Lista de obras - Ewa Tatarczyńska - Dominio Público Uruguay

1,2,3,4-tetrahydroisoquinoline derivatives: a new class of 5-HT1A receptor ligands

artículo científico publicado en 1999

1,4-Benzoxazin-3(4H)-one derivatives and related compounds as 5-HT1A and 5-HT2A receptor ligands; the effect of the terminal amide fragment on the 5-HT1A/5-HT2A affinity and functional activity.

artículo científico publicado en 1998

1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: synthesis, binding to serotonin (5-HT1A, 5-HT2A, 5-HT7), alpha1-adrenergic, and dopaminergic D2 receptors, and in vivo 5-HT1A functional characteristics

artículo científico publicado en 2005

1-Pyridyl-3,4-dihydro-beta-carbolines: synthesis and central action.

artículo científico publicado en 1986

2-H- and 2-acyl-9- [omega-[4-(2-methoxyphenyl)piperazinyl]-alkyl]-1,2,3,4-tetrahydro-beta-carbolines as ligands of 5-HT1A and 5-HT2A receptors.

artículo científico publicado en 2001

5-HT1A and 5-HT2A receptor affinity and functional profile of some N-[3-(4-aryl-1-piperazinyl)propyl] derivatives of indolin-2(1H)-one, quinolin-2(1 H)-one and isoquinolin-1(2H)-one. Part 30: Structure-activity relationship studies of CNS agents

artículo científico publicado el 1 de junio de 1997

7-Arylpiperazinylalkyl and 7-tetrahydroisoquinolinylalkyl derivatives of 8-alkoxy-purine-2,6-dione and some of their purine-2,6,8-trione analogs as 5-HT(1A), 5-HT(2A), and 5-HT(7) serotonin receptor ligands

artículo científico publicado en 2007

8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone

artículo científico publicado en 1996

A search for new 5-HT1A/5-HT2A receptor ligands. In vitro and in vivo studies of 1-[omega-(4-aryl-1-piperazinyl)alkyl]indolin-2(1H)-ones

artículo científico publicado en 1998

Anticonflict effect of ipsapirone, buspirone and gepirone is not mediated by their common metabolite 1-(2-pyrimidinyl)piperazine ⬇️

artículo científico publicado el 1 de enero de 1989

Anticonflict effects of a competitive NMDA receptor antagonist and a partial agonist at strychnine-insensitive glycine receptors

artículo científico publicado en 1996

Anticonvulsant properties of N-(4-methylpiperazin-1-yl)- and N-[3-(4-methyl-piperazin-1-yl)propyl] derivatives of 3-aryl- and 3-spirocycloalkyl-pyrrolidine-2,5-dione

artículo científico publicado en 2005

Antidepressant-like activity of ipsapirone, buspirone and gepirone in the forced swimming test in rats pretreated with proadifen

artículo científico publicado en 1990

Antidepressant-like effect of neurotensin administered in the ventral tegmental area in the forced swimming test

artículo científico publicado el 1 de enero de 1992

Antidepressant-like effect of the selective 5-HT1B receptor agonist CP 94253: a possible mechanism of action

artículo científico publicado en 2005

Antidepressant-like effects of a partial agonist at strychnine-insensitive glycine receptors and a competitive NMDA receptor antagonist.

artículo científico publicado en 1997

Anxiolytic- and antidepressant-like effects of an antagonist at glycineB receptors

artículo científico publicado en 1998

Anxiolytic- and antidepressant-like effects of group III metabotropic glutamate agonist (1S,3R,4S)-1-aminocyclopentane-1,3,4-tricarboxylic acid (ACPT-I) in rats.

artículo científico publicado en 2002

Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor agonist does not involve GABA(A) signaling

artículo científico publicado en 2004

Anxiolytic-like effects of group I metabotropic glutamate antagonist 2-methyl-6-(phenylethynyl)-pyridine (MPEP) in rats

artículo científico publicado en 2000

Anxiolytic-like effects of metabotropic glutamate antagonist (RS)-alpha-methylserine-O-phosphate in rats.

