Lista de obras - Etsuo Yonemochi - Dominio Público Uruguay

A new solvate of epalerstat, a drug for diabetic neuropathy.

artículo científico publicado en 2017

Applicability of DPI formulations for novel neurokinin receptor antagonist

artículo científico publicado en 2008

Application and mechanism of inhalation profile improvement of DPI formulations by mechanofusion with magnesium stearate

artículo científico publicado en 2008

Application of Eudragit RS to thermo-sensitive drug delivery systems: II. Effect of temperature on drug permeability through membrane consisting of Eudragit RS/PEG 400 blend polymers

artículo científico publicado en 2005

Application of eudragit RS to thermo-sensitive drug delivery systems. I. Thermo-sensitive drug release from acetaminophen matrix tablets consisting of eudragit RS/PEG 400 blend polymers

artículo científico publicado en 2002

Applying terahertz technology for nondestructive detection of crack initiation in a film-coated layer on a swelling tablet

artículo científico publicado en 2012

Changes in surface properties by granulation and physicochemical stability of granulated amorphous cefditoren pivoxil with additives

artículo científico publicado en 2004

Characterization and Quality Control of Pharmaceutical Cocrystals

artículo científico publicado en 2016

Characterization of complexes between phenethylamine enantiomers and β-cyclodextrin derivatives by capillary electrophoresis-Determination of binding constants and complex mobilities.

artículo científico publicado en 2017

Characterization of polymorphs of a novel quinolinone derivative, TA-270 (4-hydroxy-1-methyl-3-octyloxy-7-sinapinoylamino-2(1H)-quinolinone)

artículo científico publicado en 2001

Clarifying the mechanism of aggregation of particles in high-shear granulation based on their surface properties by using micro-spectroscopy.

artículo científico

Cocrystallization and amorphization induced by drug-excipient interaction improves the physical properties of acyclovir.

artículo científico publicado en 2011

Comparison of molecular mobility in the glassy state between amorphous indomethacin and salicin based on spin-lattice relaxation times

artículo científico publicado en 2005

Competition of thermodynamic and dynamic factors during formation of multicomponent particles via spray drying

artículo científico publicado en 2012

Component crystallization and physical collapse during freeze-drying of L-arginine-citric acid mixtures

artículo científico publicado en 2012

Correlation between glass-forming ability and fragility of pharmaceutical compounds.

artículo científico publicado en 2015

Crystal Structure Determination of Dimenhydrinate after More than 60 Years: Solving Salt–Cocrystal Ambiguity via Solid-State Characterizations and Solubility Study

Determination for dry layer resistance of sucrose under various primary drying conditions using a novel simulation program for designing pharmaceutical lyophilization cycle

artículo científico publicado en 2013

Development of a method for the determination of caffeine anhydrate in various designed intact tablets [correction of tables] by near-infrared spectroscopy: a comparison between reflectance and transmittance technique

artículo científico publicado en 2008

Development of a rapid process monitoring method for dry-coated tableting process by using near-infrared spectroscopy.

artículo científico publicado en 2011

Development of fast disintegrating compressed tablets using amino acid as disintegration accelerator: evaluation of wetting and disintegration of tablet on the basis of surface free energy

artículo científico publicado en 2005

Development of microparticles coated with poly-γ-glutamic acid to improve oral absorption of a poorly water-soluble drug

scientific article published on 18 June 2019

Differences in crystallization behavior between quenched and ground amorphous ursodeoxycholic acid

artículo científico publicado en 1999

Do amorphous troglitazones prepared from two diastereomer-pairs have the same molecular mobility and crystallization rate at the surface?

scientific article published on 01 January 2011

Effect of Polymers and Storage Relative Humidity on Amorphous Rebamipide and Its Solid Dispersion Transformation: Multiple Spectra Chemometrics of Powder X-Ray Diffraction and Near-Infrared Spectroscopy

scientific article published on 10 July 2020

Effect of physical properties of troglitazone crystal on the molecular interaction with PVP during heating

artículo científico publicado en 2006

Effect of sulfobutyl ether-β-cyclodextrin and propylene glycol alginate on the solubility of clozapine

scientific article published on 11 September 2018

Effect of the type of lubricant on the characteristics of orally disintegrating tablets manufactured using the phase transition of sugar alcohol

artículo científico publicado en 2008

Effect of water-soluble carriers on dissolution characteristics of nifedipine solid dispersions

