Lista de obras - Zdzisław Chilmonczyk - Dominio Público Uruguay

13C cross-polarization magic angle spinning NMR and gauge-independent atomic orbital, coupled Hartree-Fock calculations of buspirone analogues. Part 2. Hydrochlorides and perchlorates of 1-arylpiperazine-4-alkylimides

artículo científico publicado en 1999

1H, 13C, 15N NMR analysis of sildenafil base and citrate (Viagra) in solution, solid state and pharmaceutical dosage forms

artículo científico publicado en 2005

3D QSAR study of hypolipidemic asarones by comparative molecular surface analysis.

artículo científico publicado en 2005

A linear combination of pharmacophore hypotheses as a new tool in search of new active compounds--an application for 5-HT1A receptor ligands

artículo científico publicado en 2013

Assessment of the genotoxic activity of alpha-asarone and its derivatives in the comet assay

artículo científico publicado en 2013

Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line.

artículo científico publicado en 2017

Buspirone Analogs as Ligands of the 5-HT1A Receptor. 1. The Molecular Structure of Buspirone and Its Two Analogs

artículo científico publicado en 1995

Conformational flexibility of serotonin1A receptor ligands from crystallographic data. Updated model of the receptor pharmacophore.

artículo científico publicado en 1997

Corrigendum to 'Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line' Food Chem Toxicol. 111 (2018) 1-8

scientific article published on 04 May 2018

Deoxynucleosides with benzimidazoles as aglycone moiety are potent anticancer agents.

artículo científico publicado en 2017

Does molecular docking reveal alternative chemopreventive mechanism of activation of oxidoreductase by sulforaphane isothiocyanates?

artículo científico publicado en 2009

Enantioselective separation of 1,4-disubstituted piperazine derivatives on two cellulose chiralcel OD and OJ and one amylose chiralpak AD chiral selectors

scientific article published on 01 January 1999

Fluoroaryl analogs of sulforaphane - A group of compounds of anticancer and antimicrobial activity

artículo científico publicado en 2019

From Homology Models to a Set of Predictive Binding Pockets-a 5-HT1A Receptor Case Study

artículo científico publicado en 2017

Fullerene Derivatives of Nucleoside HIV Reverse Transcriptase Inhibitors-In Silico Activity Prediction

article

Functional Selectivity and Antidepressant Activity of Serotonin 1A Receptor Ligands

artículo científico publicado en 2015

Genotoxicity of alpha-asarone analogues.

artículo científico publicado en 2008

Hypolipidaemic and antiplatelet agents

artículo científico publicado en 2001

Identification of novel serotonin transporter compounds by virtual screening

artículo científico publicado en 2014

In Vitro Evaluation of Sulforaphane and a Natural Analog as Potent Inducers of 5-Fluorouracil Anticancer Activity

article published in 2018

In the triple-negative breast cancer MDA-MB-231 cell line, sulforaphane enhances the intracellular accumulation and anticancer action of doxorubicin encapsulated in liposomes

scientific article published on 12 January 2019

In-vivo effects of the 1,2,4-piperazine derivatives MM5 and MC1, putative 5-HT agonists, on dopamine and serotonin release in rat prefrontal cortex

artículo científico publicado en 2005

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors

artículo científico publicado en 2002

Intrinsic activity and comparative molecular dynamics of buspirone analogues at the 5-HT(1A) receptors.

artículo científico publicado en 2004

Ligand-5-HT1A receptor interaction

scientific article published on 01 March 2000

Ligand-directed trafficking of receptor stimulus

artículo científico publicado en 2014

Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors

artículo científico publicado en 2011

Models of 5-hydroxytryptamine receptors. A review.

artículo científico publicado en 1995

Molecular dynamics of 5-HT1A and 5-HT2A serotonin receptors with methylated buspirone analogues.

artículo científico publicado en 2001

Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol

artículo científico publicado en 2011

Molecular structure of some 3-amino-2-oxazolidinone derivatives.

artículo científico publicado en 2003

New benzimidazole-derived isothioureas as potential antileukemic agents--studies in vitro

artículo científico publicado en 2015

New enantiomeric fluorine-containing derivatives of sulforaphane: synthesis, absolute configurations and biological activity.

