Lista de obras - Joan Bosch - Dominio Público Uruguay

'Click' synthesis of a triazole-based inhibitor of Met functions in cancer cells.

artículo científico publicado en 2012

A Straightforward Synthesis of Functionalized -Perhydroisoquinolin-1-ones

artículo científico publicado en 2019

A biomimetic enantioselective approach to the decahydroquinoline class of dendrobatid alkaloids

artículo científico publicado en 2008

A general synthetic route to enantiopure 5-substituted cis-decahydroquinolines

artículo científico publicado en 2009

A practical synthetic route to enantiopure 6-substituted cis-decahydroquinolines

scientific article published on 01 December 2011

A synthetic approach to ervatamine-silicine alkaloids. Enantioselective total synthesis of (-)-16-episilicine.

artículo científico publicado en 2010

A synthetic route to a novel type of conformationally constrained N-aryloxazolidinones

artículo científico publicado en 2005

Access to Enantiopure 5-, 7-, and 5,7-Substituted cis-Decahydroquinolines: Enantioselective Synthesis of (-)-Cermizine B

artículo científico publicado en 2017

Access to Enantiopure Advanced Intermediates en Route to Madangamines

artículo científico publicado en 2019

Access to enantiopure 4-substituted 1,5-aminoalcohols from phenylglycinol-derived δ-lactams: synthesis of Haliclona alkaloids

artículo científico publicado en 2014

Alkylation of phenylglycinol-derived oxazolopiperidone lactams. Enantioselective synthesis of beta-substituted piperidines

artículo científico publicado en 2006

An enantioselective entry to cis-perhydroisoquinolines

scientific article published on 01 August 2005

An enantioselective synthetic route to cis-2,4-disubstituted and 2,4-bridged piperidines

artículo científico publicado en 2008

An unexpected oxidation in the generation of cyclopenta[c]piperidines by ring-closing metathesis

artículo científico publicado en 2009

Biogenetically inspired enantioselective approach to Indolo[2,3-a]- and benzo[a]quinolizidine alkaloids from a synthetic equivalent of secologanin

scientific article published on 01 July 2005

Biomimetic construction of the hydroquinoline ring system. Diastereodivergent enantioselective synthesis of 2,5-disubstituted cis-decahydroquinolines.

artículo científico publicado en 2010

Combined drug action of 2-phenylimidazo[2,1-b]benzothiazole derivatives on cancer cells according to their oncogenic molecular signatures

artículo científico publicado en 2012

Conjugate addition of organocuprates to chiral bicyclic delta-lactams. Enantioselective synthesis of cis-3,4-disubstituted and 3,4,5-trisubstituted piperidines.

artículo científico publicado en 2001

Conjugate additions to phenylglycinol-derived unsaturated delta-lactams. Enantioselective synthesis of uleine alkaloids.

artículo científico publicado en 2004

Diels–Alder Reactions of 5,6-Dihydro-2(1H)-pyridones

Dynamic kinetic resolution and desymmetrization of enantiotopic groups by cyclodehydration of racemic or prochiral delta-oxoesters with (R)-phenylglycinol: enantioselective synthesis of piperidines.

artículo científico publicado en 2002

Dynamic kinetic resolution and desymmetrization processes: a straightforward methodology for the enantioselective synthesis of piperidines

artículo científico publicado en 2006

Electrophilic Oxidative Additions upon 1,4-Dihydropyridines

artículo científico publicado en 1998

Enantio- and diastereoconvergent cyclocondensation reactions: synthesis of enantiopure cis-decahydroquinolines

scientific article published on 02 October 2013

Enantioselective Synthesis of Spiro[indolizidine-1,3'-oxindoles].

artículo científico publicado en 2017

Enantioselective Synthesis of the Ethyl Analog of the Marine Alkaloid Haliclorensin C

scientific article published on 18 March 2019

Enantioselective Total Synthesis of (+)-Gephyrotoxin 287C.

artículo científico publicado en 2017

Enantioselective Total Synthesis of Fluvirucinin B1.

artículo científico publicado en 2016

Enantioselective formal synthesis of (+)-dihydrocorynantheine and (-)-dihydrocorynantheol.

artículo científico publicado en 2009

Enantioselective formal synthesis of (+)-madangamine A

scientific article published on 05 June 2019

Enantioselective formal synthesis of ent-rhynchophylline and ent-isorhynchophylline

artículo científico publicado en 2013

Enantioselective formal synthesis of the marine macrolide (-)-callyspongiolide

scientific article published on 16 April 2020

Enantioselective spirocyclizations from tryptophanol-derived oxazolopiperidone lactams

scientific article published on 29 June 2007

Enantioselective synthesis of 2-arylpiperidines from chiral lactams. A concise synthesis of (-)-anabasine.