Effects of formulation and process factors on the crystal structure of freeze-dried Myo-inositol

scientific article published on 10 June 2014

Effects of solute miscibility on the micro- and macroscopic structural integrity of freeze-dried solids

scientific article published on 01 November 2010

Effects of sugar ester and hydroxypropyl methylcellulose on the physicochemical stability of amorphous cefditoren pivoxil in aqueous suspension

artículo científico publicado en 2005

Effects of water content in physical mixture and heating temperature on crystallinity of troglitazone-PVP K30 solid dispersions prepared by closed melting method

artículo científico publicado en 2005

Enhanced dissolution and skin permeation profiles of epalrestat with β-cyclodextrin derivatives using a cogrinding method

artículo científico publicado en 2017

Epalrestat tetra-hydro-furan monosolvate: crystal structure and phase transition

artículo científico publicado en 2017

Estimation of initial dissolution rate of drug substance by thermal analysis: application for carbamazepine hydrate

artículo científico publicado en 2002

Evaluation of amorphous ursodeoxycholic acid by thermal methods

artículo científico publicado en 1997

Evaluation of antitumor effect of zoledronic acid entrapped in folate-linked liposome for targeting to tumor-associated macrophages

artículo científico publicado en 2014

Evaluation of rapidly disintegrating tablets containing glycine and carboxymethylcellulose

artículo científico publicado en 2006

Evaluation of solid dispersions on a molecular level by the Raman mapping technique

artículo científico publicado en 2008

Evaluation of the crystalline and amorphous states of drug products by nanothermal analysis and Raman imaging

artículo científico publicado en 2012

Evaluation of the physical properties of dry surface-modified ibuprofen using a powder rheometer (FT4) and analysis of the influence of pharmaceutical additives on improvement of the powder flowability

artículo científico publicado en 2020

Factors affecting the apparent solubility of ursodeoxycholic acid in the grinding process

artículo científico publicado en 2003

Fluorometric Studies of Pyrene Adsorption on Porous Crystalline Cellulose

artículo científico publicado en 1998

Fluorometric study of the molecular states of 2,5-diphenyloxazole in ground mixtures with gamma-cyclodextrin

scientific article published on 01 February 1994

Formulation design of a novel fast-disintegrating tablet

artículo científico publicado en 2005

Freeze-drying of proteins in glass solids formed by basic amino acids and dicarboxylic acids

artículo científico publicado en 2009

Freeze-drying of proteins with glass-forming oligosaccharide-derived sugar alcohols

artículo científico publicado en 2010

Glass-state amorphous salt solids formed by freeze-drying of amines and hydroxy carboxylic acids: effect of hydrogen-bonding and electrostatic interactions

artículo científico publicado en 2008

Importance of excipient wettability on tablet characteristics prepared by moisture activated dry granulation (MADG).

artículo científico publicado en 2013

In vivo siRNA delivery system for targeting to the liver by poly-l-glutamic acid-coated lipoplex

artículo científico publicado en 2014

Interaction of microcrystalline cellulose and water in granules prepared by a high-shear mixer

artículo científico publicado en 2001

Investigation of the dynamic process during spray-drying to improve aerodynamic performance of inhalation particles.

artículo científico publicado en 2010

Low-density microparticles with petaloid surface structure for pulmonary drug delivery

artículo científico publicado en 2014

Mechanisms for Improved Hygroscopicity of L-Arginine Valproate Revealed by X-Ray Single Crystal Structure Analysis

artículo científico publicado en 2016

Microscopic molecular mobility of amorphous AG-041R measured by solid-state 13C NMR.

artículo científico publicado en 2004

Molecular Dynamics of Amorphous Sulfamethazine With Structurally Related Sulfonamide Impurities Evaluated Using Thermal Analysis

artículo científico publicado en 2016

Molecular properties of propranolol hydrochloride prepared as drug-resin complexes

artículo científico publicado en 2001

Molecular states of p-dimethylaminobenzonitrile coground with β-cyclodextrin investigated using solid-state fluorescence spectroscopy

scientific article published on 01 January 2011

Near IR spectroscopy to quantify the silica content and difference between silicified microcrystalline cellulose and physical mixtures of microcrystalline cellulose and silica

artículo científico publicado en 2000

New approach to optimizing risk management of the sticking problem using scale-independent critical material attributes and the quantitative process parameter

scientific article published on 15 January 2020

Novel approach to DPI carrier lactose with mechanofusion process with additives and evaluation by IGC.