artículo científico publicado en 2014

New validated HPLC methodology for the determination of (-)-trans-paroxetine and its enantiomer in pharmaceutical formulations with use of ovomucoid chiral stationary phase

artículo científico publicado en 2014

Oncotoxic Properties of Serotonin Transporter Inhibitors and 5-HT Receptor Ligands

artículo científico publicado en 2018

Organofluorine Isoselenocyanate Analogues of Sulforaphane: Synthesis and Anticancer Activity.

artículo científico publicado en 2016

Pharmacological properties and SAR of new 1,4-disubstituted piperazine derivatives with hypnotic-sedative activity

artículo científico publicado en 2002

Proapoptotic activity of heterocyclic compounds containing succinimide moiety in the promyelocytic leukemia cell line HL-60.

artículo científico publicado en 2013

Proapoptotic effects of new pentabromobenzylisothiouronium salts in a human prostate adenocarcinoma cell line.

artículo científico publicado en 2012

Proapoptotic effects of novel pentabromobenzylisothioureas in human leukemia cell lines

artículo científico publicado en 2011

Rigid analogues of buspirone and gepirone, 5-HT1A receptors partial agonists

artículo científico publicado en 2002

Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents

artículo científico publicado en 2017

Some analogues of 1,4-disubstituted piperazines as hypnotic and sedative agents

scientific article published on 01 February 1995

Structure-retention relationship in a series of chiral 1,4-disubstituted piperazine derivatives on carbohydrate chiral stationary phases.

artículo científico publicado en 2005

Sulforaphane Regulates NFE2L2/Nrf2-Dependent Xenobiotic Metabolism Phase II and Phase III Enzymes Differently in Human Colorectal Cancer and Untransformed Epithelial Colon Cells.

artículo científico publicado en 2016

Synergistic anti-leukemic effects of CK2 inhibitors and pentabromobenzylisothioureas in vitro

artículo científico publicado en 2013

Synthesis and hypolipidemic and antiplatelet activities of alpha-asarone isomers in humans (in vitro), mice (in vivo), and rats (in vivo)

artículo científico publicado en 2000

Synthesis and proapoptotic properties of new casein kinase II inhibitors

artículo científico publicado el 1 de noviembre de 2010

Synthesis, antidepressant evaluation and docking studies of long-chain alkylnitroquipazines as serotonin transporter inhibitors

artículo científico publicado en 2013

Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors

artículo científico publicado en 2012

The Comparison of MTT and CVS Assays for the Assessment of Anticancer Agent Interactions

artículo científico publicado en 2016

The development and validation of a novel virtual screening cascade protocol to identify potential serotonin 5-HT(7)R antagonists

artículo científico publicado en 2010

The ligand-binding site of buspirone analogues at the 5-HT1A receptor.

artículo científico publicado en 1997

The molecular interactions of buspirone analogues with the serotonin transporter

artículo científico publicado en 2008

The new HPLC methodology for the chiral separation of tamsulosin enantiomers on amylose tris(3,5-dimethylphenylcarbamate) stationary phase

artículo científico publicado en 2012

Up-regulation of glutathione-related genes, enzyme activities and transport proteins in human cervical cancer cells treated with doxorubicin

artículo científico publicado en 2016

Lista de obras de Zdzisław Chilmonczyk

13C cross-polarization magic angle spinning NMR and gauge-independent atomic orbital, coupled Hartree-Fock calculations of buspirone analogues. Part 2. Hydrochlorides and perchlorates of 1-arylpiperazine-4-alkylimides

1H, 13C, 15N NMR analysis of sildenafil base and citrate (Viagra) in solution, solid state and pharmaceutical dosage forms

3D QSAR study of hypolipidemic asarones by comparative molecular surface analysis.

A linear combination of pharmacophore hypotheses as a new tool in search of new active compounds--an application for 5-HT1A receptor ligands

Assessment of the genotoxic activity of alpha-asarone and its derivatives in the comet assay

Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line.

Buspirone Analogs as Ligands of the 5-HT1A Receptor. 1. The Molecular Structure of Buspirone and Its Two Analogs

Conformational flexibility of serotonin1A receptor ligands from crystallographic data. Updated model of the receptor pharmacophore.

Corrigendum to 'Autophagic cell death and premature senescence: New mechanism of 5-fluorouracil and sulforaphane synergistic anticancer effect in MDA-MB-231 triple negative breast cancer cell line' Food Chem Toxicol. 111 (2018) 1-8

Deoxynucleosides with benzimidazoles as aglycone moiety are potent anticancer agents.

Does molecular docking reveal alternative chemopreventive mechanism of activation of oxidoreductase by sulforaphane isothiocyanates?