artículo científico publicado en 1996

Central action of ipsapirone, a new anxiolytic drug, on serotoninergic, noradrenergic and dopaminergic functions

artículo científico publicado en 1987

Central antiserotonin action of fluperlapine

artículo científico publicado en 1985

Chemistry and anti-inflammatory activity of 10-methylamino-11H-indeno[1,2-b]quinolin-11-one (MB 432) derivatives

artículo científico publicado en 1983

Condensation of 1-(4,4-dimethyl-2-piperidon-6-yl)-2-propanone with benzaldehyde derivatives

artículo científico publicado en 1984

Conformational restriction in novel NAN-190 and MP3022 analogs and their 5-HT(1A) receptor activity

scientific article published on 01 September 2006

Corrigendum to “Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor antagonist does not involve GABAA signaling” [Neuropharmacology 47 (2004) 342–350]

scholarly article published in Neuropharmacology

Effect of combined administration of 5-HT1A or 5-HT1B/1D receptor antagonists and antidepressants in the forced swimming test

artículo científico publicado en 2004

Effect of glycine on antidepressant- and anxiolytic-like action of 1-aminocyclopropanecarboxylic acid (ACPC) in rats

scientific article published on 01 November 1996

Effect of linking bridge modifications on the 5-HT1A receptor activity of some 4-(omega-benzotriazol-1-yl)alkyl-1-(2-methoxy-phenyl)piperazines

artículo científico publicado en 1998

Effect of the amide fragment on 5-HT1A receptor activity of some analogs of MP 3022

scientific article published on 01 September 1999

Effect of the selective 5-HT7 receptor antagonist SB 269970 in animal models of anxiety and depression

artículo científico publicado en 2006

Effects of 8-OH-DPAT and ipsapirone in the tests used for evaluation of the antidepressant action.

artículo científico publicado en 1989

Effects of a selective 5-HT1B receptor agonist and antagonists in animal models of anxiety and depression

artículo científico publicado en 2004

Effects of combined administration of 5-HT1A and/or 5-HT1B receptor antagonists and paroxetine or fluoxetine in the forced swimming test in rats.

artículo científico publicado en 2002

Enhancement of the anti-immobility action of antidepressants by a selective 5-HT7 receptor antagonist in the forced swimming test in mice

scientific article published on 17 October 2006

Group III mGlu receptor agonists produce anxiolytic- and antidepressant-like effects after central administration in rats.

artículo científico publicado en 2004

Impact of aromatic substitution on the anticonvulsant activity of new N-(4-arylpiperazin-1-yl)-alkyl-2-azaspiro[4,5]decane-1,3-dione derivatives

scientific article published on 01 March 2006

Influence of the aliphatic spacer length on the 5-HT1A receptor activity of new arylpiperazines with an indazole system

artículo científico publicado en 2000

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors

artículo científico publicado en 2002

Involvement of 5-HT1A receptors in the antidepressant-like activity of gepirone in the forced swimming test in rats ⬇️

artículo científico publicado el 1 de julio de 1991

Multiple MPEP administrations evoke anxiolytic- and antidepressant-like effects in rats

artículo científico publicado en 2002

N-aminoalkylderivatives of 1,2,3,4-tetrahydro-beta-carboline-1-spiro-4'-N'- benzylpiperidine--a putative way to novel anxiolytic agents

artículo científico publicado en 1989

New 4-[omega-(diarylmethylamino)alkyl]- and 4-[omega-(diarylmethoxy)alkyl]-1-arylpiperazines as selective 5-HT1A/5-HT2A receptor ligands with differentiated in vivo activity.

artículo científico publicado en 2004

New 9- or 10-arylpiperazinoalkyl substituted pyrimido- or diazepino[2,1-f]purines with partial or full 5-HT1A agonistic activity