artículo científico publicado en 2002

Enantioselective synthesis of 3,3-disubstituted piperidine derivatives by enolate dialkylation of phenylglycinol-derived oxazolopiperidone lactams

scientific article published on 09 May 2007

Enantioselective synthesis of cis- and trans-3,5-disubstituted piperidines. Synthesis of 20S- and 20R-dihydrocleavamine

scientific article published on 01 August 2003

Enantioselective synthesis of lepadins A-D from a phenylglycinol-derived hydroquinolone lactam

artículo científico publicado en 2015

Enantioselective synthesis of piperidine, indolizidine, and quinolizidine alkaloids from a phenylglycinol-derived delta-lactam.

artículo científico publicado en 2003

Enantioselective total synthesis of Wieland-Gumlich aldehyde and (-)-strychnine

scientific article published on 01 February 2000

Enantioselective total synthesis of the indole alkaloid 16-episilicine.

artículo científico publicado en 2009

Enantioselective, protecting group-free synthesis of 1S-ethyl-4-substituted quinolizidines

artículo científico publicado en 2012

First asymmetric cascade reaction catalysed by chiral primary aminoalcohols

artículo científico publicado en 2011

First enantioselective synthesis of tetracyclic intermediates en route to madangamine D

artículo científico publicado en 2013

First enantioselective synthesis of the diazatricyclic core of madangamine alkaloids

artículo científico publicado en 2010

Generation and Intermolecular Reactions of 2-Indolylacyl Radicals

artículo científico publicado en 2001

Generation and intermolecular reactions of 3-indolylacyl radicals

artículo científico publicado en 2002

Highly enantioselective dynamic kinetic resolution and desymmetrization processes by cyclocondensation of chiral aminoalcohols with racemic or prochiral delta-oxoacid derivatives

artículo científico publicado en 2005

Highly stereoselective double (R)-phenylglycinol-induced cyclocondensation reactions of symmetric aryl bis(oxoacids)

artículo científico publicado en 2011

Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling ⬇️

artículo científico publicado el 4 de noviembre de 2011

Model studies on the synthesis of madangamine alkaloids. Assembly of the macrocyclic rings

artículo científico publicado en 2012

New cascade 2-indolylacyl radical addition-cyclization reactions

artículo científico publicado en 2001

New potential antibacterials: a synthetic route to N-aryloxazolidinone/3-aryltetrahydroisoquinoline hybrids

artículo científico publicado en 2005

On the Origin of the Stereoselectivity in the Alkylation of Oxazolopiperidone Enolates

artículo científico publicado en 2006

Oxidative diphosphonylation of 1,4-dihydropyridines and pyridinium salts

artículo científico publicado en 2000

Palladium(0)-Catalyzed Heteroarylation of 2- and 3-Indolylzinc Derivatives. An Efficient General Method for the Preparation of (2-Pyridyl)indoles and Their Application to Indole Alkaloid Synthesis

scientific article published on 01 May 1997

Preparation and double Michael addition reactions of a synthetic equivalent of the Nazarov reagent

artículo científico publicado en 2013

Stereocontrolled Access to Enantiopure 7-Substituted cis- and trans-Octahydroindoles.

artículo científico publicado en 2016

Stereocontrolled Annulations of Indolo[2,3-a]quinolizidine-Derived Lactams with a Silylated Nazarov Reagent: Access to Allo and Epiallo Yohimbine-Type Derivatives

scientific article published on 01 September 2015

Stereodivergent synthesis of enantiopure cis- and trans-3-Ethyl-4-piperidineacetates

artículo científico publicado en 2002

Stereoselective conjugate addition reactions to phenylglycinol-derived, unsaturated oxazolopiperidone lactams

artículo científico publicado en 2011

Stereoselective syntheses of the antihistaminic drug olopatadine and its E-isomer

artículo científico publicado en 2012

Stereoselective synthesis of (-)-lepadins A-C.

artículo científico publicado en 2013

Stereoselective total synthesis of the putative structure of nitraraine

artículo científico publicado en 2014

Straightforward Methodology for the Enantioselective Synthesis of Benzo[a]- and Indolo[2,3-a]quinolizidines

artículo científico publicado en 2007

Structure-directed reversion in the pi-facial stereoselective alkylation of chiral bicyclic lactams.