artículo científico publicado en 2006

Novel approach to evaluating granulation and segregation level considering the contribution of hydroxypropyl cellulose to the surface property change of granules

artículo científico publicado en 2020

Novel, lean and environment-friendly granulation method: Green fluidized bed granulation (GFBG)

artículo científico publicado en 2018

Optimization of primary drying condition for pharmaceutical lyophilization using a novel simulation program with a predictive model for dry layer resistance

artículo científico publicado en 2014

Physicochemical Properties of Ursodeoxycholic Acid Dispersed in Controlled Pore Glass

scientific article published on 01 August 1999

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs I: anhydrates and hydrate.

artículo científico publicado en 2014

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs II: Solvate and cocrystal

scientific article published on 17 March 2015

Physicochemical properties of amorphous clarithromycin obtained by grinding and spray drying

artículo científico publicado en 1999

Potential of synchrotron X-ray powder diffractometry for detection and quantification of small amounts of crystalline drug substances in pharmaceutical tablets

artículo científico publicado en 2011

Practical approach for measuring heat capacity of pharmaceutical crystals/glasses by modulated-temperature differential scanning calorimetry

scientific article published on 01 January 2013

Quantitative correlation between initial dissolution rate and heat of fusion of drug substance

scientific article published on 01 August 2000

Quantitative correlation between initial dissolution rate and heat of solution of drug

artículo científico publicado en 2000

Quantitative determination of amorphous nicardipine hydrochloride in long acting formula (NIC-LA) using light anhydrous silicic acid

artículo científico publicado en 2004

Quantitative relationship between solubility, initial dissolution rate and heat of solution of chiral drugs

artículo científico publicado en 2000

Reevaluation of solubility of tolbutamide and polymorphic transformation from Form I to unknown crystal form.

artículo científico publicado en 2008

Relationship between crystallization tendencies during cooling from melt and isothermal storage: toward a general understanding of physical stability of pharmaceutical glasses

artículo científico publicado en 2014

Sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA could effectively deliver siRNA to the liver

artículo científico publicado en 2014

Solid states fluorescence study of p-dimethylaminobenzonitrile by co-grinding with cyclodextrins

artículo científico publicado en 2009

Solid-state 13C NMR study of indomethacin polymorphism

artículo científico publicado en 2006

Solid-state fluorescence study of naphthalene adsorption on porous material.

artículo científico publicado en 2002

Solubility Improvement of Benexate through Salt Formation Using Artificial Sweetener.

artículo científico publicado en 2018

Stabilization of protein structure in freeze-dried amorphous organic acid buffer salts.

artículo científico publicado en 2009

Study of the pseudo-crystalline transformation from form i to form II of thiamine hydrochloride (vitamin B(1))

scientific article published on 01 January 2011

Studying the morphology of lyophilized protein solids using X-ray micro-CT: effect of post-freeze annealing and controlled nucleation

artículo científico publicado en 2014

Swelling kinetics of spray-dried chitosan acetate assessed by magnetic resonance imaging and their relation to drug release kinetics of chitosan matrix tablets

artículo científico publicado en 2010

Synthesis and Characterization of Cholesteryl Conjugated Lysozyme (CHLysozyme)

artículo científico publicado en 2020

The effect of structurally related impurities on crystallinity reduction of sulfamethazine by grinding.

artículo científico publicado en 2016

The importance of binder moisture content in Metformin HCL high-dose formulations prepared by moist aqueous granulation (MAG).

artículo científico publicado en 2015

Therapeutic effect for liver-metastasized tumor by sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA.

artículo científico publicado en 2015

Triboelectrification of active pharmaceutical ingredients: week acids and their salts

artículo científico publicado en 2015

Tumor delivery of liposomal doxorubicin prepared with poly-L-glutamic acid as a drug-trapping agent.

artículo científico publicado en 2016

Uniformity and physical states of troglitazone in solid dispersions determined by electron probe microanalysis and microthermal analysis

artículo científico publicado en 2004

Water sorption and near IR spectroscopy to study the differences between microcrystalline cellulose and silicified microcrystalline cellulose before and after wet granulation

artículo científico publicado en 1999

Zoledronic acid enhances antitumor efficacy of liposomal doxorubicin

artículo científico publicado en 2015

siRNA delivery to lung-metastasized tumor by systemic injection with cationic liposomes

artículo científico publicado en 2015

Lista de obras de Etsuo Yonemochi

A new solvate of epalerstat, a drug for diabetic neuropathy.

