G protein-coupled receptors: novel ligands of the bradykinin B2 (rhodopsin family) receptor and parathyroid hormone PTH1 (secretin family) receptor

artículo científico publicado en 2013

Guest editorial for the special issue peptide receptors: focus on neuropeptides and kinins

scientific article published on 20 October 2009

High affinity capture and concentration of quinacrine in polymorphonuclear neutrophils via vacuolar ATPase-mediated ion trapping: comparison with other peripheral blood leukocytes and implications for the distribution of cationic drugs

artículo científico publicado en 2013

High agonist-independent clearance of rabbit kinin B1 receptors in cultured cells.

artículo científico publicado en 2003

Human kallikrein hK2 has low kininogenase activity while prostate-specific antigen (hK3) has none

artículo científico publicado en 1997

In Vitro Modeling of Bradykinin-Mediated Angioedema States

artículo científico publicado en 2020

In Vitro Pharmacological Profile of a New Small Molecule Bradykinin B2 Receptor Antagonist

artículo científico publicado en 2020

In Vivo Effects of Bradykinin B2 Receptor Agonists with Varying Susceptibility to Peptidases.

artículo científico publicado en 2015

Increased fibrinolysis-induced bradykinin formation in hereditary angioedema confirmed using stored plasma and biotechnological inhibitors

artículo científico publicado en 2019

Induction of beta 1-receptors for kinins in the rabbit by a bacterial lipopolysaccharide

artículo científico publicado en 1981

Inflammatory hyperalgesia induced by zymosan in the plantar tissue of the rat: effect of kinin receptor antagonists

scientific article published on 01 February 2000

Infrared-emitting, peptidase-resistant fluorescent ligands of the bradykinin B2 receptor: application to cytofluorometry and imaging

artículo científico publicado en 2016

Inhibition of human and rabbit arterial smooth muscle cell migration mediated by the kinin B1 receptor: role of receptor density and released mediators

artículo científico publicado en 2006

Inhibitory effects of cytoskeleton disrupting drugs and GDP-locked Rab mutants on bradykinin B₂ receptor cycling

artículo científico publicado en 2013

Intense pseudotransport of a cationic drug mediated by vacuolar ATPase: procainamide-induced autophagic cell vacuolization

artículo científico publicado en 2008

International union of pharmacology. XLV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences

artículo científico publicado en 2005

Intracellular sequestration of amiodarone: role of vacuolar ATPase and macroautophagic transition of the resulting vacuolar cytopathology.

artículo científico publicado en 2009

Introduction: Natural product-based drug discovery in Immunopharmacology.

artículo científico publicado en 2016

Kinin B1 receptors: a review.

artículo científico publicado en 1995

Kinin receptors

artículo científico publicado en 1998

Kinin receptors: functional aspects.

artículo científico publicado en 2002

Kininases and vascular responses to kinins

artículo científico publicado en 1982

Lack of direct interaction between enalaprilat and the kinin B1 receptors

artículo científico publicado en 2007

Ligand-mediated regulation of kinin receptors in the rabbit.

artículo científico publicado en 2001

Long-term culture and characterization of human limbal microvascular endothelial cells

artículo científico publicado en 1990

Loss of function of vascular smooth muscle cells by nitric oxide-dependent and -independent interactions with tumorigenic cells

artículo científico publicado en 2004

Lysosomotropic cationic drugs induce cytostatic and cytotoxic effects: Role of liposolubility and autophagic flux and antagonism by cholesterol ablation.

artículo científico publicado en 2016

Massive cell vacuolization induced by organic amines such as procainamide.