New arylpiperazine 5-HT(1A) receptor ligands containing the pyrimido[2,1-f]purine fragment: synthesis, in vitro, and in vivo pharmacological evaluation

artículo científico publicado en 2004

New hexahydro[1,4]diazepine-7H-5,7-diones with potential neurotropic activity

artículo científico publicado en 1984

Novel class of arylpiperazines containing N-acylated amino acids: their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation

artículo científico publicado en 2007

Novel, flexible, and conformationally defined analogs of gepirone: synthesis and 5-HT1A, 5-HT2A, and D2 receptor activity.

artículo científico publicado en 2005

Pharmacological properties and SAR of new 1,4-disubstituted piperazine derivatives with hypnotic-sedative activity

artículo científico publicado en 2002

Potential anxiolytic- and antidepressant-like effects of MPEP, a potent, selective and systemically active mGlu5 receptor antagonist

artículo científico publicado en 2001

Role of 5-HT1A receptors in the antinociceptive action of 8-hydroxy-2-(di-n- propylamino)tetralin in the rat

scientific article published on 01 September 1994

Some pharmacological properties of new analogs of MP 3022, the 5-HT1A receptor antagonist

artículo científico publicado en 1999

Stimulation of 5-HT1A receptors in the dorsal hippocampus impairs acquisition and performance of a spatial task in a water maze

artículo científico publicado el 6 de noviembre de 1992

Stimulation of group II metabotropic glutamate receptors or inhibition of group I ones exerts anxiolytic-like effects in rats

artículo científico publicado en 2000

Stimulation of hippocampal 5-HT1A receptors causes amnesia and anxiolytic-like but not antidepressant-like effects in the rat.

artículo científico publicado en 1993

Structure-activity relationship studies of CNS agents. Part 1: The Free-Wilson analysis of acute toxicity and sedative effect of some 1,2,3,4-tetrahydro-beta-carbolines.

artículo científico publicado en 1990

Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

artículo científico publicado en 1999

Structure-intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl)cyclohexane derivatives; new, potent 5-HT1A receptor agents with anxiolytic- like activity.

artículo científico publicado en 2005

Synthesis and 5-HT(1A), 5-HT(2A) receptor activity of new beta-tetralonohydantoins

artículo científico publicado en 2005

Synthesis and 5-HT1A/5-HT2A activity of some butyl analogs in the group of phenylpiperazine alkyl pyrimido[2,1-f]theophyllines.

artículo científico publicado en 2005

Synthesis and 5-HT1A/5-HT2A receptor activity of N-(4-arylpiperazin-1-yl)alkyl derivatives of 2-azaspiro([4.4]nonane and [4.5]decane-1,3-dione.

artículo científico publicado en 2006

Synthesis and 5-HT1A/5-HT2A receptor activity of new N-[3-(4-phenylpiperazin-1-yl)-propyl] derivatives of 3-spiro-cyclohexanepyrrolidine-2,5-dione and 3-spiro-beta-tetralonepyrrolidine-2,5-dione

artículo científico publicado el 1 de julio de 2003

Synthesis and anticonvulsant properties of N-methylpyridyl derivatives of m- and p-bromophenylsuccinimides

artículo científico publicado en 1987

Synthesis and pharmacological activity of some 2,3-dihydrofuran-2,3-dione derivatives

artículo científico publicado en 1982

Synthesis and pharmacological evaluation of new 5-(cyclo)alkyl-5-phenyl- and 5-spiroimidazolidine-2,4-dione derivatives. Novel 5-HT1A receptor agonist with potential antidepressant and anxiolytic activity

artículo científico publicado en 2009

Synthesis and pharmacological evaluation of new arylpiperazines. 3-[4-[4-(3-chlorophenyl)-1-piperazinyl]butyl]-quinazolidin-4-one - a dual serotonin 5-HT(1A)/5-HT(2A) receptor ligand with an anxiolytic-like activity

artículo científico publicado en 2002

Synthesis and pharmacological properties of N-(4-substituted-1-piperazinylalkyl)-1-butyl-2,5-dimethylpyrrole-3,4- dicarboxyimide derivatives.