artículo científico publicado en 2008

Studies on the Configurational Stability of 3-(2-Piperidyl)indoles

artículo científico publicado en 1996

Studies on the Synthesis of Phlegmarine-Type Lycopodium Alkaloids: Enantioselective Synthesis of (-)-Cermizine B, (+)-Serratezomine E, and (+)-Luciduline

artículo científico publicado en 2018

Synthesis and biological evaluation of 1,3,4-triaryl-3-pyrrolin-2-ones, a new class of selective cyclooxygenase-2 inhibitors

artículo científico publicado en 2000

Synthesis and dopaminergic activity of heterocyclic analogues of 5,6-dihydroxy-2-aminotetralins

scientific article published on 01 March 2000

Synthesis of water-soluble phenytoin prodrugs

scientific article published on 01 July 1999

Synthetic route to 6-functionalized 2-azabicyclo[3.3.1]nonanes

Total Synthesis of (-)-Strychnine via the Wieland-Gumlich Aldehyde

artículo científico publicado en 1999

Total synthesis of (+)-madangamine D

scientific article published on 02 May 2014

Unprecedented oxidation of a phenylglycinol-derived 2-pyridone: enantioselective synthesis of polyhydroxypiperidines

artículo científico publicado en 2001

Unusual oxidative bond-forming reactions upon 1,4-dihydropyridines: manganese(III)-promoted, single- and double-malonate additions

artículo científico publicado en 2001

Lista de obras de Joan Bosch

'Click' synthesis of a triazole-based inhibitor of Met functions in cancer cells.

A Straightforward Synthesis of Functionalized -Perhydroisoquinolin-1-ones

A biomimetic enantioselective approach to the decahydroquinoline class of dendrobatid alkaloids

A general synthetic route to enantiopure 5-substituted cis-decahydroquinolines

A practical synthetic route to enantiopure 6-substituted cis-decahydroquinolines

A synthetic approach to ervatamine-silicine alkaloids. Enantioselective total synthesis of (-)-16-episilicine.

A synthetic route to a novel type of conformationally constrained N-aryloxazolidinones

Access to Enantiopure 5-, 7-, and 5,7-Substituted cis-Decahydroquinolines: Enantioselective Synthesis of (-)-Cermizine B

Access to Enantiopure Advanced Intermediates en Route to Madangamines

Access to enantiopure 4-substituted 1,5-aminoalcohols from phenylglycinol-derived δ-lactams: synthesis of Haliclona alkaloids

Alkylation of phenylglycinol-derived oxazolopiperidone lactams. Enantioselective synthesis of beta-substituted piperidines

An enantioselective entry to cis-perhydroisoquinolines

An enantioselective synthetic route to cis-2,4-disubstituted and 2,4-bridged piperidines

An unexpected oxidation in the generation of cyclopenta[c]piperidines by ring-closing metathesis

Biogenetically inspired enantioselective approach to Indolo[2,3-a]- and benzo[a]quinolizidine alkaloids from a synthetic equivalent of secologanin

Biomimetic construction of the hydroquinoline ring system. Diastereodivergent enantioselective synthesis of 2,5-disubstituted cis-decahydroquinolines.

Combined drug action of 2-phenylimidazo[2,1-b]benzothiazole derivatives on cancer cells according to their oncogenic molecular signatures

Conjugate addition of organocuprates to chiral bicyclic delta-lactams. Enantioselective synthesis of cis-3,4-disubstituted and 3,4,5-trisubstituted piperidines.

Conjugate additions to phenylglycinol-derived unsaturated delta-lactams. Enantioselective synthesis of uleine alkaloids.

Diels–Alder Reactions of 5,6-Dihydro-2(1H)-pyridones

Dynamic kinetic resolution and desymmetrization of enantiotopic groups by cyclodehydration of racemic or prochiral delta-oxoesters with (R)-phenylglycinol: enantioselective synthesis of piperidines.

Dynamic kinetic resolution and desymmetrization processes: a straightforward methodology for the enantioselective synthesis of piperidines

Electrophilic Oxidative Additions upon 1,4-Dihydropyridines

Enantio- and diastereoconvergent cyclocondensation reactions: synthesis of enantiopure cis-decahydroquinolines

Enantioselective Synthesis of Spiro[indolizidine-1,3'-oxindoles].

Enantioselective Synthesis of the Ethyl Analog of the Marine Alkaloid Haliclorensin C

Enantioselective Total Synthesis of (+)-Gephyrotoxin 287C.

Enantioselective Total Synthesis of Fluvirucinin B1.

Enantioselective formal synthesis of (+)-dihydrocorynantheine and (-)-dihydrocorynantheol.