artículo científico publicado en 2004

Measurement of Bradykinin Formation and Degradation in Blood Plasma: Relevance for Acquired Angioedema Associated With Angiotensin Converting Enzyme Inhibition and for Hereditary Angioedema Due to Factor XII or Plasminogen Gene Variants

artículo científico publicado en 2020

Mechanism of the contractile effect of diaspirin-cross-linked hemoglobin in rat isolated aorta strip denuded of endothelium as revealed using an oil-immersion procedure

scientific article published on 01 October 1996

Met-Lys-bradykinin-Ser-Ser, a peptide produced by the neutrophil from kininogen, is metabolically activated by angiotensin converting enzyme in vascular tissue

artículo científico publicado en 2011

Mitogenic effect of bradykinin and of des-Arg9-bradykinin on cultured fibroblasts.

artículo científico publicado en 1986

Molecular identification and pharmacological profile of the bovine kinin B1 receptor

artículo científico publicado en 2006

N-substituted 4-aminobenzamides (procainamide analogs): an assessment of multiple cellular effects concerning ion trapping

artículo científico publicado en 2005

N-terminal extended conjugates of the agonists and antagonists of both bradykinin receptor subtypes: structure-activity relationship, cell imaging using ligands conjugated with fluorophores and prospect for functionally active cargoes.

artículo científico

NLRP3 promotes autophagy of urate crystals phagocytized by human osteoblasts.

artículo científico publicado en 2013

NTPDase1 (CD39) controls nucleotide-dependent vasoconstriction in mouse.

artículo científico publicado en 2010

Non-competitive pharmacological antagonism at the rabbit B(1) receptor.

artículo científico publicado en 2000

Pharmacological effects of recombinant human tissue kallikrein on bradykinin B2 receptors

artículo científico publicado en 2015

Pharmacological evidence of bradykinin regeneration from extended sequences that behave as peptidase-activated B2 receptor agonists.

artículo científico publicado en 2014

Pharmacological modulation of interleukin 1 production by cultured endothelial cells from human umbilical veins ⬇️

artículo científico publicado el 1 de marzo de 1990

Pharmacological modulation of the up-regulated responses to des-Arg9-bradykinin in vivo and in vitro

artículo científico publicado en 1989

Pharmacological profile of a bifunctional ligand of the formyl peptide receptor1 fused to the myc epitope.

artículo científico publicado en 2015

Pharmacology of kinins: Their relevance to tissue injury and inflammation ⬇️

artículo científico publicado el 1 de enero de 1983

Production and evaluation of parathyroid hormone receptor1 ligands with intrinsic or assembled peroxidase domains

artículo científico publicado en 2017

Prolonged signalling and trafficking of the bradykinin B2 receptor stimulated with the amphibian peptide maximakinin: insight into the endosomal inactivation of kinins

artículo científico publicado en 2011

Quantification of des-Arg9-bradykinin using a chemiluminescence enzyme immunoassay: application to its kinetic profile during plasma activation

scientific article published on 01 March 1995

Rapid assay of human plasma carboxypeptidase N by high-performance liquid chromatographic separation of hippuryl-lysine and its product

artículo científico publicado en 1983

Receptor tyrosine kinases as mediators of injury-induced bradykinin B1 receptor expression in rabbit aortic smooth muscle.

artículo científico publicado en 2009

Receptor-independent, vacuolar ATPase-mediated cellular uptake of histamine receptor-1 ligands: possible origin of pharmacological distortions and side effects

artículo científico publicado en 2008

Recombinant Human Hemoglobin (rHb1.1) Selectively Inhibits Vasorelaxation Elicited by Nitric Oxide Donors in Rabbit Isolated Aortic Rings ⬇️

artículo científico publicado el 1 de abril de 1995

Reprint of: Editorial: Correspondence from Chirumbolo and Bjorklund

scientific article published on 07 July 2018

Role of nuclear factor-kappaB and protein kinase C signaling in the expression of the kinin B1 receptor in human vascular smooth muscle cells

artículo científico publicado en 2006

S100A9 potentiates the activation of neutrophils by the etiological agent of gout, monosodium urate crystals.