Applicability of DPI formulations for novel neurokinin receptor antagonist

Application and mechanism of inhalation profile improvement of DPI formulations by mechanofusion with magnesium stearate

Application of Eudragit RS to thermo-sensitive drug delivery systems: II. Effect of temperature on drug permeability through membrane consisting of Eudragit RS/PEG 400 blend polymers

Application of eudragit RS to thermo-sensitive drug delivery systems. I. Thermo-sensitive drug release from acetaminophen matrix tablets consisting of eudragit RS/PEG 400 blend polymers

Applying terahertz technology for nondestructive detection of crack initiation in a film-coated layer on a swelling tablet

Changes in surface properties by granulation and physicochemical stability of granulated amorphous cefditoren pivoxil with additives

Characterization and Quality Control of Pharmaceutical Cocrystals

Characterization of complexes between phenethylamine enantiomers and β-cyclodextrin derivatives by capillary electrophoresis-Determination of binding constants and complex mobilities.

Characterization of polymorphs of a novel quinolinone derivative, TA-270 (4-hydroxy-1-methyl-3-octyloxy-7-sinapinoylamino-2(1H)-quinolinone)

Clarifying the mechanism of aggregation of particles in high-shear granulation based on their surface properties by using micro-spectroscopy.

Cocrystallization and amorphization induced by drug-excipient interaction improves the physical properties of acyclovir.

Comparison of molecular mobility in the glassy state between amorphous indomethacin and salicin based on spin-lattice relaxation times

Competition of thermodynamic and dynamic factors during formation of multicomponent particles via spray drying

Component crystallization and physical collapse during freeze-drying of L-arginine-citric acid mixtures

Correlation between glass-forming ability and fragility of pharmaceutical compounds.

Crystal Structure Determination of Dimenhydrinate after More than 60 Years: Solving Salt–Cocrystal Ambiguity via Solid-State Characterizations and Solubility Study

Determination for dry layer resistance of sucrose under various primary drying conditions using a novel simulation program for designing pharmaceutical lyophilization cycle

Development of a method for the determination of caffeine anhydrate in various designed intact tablets [correction of tables] by near-infrared spectroscopy: a comparison between reflectance and transmittance technique

Development of a rapid process monitoring method for dry-coated tableting process by using near-infrared spectroscopy.

Development of fast disintegrating compressed tablets using amino acid as disintegration accelerator: evaluation of wetting and disintegration of tablet on the basis of surface free energy

Development of microparticles coated with poly-γ-glutamic acid to improve oral absorption of a poorly water-soluble drug

Differences in crystallization behavior between quenched and ground amorphous ursodeoxycholic acid

Do amorphous troglitazones prepared from two diastereomer-pairs have the same molecular mobility and crystallization rate at the surface?

Effect of Polymers and Storage Relative Humidity on Amorphous Rebamipide and Its Solid Dispersion Transformation: Multiple Spectra Chemometrics of Powder X-Ray Diffraction and Near-Infrared Spectroscopy

Effect of physical properties of troglitazone crystal on the molecular interaction with PVP during heating

Effect of sulfobutyl ether-β-cyclodextrin and propylene glycol alginate on the solubility of clozapine

Effect of the type of lubricant on the characteristics of orally disintegrating tablets manufactured using the phase transition of sugar alcohol

Effect of water-soluble carriers on dissolution characteristics of nifedipine solid dispersions

Effects of formulation and process factors on the crystal structure of freeze-dried Myo-inositol

Effects of solute miscibility on the micro- and macroscopic structural integrity of freeze-dried solids

Effects of sugar ester and hydroxypropyl methylcellulose on the physicochemical stability of amorphous cefditoren pivoxil in aqueous suspension

Effects of water content in physical mixture and heating temperature on crystallinity of troglitazone-PVP K30 solid dispersions prepared by closed melting method

Enhanced dissolution and skin permeation profiles of epalrestat with β-cyclodextrin derivatives using a cogrinding method

Epalrestat tetra-hydro-furan monosolvate: crystal structure and phase transition

Estimation of initial dissolution rate of drug substance by thermal analysis: application for carbamazepine hydrate