Enantioselective separation of 1,4-disubstituted piperazine derivatives on two cellulose chiralcel OD and OJ and one amylose chiralpak AD chiral selectors

Fluoroaryl analogs of sulforaphane - A group of compounds of anticancer and antimicrobial activity

From Homology Models to a Set of Predictive Binding Pockets-a 5-HT1A Receptor Case Study

Fullerene Derivatives of Nucleoside HIV Reverse Transcriptase Inhibitors-In Silico Activity Prediction

Functional Selectivity and Antidepressant Activity of Serotonin 1A Receptor Ligands

Genotoxicity of alpha-asarone analogues.

Hypolipidaemic and antiplatelet agents

Identification of novel serotonin transporter compounds by virtual screening

In Vitro Evaluation of Sulforaphane and a Natural Analog as Potent Inducers of 5-Fluorouracil Anticancer Activity

In the triple-negative breast cancer MDA-MB-231 cell line, sulforaphane enhances the intracellular accumulation and anticancer action of doxorubicin encapsulated in liposomes

In-vivo effects of the 1,2,4-piperazine derivatives MM5 and MC1, putative 5-HT agonists, on dopamine and serotonin release in rat prefrontal cortex

Interaction of 1,2,4-substituted piperazines, new serotonin receptor ligands, with 5-HT1A and 5-HT2A receptors

Intrinsic activity and comparative molecular dynamics of buspirone analogues at the 5-HT(1A) receptors.

Ligand-5-HT1A receptor interaction

Ligand-directed trafficking of receptor stimulus

Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors

Models of 5-hydroxytryptamine receptors. A review.

Molecular dynamics of 5-HT1A and 5-HT2A serotonin receptors with methylated buspirone analogues.

Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol

Molecular structure of some 3-amino-2-oxazolidinone derivatives.

New benzimidazole-derived isothioureas as potential antileukemic agents--studies in vitro

New enantiomeric fluorine-containing derivatives of sulforaphane: synthesis, absolute configurations and biological activity.

New validated HPLC methodology for the determination of (-)-trans-paroxetine and its enantiomer in pharmaceutical formulations with use of ovomucoid chiral stationary phase

Oncotoxic Properties of Serotonin Transporter Inhibitors and 5-HT Receptor Ligands

Organofluorine Isoselenocyanate Analogues of Sulforaphane: Synthesis and Anticancer Activity.

Pharmacological properties and SAR of new 1,4-disubstituted piperazine derivatives with hypnotic-sedative activity

Proapoptotic activity of heterocyclic compounds containing succinimide moiety in the promyelocytic leukemia cell line HL-60.

Proapoptotic effects of new pentabromobenzylisothiouronium salts in a human prostate adenocarcinoma cell line.

Proapoptotic effects of novel pentabromobenzylisothioureas in human leukemia cell lines

Rigid analogues of buspirone and gepirone, 5-HT1A receptors partial agonists

Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents

Some analogues of 1,4-disubstituted piperazines as hypnotic and sedative agents

Structure-retention relationship in a series of chiral 1,4-disubstituted piperazine derivatives on carbohydrate chiral stationary phases.

Sulforaphane Regulates NFE2L2/Nrf2-Dependent Xenobiotic Metabolism Phase II and Phase III Enzymes Differently in Human Colorectal Cancer and Untransformed Epithelial Colon Cells.

Synergistic anti-leukemic effects of CK2 inhibitors and pentabromobenzylisothioureas in vitro

Synthesis and hypolipidemic and antiplatelet activities of alpha-asarone isomers in humans (in vitro), mice (in vivo), and rats (in vivo)

Synthesis and proapoptotic properties of new casein kinase II inhibitors

Synthesis, antidepressant evaluation and docking studies of long-chain alkylnitroquipazines as serotonin transporter inhibitors

Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors

The Comparison of MTT and CVS Assays for the Assessment of Anticancer Agent Interactions

The development and validation of a novel virtual screening cascade protocol to identify potential serotonin 5-HT(7)R antagonists

The ligand-binding site of buspirone analogues at the 5-HT1A receptor.

The molecular interactions of buspirone analogues with the serotonin transporter

The new HPLC methodology for the chiral separation of tamsulosin enantiomers on amylose tris(3,5-dimethylphenylcarbamate) stationary phase

Up-regulation of glutathione-related genes, enzyme activities and transport proteins in human cervical cancer cells treated with doxorubicin