artículo científico publicado en 2017

Selective induction of cardiovascular responses to des-Arg9-bradykinin by bacterial endotoxin

artículo científico publicado en 1984

Species-specific pharmacology of maximakinin, an amphibian homologue of bradykinin: putative prodrug activity at the human B2 receptor and peptidase resistance in rats

artículo científico publicado en 2017

Structural modification of the highly potent peptide bradykinin B1 receptor antagonist B9958.

artículo científico publicado en 2007

Studies on rabbit natural and recombinant tissue factors: intracellular retention and regulation of surface expression in cultured cells

artículo científico publicado en 2005

Synthetic C5a receptor agonists. Pharmacology, metabolism and in vivo cardiovascular and hematologic effects

artículo científico publicado en 1993

The Development of a Targeted and More Potent, Anti-Inflammatory Derivative of Colchicine: Implications for Gout

artículo científico publicado en 2020

The ability of des-Arg9-bradykinin to relax rabbit isolated mesenteric arteries is acquired during in vitro incubation

scientific article published on 01 October 1987

The antiwrinkle effect of topical concentrated 2-dimethylaminoethanol involves a vacuolar cytopathology

artículo científico publicado en 2007

The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors

artículo científico publicado en 2006

The isolated human umbilical vein as a bioassay for kinin-generating proteases: An in vitro model for therapeutic angioedema agents

artículo científico publicado en 2016

The kallikrein-kinin system: current and future pharmacological targets.

artículo científico publicado en 2005

The kallikrein-kininogen-kinin system: lessons from the quantification of endogenous kinins.

artículo científico publicado en 2000

The kinin B<SUB>1 </SUB>receptor: an inducible G protein coupled receptor

artículo científico publicado el 1 de junio de 1997

Tissue kallikrein actions at the rabbit natural or recombinant kinin B2 receptors.

artículo científico publicado en 2003

Trapping of adrenergic decongestant drugs into cellular endomembrane compartments: toxicological and pharmacological consequences

artículo científico publicado en 2007

Tumor cells expressing tissue factor influence the migration of smooth muscle cells in a catalytic activity-dependent way.

artículo científico publicado en 2009

Vacuolar ATPase-mediated cellular concentration and retention of quinacrine: a model for the distribution of lipophilic cationic drugs to autophagic vacuoles

artículo científico publicado en 2009

Vacuolar ATPase-mediated sequestration of local anesthetics in swollen macroautophagosomes.

artículo científico publicado en 2010

Vascular smooth muscle contractility assays for inflammatory and immunological mediators

artículo científico publicado en 2010

Vasopeptidase-activated latent ligands of the histamine receptor-1.

artículo científico publicado en 2013

Wortmannin alters the intracellular trafficking of the bradykinin B2 receptor: role of phosphoinositide 3-kinase and Rab5.

artículo científico publicado en 2003

[Anti-wrinkle properties of amines: vacuolar cytopathology mediated by the V-ATPase]

scientific article published on 01 June 2007

Lista de obras de François Marceau

A fluorescent version of the bradykinin B2 receptor antagonist B-9430: pharmacological characterization and use in live cell imaging

A ligand-based approach to investigate the expression and function of angiotensin converting enzyme in intact human umbilical vein endothelial cells

A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor

A nonpeptide antagonist reveals a highly glycosylated state of the rabbit kinin B1 receptor.

A novel nonpeptide antagonist of the kinin B1 receptor: effects at the rabbit receptor

A possible common pharmacophore in the non-peptide antagonists of the bradykinin B1 receptor

A tagged parathyroid hormone derivative as a carrier of antibody cargoes transported by the G protein coupled PTH1 receptor.

Absence of ligand-induced regulation of kinin receptor expression in the rabbit

Abstracts from the 10th C1-inhibitor deficiency workshop.

Advances in the development of bradykinin receptor ligands

Agonist-induced translocation of the kinin B(1) receptor to caveolae-related rafts.

Altered cardiac bradykinin metabolism in experimental diabetes caused by the variations of angiotensin-converting enzyme and other peptidases.