artículo científico publicado en 1993

Synthesis and pharmacological properties of N-aroyl-beta-(1-indanyl)-ethylamines.

artículo científico publicado en 1980

Synthesis and pharmacological properties of N-arylpiperazine-N'-alkylindanes

artículo científico publicado el 1 de noviembre de 1984

Synthesis and pharmacological properties of decahydro-5H-pyrido [1',2'; 5,1]imidazo[3,4-a]-beta-carbolines

artículo científico publicado en 1986

Synthesis and pharmacological properties of decahydro-5H-pyrido [1',2';5,1] imidazo [3,4-a]-beta-carbolines. Part II.

artículo científico publicado en 1988

Synthesis and pharmacological properties of some 2-(3-aminopropionyl)- and 2-(3-aminopropyl)-1-(3-pyridyl)-1,2,3,4-tetrahydro-beta-carbolines

artículo científico publicado en 1988

Synthesis and pharmacological properties of some 2-pyrrolidinone Mannich bases

scientific article published on 01 November 1982

Synthesis and pharmacological properties of some 2-substituted 1-(3-pyridyl)-1,2,3,4-tetrahydro-beta-carbolines

artículo científico publicado en 1987

Synthesis and pharmacological properties of some N-aroylhomotryptamines

artículo científico publicado el 1 de marzo de 1979

Synthesis and pharmacological properties of some dipyrido[1,3]diazepinones

artículo científico publicado el 1 de septiembre de 1991

Synthesis and pharmacological properties of the products of condensation of tryptamine derivatives with pyridoxal

artículo científico publicado en 1984

Synthesis and preliminary pharmacological evaluation of imidazo[2,1-f]purine-2,4-dione derivatives

artículo científico publicado en 2009

Synthesis, in vitro and in vivo 5-HT1A/5-HT2A serotonin receptor activity of new hybrid 1,2,3,4-tetrahydro-gamma-carbolines with 1-(2-methoxyphenyl)piperazine moiety.

artículo científico publicado en 2003

The anti-inflammatory and analgesic activity of N-3-pyridoyltryptamine (tryptamide)

artículo científico publicado en 1987

The antianxiety-like effects of antagonists of group I and agonists of group II and III metabotropic glutamate receptors after intrahippocampal administration

artículo científico publicado en 2001

The anxiolytic-like activity of AIDA (1-aminoindan-1,5-dicarboxylic acid), an mGLu 1 receptor antagonist.

artículo científico publicado en 2004

The anxiolytic-like effect of 5-HT1B receptor ligands in rats: a possible mechanism of action

artículo científico publicado en 2005

The anxiolytic-like effect of metabotropic glutamate receptor antagonists after intrahippocampal injection in rats

artículo científico publicado en 1997

The behavioural, but not the hypothermic or corticosterone, response to 8-hydroxy-2-(DI-n-propylamino)-tetralin, is antagonized by NAN-190 in the rat

artículo científico publicado en 1990

The central action of 1-(2-pyrimidinyl)-piperazine, an ipsapirone metabolite

artículo científico publicado en 1989

The central action of carbamazepine as a potential antidepressant drug

artículo científico publicado en 1985

The influence of memantine on the anticonvulsant effects of the antiepileptic drugs.

artículo científico publicado en 1983

The influence of modifications in imide fragment structure on 5-HT(1A) and 5-HT(7) receptor affinity and in vivo pharmacological properties of some new 1-(m-trifluoromethylphenyl)piperazines

artículo científico publicado en 2007

The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT(1A)/5-HT(2A) receptor activities of its 1-adamantoyloaminoalkyl derivatives

artículo científico publicado en 2002

The influence of the benzodiazepine receptor antagonist flumazenil on the anxiolytic-like effects of CGP 37849 and ACPC in rats

artículo científico publicado en 2000

The novel buspirone analogue, 8-[4-[2-(1,2,3,4-tetrahydroisoquinolinyl)[butyl]-8-azaspiro [4.5 ]decane-7,9-dione, with anxiolytic-like and antidepressant-like effects in rats

artículo científico publicado en 1998

The pharmacological profile of chlordesmethyldiazepam and other benzodiazepines.