Enantioselective formal synthesis of (+)-madangamine A

Enantioselective formal synthesis of ent-rhynchophylline and ent-isorhynchophylline

Enantioselective formal synthesis of the marine macrolide (-)-callyspongiolide

Enantioselective spirocyclizations from tryptophanol-derived oxazolopiperidone lactams

Enantioselective synthesis of 2-arylpiperidines from chiral lactams. A concise synthesis of (-)-anabasine.

Enantioselective synthesis of 3,3-disubstituted piperidine derivatives by enolate dialkylation of phenylglycinol-derived oxazolopiperidone lactams

Enantioselective synthesis of cis- and trans-3,5-disubstituted piperidines. Synthesis of 20S- and 20R-dihydrocleavamine

Enantioselective synthesis of lepadins A-D from a phenylglycinol-derived hydroquinolone lactam

Enantioselective synthesis of piperidine, indolizidine, and quinolizidine alkaloids from a phenylglycinol-derived delta-lactam.

Enantioselective total synthesis of Wieland-Gumlich aldehyde and (-)-strychnine

Enantioselective total synthesis of the indole alkaloid 16-episilicine.

Enantioselective, protecting group-free synthesis of 1S-ethyl-4-substituted quinolizidines

First asymmetric cascade reaction catalysed by chiral primary aminoalcohols

First enantioselective synthesis of tetracyclic intermediates en route to madangamine D

First enantioselective synthesis of the diazatricyclic core of madangamine alkaloids

Generation and Intermolecular Reactions of 2-Indolylacyl Radicals

Generation and intermolecular reactions of 3-indolylacyl radicals

Highly enantioselective dynamic kinetic resolution and desymmetrization processes by cyclocondensation of chiral aminoalcohols with racemic or prochiral delta-oxoacid derivatives

Highly stereoselective double (R)-phenylglycinol-induced cyclocondensation reactions of symmetric aryl bis(oxoacids)

Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling ⬇️

Model studies on the synthesis of madangamine alkaloids. Assembly of the macrocyclic rings

New cascade 2-indolylacyl radical addition-cyclization reactions

New potential antibacterials: a synthetic route to N-aryloxazolidinone/3-aryltetrahydroisoquinoline hybrids

On the Origin of the Stereoselectivity in the Alkylation of Oxazolopiperidone Enolates

Oxidative diphosphonylation of 1,4-dihydropyridines and pyridinium salts

Palladium(0)-Catalyzed Heteroarylation of 2- and 3-Indolylzinc Derivatives. An Efficient General Method for the Preparation of (2-Pyridyl)indoles and Their Application to Indole Alkaloid Synthesis

Preparation and double Michael addition reactions of a synthetic equivalent of the Nazarov reagent

Stereocontrolled Access to Enantiopure 7-Substituted cis- and trans-Octahydroindoles.

Stereocontrolled Annulations of Indolo[2,3-a]quinolizidine-Derived Lactams with a Silylated Nazarov Reagent: Access to Allo and Epiallo Yohimbine-Type Derivatives

Stereodivergent synthesis of enantiopure cis- and trans-3-Ethyl-4-piperidineacetates

Stereoselective conjugate addition reactions to phenylglycinol-derived, unsaturated oxazolopiperidone lactams

Stereoselective syntheses of the antihistaminic drug olopatadine and its E-isomer

Stereoselective synthesis of (-)-lepadins A-C.

Stereoselective total synthesis of the putative structure of nitraraine

Straightforward Methodology for the Enantioselective Synthesis of Benzo[a]- and Indolo[2,3-a]quinolizidines

Structure-directed reversion in the pi-facial stereoselective alkylation of chiral bicyclic lactams.

Studies on the Configurational Stability of 3-(2-Piperidyl)indoles

Studies on the Synthesis of Phlegmarine-Type Lycopodium Alkaloids: Enantioselective Synthesis of (-)-Cermizine B, (+)-Serratezomine E, and (+)-Luciduline

Synthesis and biological evaluation of 1,3,4-triaryl-3-pyrrolin-2-ones, a new class of selective cyclooxygenase-2 inhibitors

Synthesis and dopaminergic activity of heterocyclic analogues of 5,6-dihydroxy-2-aminotetralins

Synthesis of water-soluble phenytoin prodrugs

Synthetic route to 6-functionalized 2-azabicyclo[3.3.1]nonanes

Total Synthesis of (-)-Strychnine via the Wieland-Gumlich Aldehyde

Total synthesis of (+)-madangamine D

Unprecedented oxidation of a phenylglycinol-derived 2-pyridone: enantioselective synthesis of polyhydroxypiperidines

Unusual oxidative bond-forming reactions upon 1,4-dihydropyridines: manganese(III)-promoted, single- and double-malonate additions