Altered frequency of a promoter polymorphic allele of the kinin B1 receptor gene in inflammatory bowel disease

Altered frequency of a promoter polymorphism of the kinin B2 receptor gene in hypertensive African-Americans.

Aminopeptidase modulation of the pharmacological responses to synthetic thrombin receptor agonists

An in vitro reconstitution system to address the mechanism of the vascular expression of the bradykinin B₁ receptor in response to angiotensin converting enzyme inhibition

Anaphylatoxin C5a fails to promote prostacyclin release in cultured endothelial cells from human umbilical veins

Angiotensin converting enzyme inhibitor induced angio-oedema: a review of the pathophysiology and risk factors.

Antagonist, partial agonist and antiproliferative actions of B-9870 (CU201) as a function of the expression and density of the bradykinin B1 and B2 receptors

Assessment of cation trapping by cellular acidic compartments.

Autophagic flux inhibition and lysosomogenesis ensuing cellular capture and retention of the cationic drug quinacrine in murine models

B-9972 (D-Arg-[Hyp3,Igl5,Oic7,Igl8]-bradykinin) is an inactivation-resistant agonist of the bradykinin B2 receptor derived from the peptide antagonist B-9430 (D-Arg-[Hyp3,Igl5,D-Igl7,Oic8]-bradykinin): pharmacologic profile and effective induction o

Bacitracin U.S.P. contains a factor that stimulates receptors for 5-hydroxytryptamine on rabbit aortic strips

Bifunctional epitope-agonist ligands of the bradykinin B(2) receptor

Bifunctional fusion proteins containing the sequence of the bradykinin homologue maximakinin: activities at the rat bradykinin B₂ receptor

Bifunctional ligands of the bradykinin B2 and B1 receptors: An exercise in peptide hormone plasticity

Biotechnological Fluorescent Ligands of the Bradykinin B1 Receptor: Protein Ligands for a Peptide Receptor

Bradykinin B2 receptor gene polymorphism is associated with altered urinary albumin/creatinine values in diabetic patients.

Bradykinin B₂ receptor-mediated transport into intact cells: anti-receptor antibody-based cargoes

Bradykinin forming capacity of oversulfated chondroitin sulfate contaminated heparin in vitro

Bradykinin receptor ligands: therapeutic perspectives

Bradykinin receptors: Agonists, antagonists, expression, signaling, and adaptation to sustained stimulation

C-C chemokine receptor-7 mediated endocytosis of antibody cargoes into intact cells

Carboxypeptidase N (kininase I) activity in blood and synovial fluid from patients with arthritis

Cardiovascular expression of inflammatory signaling molecules, the kinin B1 receptor and COX2, in the rabbit: effects of LPS, anti-inflammatory and anti-hypertensive drugs

Cation trapping by cellular acidic compartments: beyond the concept of lysosomotropic drugs

Characterization of a fluorescent conjugate of the rabbit angiotensin AT(1) receptor.

Characterization of a polymorphism in the coding region of the human C5a anaphylatoxin receptor

Cloning and preliminary pharmacological characterization of the anaphylatoxin C5a receptor in the rabbit.

Comparing Pathways of Bradykinin Formation in Whole Blood From Healthy Volunteers and Patients With Hereditary Angioedema Due to C1 Inhibitor Deficiency

Comparison of two classes of non-peptide drugs as antagonists of neutrophil receptors for f-Met-Leu-Phe. Pyrazolons and iodinated radiographic contrast agents

Contractile effect of anaphylatoxin C5a and of a mimetic peptide on the human umbilical artery: further evidence for leukocyte-dependent vasomotion

D-Arg0-Bradykinin-Arg-Arg, a Latent Vasoactive Bradykinin B2 Receptor Agonist Metabolically Activated by Carboxypeptidases

Design of fluorescent bradykinin analogs: application to imaging of B2 receptor-mediated agonist endocytosis and trafficking and angiotensin-converting enzyme

Development of a binding assay for the B1 receptors for kinins

Discovery of a dual-function peptide that combines aminopeptidase N inhibition and kinin B1 receptor antagonism

Dissociation of the vacuolar and macroautophagic cytopathology from the cytotoxicity induced by the lipophilic local anesthetic bupivacaine

Do angiotensin-converting enzyme inhibitors directly stimulate the kinin B1 receptor?