artículo científico publicado en 1986

The role of 5-hydroxytryptamine1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists

artículo científico publicado en 1994

The role of hippocampal 5-hydroxytryptamine 1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists

scientific article published on 01 September 1995

The role of postsynaptic 5-HT1A receptors in the anticonflict effect of ipsapirone

artículo científico publicado en 1994

Tolerance to anxiolytic- and antidepressant-like effects of a partial agonist of glycineB receptors

artículo científico publicado en 1999

Lista de obras de Ewa Tatarczyńska

1,2,3,4-tetrahydroisoquinoline derivatives: a new class of 5-HT1A receptor ligands

1,4-Benzoxazin-3(4H)-one derivatives and related compounds as 5-HT1A and 5-HT2A receptor ligands; the effect of the terminal amide fragment on the 5-HT1A/5-HT2A affinity and functional activity.

1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: synthesis, binding to serotonin (5-HT1A, 5-HT2A, 5-HT7), alpha1-adrenergic, and dopaminergic D2 receptors, and in vivo 5-HT1A functional characteristics

1-Pyridyl-3,4-dihydro-beta-carbolines: synthesis and central action.

2-H- and 2-acyl-9- [omega-[4-(2-methoxyphenyl)piperazinyl]-alkyl]-1,2,3,4-tetrahydro-beta-carbolines as ligands of 5-HT1A and 5-HT2A receptors.

5-HT1A and 5-HT2A receptor affinity and functional profile of some N-[3-(4-aryl-1-piperazinyl)propyl] derivatives of indolin-2(1H)-one, quinolin-2(1 H)-one and isoquinolin-1(2H)-one. Part 30: Structure-activity relationship studies of CNS agents

7-Arylpiperazinylalkyl and 7-tetrahydroisoquinolinylalkyl derivatives of 8-alkoxy-purine-2,6-dione and some of their purine-2,6,8-trione analogs as 5-HT(1A), 5-HT(2A), and 5-HT(7) serotonin receptor ligands

8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone

A search for new 5-HT1A/5-HT2A receptor ligands. In vitro and in vivo studies of 1-[omega-(4-aryl-1-piperazinyl)alkyl]indolin-2(1H)-ones

Anticonflict effect of ipsapirone, buspirone and gepirone is not mediated by their common metabolite 1-(2-pyrimidinyl)piperazine ⬇️

Anticonflict effects of a competitive NMDA receptor antagonist and a partial agonist at strychnine-insensitive glycine receptors

Anticonvulsant properties of N-(4-methylpiperazin-1-yl)- and N-[3-(4-methyl-piperazin-1-yl)propyl] derivatives of 3-aryl- and 3-spirocycloalkyl-pyrrolidine-2,5-dione

Antidepressant-like activity of ipsapirone, buspirone and gepirone in the forced swimming test in rats pretreated with proadifen

Antidepressant-like effect of neurotensin administered in the ventral tegmental area in the forced swimming test

Antidepressant-like effect of the selective 5-HT1B receptor agonist CP 94253: a possible mechanism of action

Antidepressant-like effects of a partial agonist at strychnine-insensitive glycine receptors and a competitive NMDA receptor antagonist.

Anxiolytic- and antidepressant-like effects of an antagonist at glycineB receptors

Anxiolytic- and antidepressant-like effects of group III metabotropic glutamate agonist (1S,3R,4S)-1-aminocyclopentane-1,3,4-tricarboxylic acid (ACPT-I) in rats.

Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor agonist does not involve GABA(A) signaling

Anxiolytic-like effects of group I metabotropic glutamate antagonist 2-methyl-6-(phenylethynyl)-pyridine (MPEP) in rats

Anxiolytic-like effects of metabotropic glutamate antagonist (RS)-alpha-methylserine-O-phosphate in rats.

Central action of ipsapirone, a new anxiolytic drug, on serotoninergic, noradrenergic and dopaminergic functions

Central antiserotonin action of fluperlapine

Chemistry and anti-inflammatory activity of 10-methylamino-11H-indeno[1,2-b]quinolin-11-one (MB 432) derivatives

Condensation of 1-(4,4-dimethyl-2-piperidon-6-yl)-2-propanone with benzaldehyde derivatives

Conformational restriction in novel NAN-190 and MP3022 analogs and their 5-HT(1A) receptor activity

Corrigendum to “Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor antagonist does not involve GABAA signaling” [Neuropharmacology 47 (2004) 342–350]

Effect of combined administration of 5-HT1A or 5-HT1B/1D receptor antagonists and antidepressants in the forced swimming test

Effect of glycine on antidepressant- and anxiolytic-like action of 1-aminocyclopropanecarboxylic acid (ACPC) in rats

Effect of linking bridge modifications on the 5-HT1A receptor activity of some 4-(omega-benzotriazol-1-yl)alkyl-1-(2-methoxy-phenyl)piperazines

Effect of the amide fragment on 5-HT1A receptor activity of some analogs of MP 3022

Effect of the selective 5-HT7 receptor antagonist SB 269970 in animal models of anxiety and depression

Effects of 8-OH-DPAT and ipsapirone in the tests used for evaluation of the antidepressant action.

Effects of a selective 5-HT1B receptor agonist and antagonists in animal models of anxiety and depression

Effects of combined administration of 5-HT1A and/or 5-HT1B receptor antagonists and paroxetine or fluoxetine in the forced swimming test in rats.

Enhancement of the anti-immobility action of antidepressants by a selective 5-HT7 receptor antagonist in the forced swimming test in mice

Group III mGlu receptor agonists produce anxiolytic- and antidepressant-like effects after central administration in rats.

Impact of aromatic substitution on the anticonvulsant activity of new N-(4-arylpiperazin-1-yl)-alkyl-2-azaspiro[4,5]decane-1,3-dione derivatives

Influence of the aliphatic spacer length on the 5-HT1A receptor activity of new arylpiperazines with an indazole system

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors

Involvement of 5-HT1A receptors in the antidepressant-like activity of gepirone in the forced swimming test in rats ⬇️

Multiple MPEP administrations evoke anxiolytic- and antidepressant-like effects in rats

N-aminoalkylderivatives of 1,2,3,4-tetrahydro-beta-carboline-1-spiro-4'-N'- benzylpiperidine--a putative way to novel anxiolytic agents

New 4-[omega-(diarylmethylamino)alkyl]- and 4-[omega-(diarylmethoxy)alkyl]-1-arylpiperazines as selective 5-HT1A/5-HT2A receptor ligands with differentiated in vivo activity.

New 9- or 10-arylpiperazinoalkyl substituted pyrimido- or diazepino[2,1-f]purines with partial or full 5-HT1A agonistic activity

New arylpiperazine 5-HT(1A) receptor ligands containing the pyrimido[2,1-f]purine fragment: synthesis, in vitro, and in vivo pharmacological evaluation

New hexahydro[1,4]diazepine-7H-5,7-diones with potential neurotropic activity

Novel class of arylpiperazines containing N-acylated amino acids: their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation

Novel, flexible, and conformationally defined analogs of gepirone: synthesis and 5-HT1A, 5-HT2A, and D2 receptor activity.