Evaluation of amorphous ursodeoxycholic acid by thermal methods

Evaluation of antitumor effect of zoledronic acid entrapped in folate-linked liposome for targeting to tumor-associated macrophages

Evaluation of rapidly disintegrating tablets containing glycine and carboxymethylcellulose

Evaluation of solid dispersions on a molecular level by the Raman mapping technique

Evaluation of the crystalline and amorphous states of drug products by nanothermal analysis and Raman imaging

Evaluation of the physical properties of dry surface-modified ibuprofen using a powder rheometer (FT4) and analysis of the influence of pharmaceutical additives on improvement of the powder flowability

Factors affecting the apparent solubility of ursodeoxycholic acid in the grinding process

Fluorometric Studies of Pyrene Adsorption on Porous Crystalline Cellulose

Fluorometric study of the molecular states of 2,5-diphenyloxazole in ground mixtures with gamma-cyclodextrin

Formulation design of a novel fast-disintegrating tablet

Freeze-drying of proteins in glass solids formed by basic amino acids and dicarboxylic acids

Freeze-drying of proteins with glass-forming oligosaccharide-derived sugar alcohols

Glass-state amorphous salt solids formed by freeze-drying of amines and hydroxy carboxylic acids: effect of hydrogen-bonding and electrostatic interactions

Importance of excipient wettability on tablet characteristics prepared by moisture activated dry granulation (MADG).

In vivo siRNA delivery system for targeting to the liver by poly-l-glutamic acid-coated lipoplex

Interaction of microcrystalline cellulose and water in granules prepared by a high-shear mixer

Investigation of the dynamic process during spray-drying to improve aerodynamic performance of inhalation particles.

Low-density microparticles with petaloid surface structure for pulmonary drug delivery

Mechanisms for Improved Hygroscopicity of L-Arginine Valproate Revealed by X-Ray Single Crystal Structure Analysis

Microscopic molecular mobility of amorphous AG-041R measured by solid-state 13C NMR.

Molecular Dynamics of Amorphous Sulfamethazine With Structurally Related Sulfonamide Impurities Evaluated Using Thermal Analysis

Molecular properties of propranolol hydrochloride prepared as drug-resin complexes

Molecular states of p-dimethylaminobenzonitrile coground with β-cyclodextrin investigated using solid-state fluorescence spectroscopy

Near IR spectroscopy to quantify the silica content and difference between silicified microcrystalline cellulose and physical mixtures of microcrystalline cellulose and silica

New approach to optimizing risk management of the sticking problem using scale-independent critical material attributes and the quantitative process parameter

Novel approach to DPI carrier lactose with mechanofusion process with additives and evaluation by IGC.

Novel approach to evaluating granulation and segregation level considering the contribution of hydroxypropyl cellulose to the surface property change of granules

Novel, lean and environment-friendly granulation method: Green fluidized bed granulation (GFBG)

Optimization of primary drying condition for pharmaceutical lyophilization using a novel simulation program with a predictive model for dry layer resistance

Physicochemical Properties of Ursodeoxycholic Acid Dispersed in Controlled Pore Glass

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs I: anhydrates and hydrate.

Physicochemical and crystal structure analysis of pranlukast pseudo-polymorphs II: Solvate and cocrystal

Physicochemical properties of amorphous clarithromycin obtained by grinding and spray drying

Potential of synchrotron X-ray powder diffractometry for detection and quantification of small amounts of crystalline drug substances in pharmaceutical tablets

Practical approach for measuring heat capacity of pharmaceutical crystals/glasses by modulated-temperature differential scanning calorimetry

Quantitative correlation between initial dissolution rate and heat of fusion of drug substance

Quantitative correlation between initial dissolution rate and heat of solution of drug

Quantitative determination of amorphous nicardipine hydrochloride in long acting formula (NIC-LA) using light anhydrous silicic acid

Quantitative relationship between solubility, initial dissolution rate and heat of solution of chiral drugs

Reevaluation of solubility of tolbutamide and polymorphic transformation from Form I to unknown crystal form.

Relationship between crystallization tendencies during cooling from melt and isothermal storage: toward a general understanding of physical stability of pharmaceutical glasses

Sequential intravenous injection of anionic polymer and cationic lipoplex of siRNA could effectively deliver siRNA to the liver

Solid states fluorescence study of p-dimethylaminobenzonitrile by co-grinding with cyclodextrins