Does zaltoprofen antagonize the bradykinin receptors?

Down-regulation of interleukin-1beta production and PGE2 accumulation by an indomethacin-phenylalanine derivative in human monocytes

Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists

Editorial: Correspondence from Chirumbolo and Bjorklund.

Editorial: Improving the data reproducibility and general interest of natural product submissions

Effect of interferon-γ on inflammatory cytokine-induced bradykinin B1 receptor expression in human vascular cells.

Effects of experimental conditions on the production of interleukin-1 alpha and -1 beta by human endothelial cells cultured in vitro

Effects of inactivation-resistant agonists on the signalling, desensitization and down-regulation of bradykinin B(2) receptors.

Effects of low molecular weight fibrin degradation products 6A and 6D on rabbit aorta strips

Endogenous aminopeptidase N decreases the potency of peptide agonists and antagonists of the kinin B1 receptors in the rabbit aorta

Epidermal growth factor-induced rapid relaxation of the isolated rabbit mesenteric artery

Evidence for vascular tone regulation by resident or infiltrating leukocytes.

Expression of kinin B(1) receptor in fresh or cultured rabbit aortic smooth muscle: role of NF-kappa B.

Expression of metallopeptidases and kinin receptors in swine oropharyngeal tissues: effects of angiotensin I-converting enzyme inhibition and inflammation.

Fluorescent ligands of the bradykinin B1 receptors: pharmacologic characterization and application to the study of agonist-induced receptor translocation and cell surface receptor expression.

Further analysis of the upregulation of bradykinin B1 receptors in isolated rabbit aorta by using metabolic inhibitors

Generation of kinins during preparation and storage of whole blood-derived platelet concentrates

Green fluorescent protein fused to peptide agonists of two dissimilar G protein-coupled receptors: novel ligands of the bradykinin B2 (rhodopsin family) receptor and parathyroid hormone PTH1 (secretin family) receptor

Guest editorial for the special issue peptide receptors: focus on neuropeptides and kinins

High affinity capture and concentration of quinacrine in polymorphonuclear neutrophils via vacuolar ATPase-mediated ion trapping: comparison with other peripheral blood leukocytes and implications for the distribution of cationic drugs

High agonist-independent clearance of rabbit kinin B1 receptors in cultured cells.

Human kallikrein hK2 has low kininogenase activity while prostate-specific antigen (hK3) has none

In Vitro Modeling of Bradykinin-Mediated Angioedema States

In Vitro Pharmacological Profile of a New Small Molecule Bradykinin B2 Receptor Antagonist

In Vivo Effects of Bradykinin B2 Receptor Agonists with Varying Susceptibility to Peptidases.

Increased fibrinolysis-induced bradykinin formation in hereditary angioedema confirmed using stored plasma and biotechnological inhibitors

Induction of beta 1-receptors for kinins in the rabbit by a bacterial lipopolysaccharide

Inflammatory hyperalgesia induced by zymosan in the plantar tissue of the rat: effect of kinin receptor antagonists

Infrared-emitting, peptidase-resistant fluorescent ligands of the bradykinin B2 receptor: application to cytofluorometry and imaging

Inhibition of human and rabbit arterial smooth muscle cell migration mediated by the kinin B1 receptor: role of receptor density and released mediators

Inhibitory effects of cytoskeleton disrupting drugs and GDP-locked Rab mutants on bradykinin B₂ receptor cycling

The kinin B<SUB>1 </SUB>receptor: an inducible G protein coupled receptor