Pharmacological properties and SAR of new 1,4-disubstituted piperazine derivatives with hypnotic-sedative activity

Potential anxiolytic- and antidepressant-like effects of MPEP, a potent, selective and systemically active mGlu5 receptor antagonist

Role of 5-HT1A receptors in the antinociceptive action of 8-hydroxy-2-(di-n- propylamino)tetralin in the rat

Some pharmacological properties of new analogs of MP 3022, the 5-HT1A receptor antagonist

Stimulation of 5-HT1A receptors in the dorsal hippocampus impairs acquisition and performance of a spatial task in a water maze

Stimulation of group II metabotropic glutamate receptors or inhibition of group I ones exerts anxiolytic-like effects in rats

Stimulation of hippocampal 5-HT1A receptors causes amnesia and anxiolytic-like but not antidepressant-like effects in the rat.

Structure-activity relationship studies of CNS agents. Part 1: The Free-Wilson analysis of acute toxicity and sedative effect of some 1,2,3,4-tetrahydro-beta-carbolines.

Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

Structure-intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl)cyclohexane derivatives; new, potent 5-HT1A receptor agents with anxiolytic- like activity.

Synthesis and 5-HT(1A), 5-HT(2A) receptor activity of new beta-tetralonohydantoins

Synthesis and 5-HT1A/5-HT2A activity of some butyl analogs in the group of phenylpiperazine alkyl pyrimido[2,1-f]theophyllines.

Synthesis and 5-HT1A/5-HT2A receptor activity of N-(4-arylpiperazin-1-yl)alkyl derivatives of 2-azaspiro([4.4]nonane and [4.5]decane-1,3-dione.

Synthesis and 5-HT1A/5-HT2A receptor activity of new N-[3-(4-phenylpiperazin-1-yl)-propyl] derivatives of 3-spiro-cyclohexanepyrrolidine-2,5-dione and 3-spiro-beta-tetralonepyrrolidine-2,5-dione

Synthesis and anticonvulsant properties of N-methylpyridyl derivatives of m- and p-bromophenylsuccinimides

Synthesis and pharmacological activity of some 2,3-dihydrofuran-2,3-dione derivatives

Synthesis and pharmacological evaluation of new 5-(cyclo)alkyl-5-phenyl- and 5-spiroimidazolidine-2,4-dione derivatives. Novel 5-HT1A receptor agonist with potential antidepressant and anxiolytic activity

Synthesis and pharmacological evaluation of new arylpiperazines. 3-[4-[4-(3-chlorophenyl)-1-piperazinyl]butyl]-quinazolidin-4-one - a dual serotonin 5-HT(1A)/5-HT(2A) receptor ligand with an anxiolytic-like activity

Synthesis and pharmacological properties of N-(4-substituted-1-piperazinylalkyl)-1-butyl-2,5-dimethylpyrrole-3,4- dicarboxyimide derivatives.

Synthesis and pharmacological properties of N-aroyl-beta-(1-indanyl)-ethylamines.

Synthesis and pharmacological properties of N-arylpiperazine-N'-alkylindanes

Synthesis and pharmacological properties of decahydro-5H-pyrido [1',2'; 5,1]imidazo[3,4-a]-beta-carbolines

Synthesis and pharmacological properties of decahydro-5H-pyrido [1',2';5,1] imidazo [3,4-a]-beta-carbolines. Part II.

Synthesis and pharmacological properties of some 2-(3-aminopropionyl)- and 2-(3-aminopropyl)-1-(3-pyridyl)-1,2,3,4-tetrahydro-beta-carbolines

Synthesis and pharmacological properties of some 2-pyrrolidinone Mannich bases

Synthesis and pharmacological properties of some 2-substituted 1-(3-pyridyl)-1,2,3,4-tetrahydro-beta-carbolines

Synthesis and pharmacological properties of some N-aroylhomotryptamines

Synthesis and pharmacological properties of some dipyrido[1,3]diazepinones

Synthesis and pharmacological properties of the products of condensation of tryptamine derivatives with pyridoxal

Synthesis and preliminary pharmacological evaluation of imidazo[2,1-f]purine-2,4-dione derivatives