Lista de obras - Taleb H Al-Tel - Dominio Público Uruguay

BACE1 inhibitors: Current status and future directions in treating Alzheimer's disease

artículo científico publicado en 2019

Design and synthesis of novel tetrahydro-2H-Pyrano[3,2-c]Pyridazin-3(6H)-one derivatives as potential anticancer agents ⬇️

artículo científico publicado el 17 de septiembre de 2010

Design, synthesis and SAR analysis of potent BACE1 inhibitors: Possible lead drug candidates for Alzheimer's disease.

artículo científico publicado en 2016

Design, synthesis and biological evaluation of new pyrrolidine carboxamide analogues as potential chemotherapeutic agents for hepatocellular carcinoma.

artículo científico publicado en 2017

Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs

artículo científico publicado en 2011

Design, synthesis and qualitative structure-activity evaluations of novel hexahydropyrano[3,2-c][1,2]diazepin-3(4H)-one and tetrahydropyrano[3,2-b]pyrrol-2(1H)-one derivatives as anticancer agents

artículo científico publicado el 21 de julio de 2010

Design, synthesis, and qualitative structure-activity evaluations of novel β-secretase inhibitors as potential Alzheimer's drug leads.

artículo científico publicado en 2011

Differential use of anhydropyranosides for enantiopure routes to bis-gamma-butyrolactones: a new approach to the frameworks of antibiotic and anticancer agents isoavenaciolide and ethisolide.

artículo científico publicado en 2009

Divergent Strategy for Diastereocontrolled Synthesis of Small- and Medium-Ring Architectures

artículo científico publicado en 2020

Domino Transformations of Ene/Yne Tethered Salicylaldehyde Derivatives: Pluripotent Platforms for the Construction of High sp3 Content and Privileged Architectures

artículo científico publicado en 2019

Drug development post COVID-19 pandemic: toward a better system to meet current and future global health challenges

artículo científico publicado en 2020

Epigenetics and miRNA as predictive markers and targets for lung cancer chemotherapy.

artículo científico publicado en 2015

Flexible, polymer-supported synthesis of sphingosine derivatives provides ceramides with enhanced biological activity.

artículo científico publicado en 2014

Modulation of DNA damage response and induction of apoptosis mediates synergism between doxorubicin and a new imidazopyridine derivative in breast and lung cancer cells.

artículo científico publicado en 2015

Multidirectional desymmetrization of pluripotent building block en route to diastereoselective synthesis of complex nature-inspired scaffolds

artículo científico publicado en 2018

Mutations in the nonstructural protein 3A confer resistance to the novel enterovirus replication inhibitor TTP-8307.

artículo científico publicado en 2009

One-Pot Synthesis of Diverse Collections of Benzoxazepine and Indolopyrazine Fused to Heterocyclic Systems

artículo científico publicado en 2019

Post Groebke-Blackburn multicomponent protocol: synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents.

artículo científico publicado en 2010

Post-Ugi Cascade Transformations for Accessing Diverse Chromenopyrrole Collections.

artículo científico publicado en 2018

Rational design and synthesis of potent dibenzazepine motifs as beta-secretase inhibitors

artículo científico publicado en 2009

Sequencing [4 + 1]-Cycloaddition and Aza-Michael Addition Reactions: A Diastereoselective Cascade for the Rapid Access of Pyrido[2',1':2,3]/Thiazolo[2',3':2,3]imidazo[1,5-a]quinolone Scaffolds as Potential Antibacterial and Anticancer Motifs

scientific article published on 31 October 2019

Stereocontrolled transformations of cyclohexadienone derivatives to access stereochemically rich and natural product-inspired architectures

artículo científico publicado en 2020

Structure activity relationship of phenolic acid inhibitors of α-synuclein fibril formation and toxicity

artículo científico publicado en 2014

Superbugs but no drugs: steps in averting a post-antibiotic era

scientific article published on 16 August 2019

Synthesis and antimicrobial activity of cholic acid hydrazone analogues

artículo científico publicado en 2010

Synthesis of a new series of heterocyclic scaffolds for medicinal purposes

scientific article published on 22 June 2006

Tandem Achmatowicz-Knoevenagel protocol: diastereoselective synthesis and anticancer evaluation of cyclopenta[b]pyrane derivatives ⬇️

artículo científico publicado el 20 de septiembre de 2010

Tandem multicomponent reactions toward the design and synthesis of novel antibacterial and cytotoxic motifs.

artículo científico publicado en 2013

Lista de obras de Taleb H Al-Tel

BACE1 inhibitors: Current status and future directions in treating Alzheimer's disease

Design and synthesis of novel tetrahydro-2H-Pyrano[3,2-c]Pyridazin-3(6H)-one derivatives as potential anticancer agents ⬇️

Design, synthesis and SAR analysis of potent BACE1 inhibitors: Possible lead drug candidates for Alzheimer's disease.

Design, synthesis and biological evaluation of new pyrrolidine carboxamide analogues as potential chemotherapeutic agents for hepatocellular carcinoma.

Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs

Design, synthesis and qualitative structure-activity evaluations of novel hexahydropyrano[3,2-c][1,2]diazepin-3(4H)-one and tetrahydropyrano[3,2-b]pyrrol-2(1H)-one derivatives as anticancer agents

Design, synthesis, and qualitative structure-activity evaluations of novel β-secretase inhibitors as potential Alzheimer's drug leads.

Differential use of anhydropyranosides for enantiopure routes to bis-gamma-butyrolactones: a new approach to the frameworks of antibiotic and anticancer agents isoavenaciolide and ethisolide.

Divergent Strategy for Diastereocontrolled Synthesis of Small- and Medium-Ring Architectures

Domino Transformations of Ene/Yne Tethered Salicylaldehyde Derivatives: Pluripotent Platforms for the Construction of High sp3 Content and Privileged Architectures

Drug development post COVID-19 pandemic: toward a better system to meet current and future global health challenges

Epigenetics and miRNA as predictive markers and targets for lung cancer chemotherapy.

Flexible, polymer-supported synthesis of sphingosine derivatives provides ceramides with enhanced biological activity.

Modulation of DNA damage response and induction of apoptosis mediates synergism between doxorubicin and a new imidazopyridine derivative in breast and lung cancer cells.

Multidirectional desymmetrization of pluripotent building block en route to diastereoselective synthesis of complex nature-inspired scaffolds

Mutations in the nonstructural protein 3A confer resistance to the novel enterovirus replication inhibitor TTP-8307.

One-Pot Synthesis of Diverse Collections of Benzoxazepine and Indolopyrazine Fused to Heterocyclic Systems

Post Groebke-Blackburn multicomponent protocol: synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents.

Post-Ugi Cascade Transformations for Accessing Diverse Chromenopyrrole Collections.

Rational design and synthesis of potent dibenzazepine motifs as beta-secretase inhibitors

Sequencing [4 + 1]-Cycloaddition and Aza-Michael Addition Reactions: A Diastereoselective Cascade for the Rapid Access of Pyrido[2',1':2,3]/Thiazolo[2',3':2,3]imidazo[1,5-a]quinolone Scaffolds as Potential Antibacterial and Anticancer Motifs

Stereocontrolled transformations of cyclohexadienone derivatives to access stereochemically rich and natural product-inspired architectures

Structure activity relationship of phenolic acid inhibitors of α-synuclein fibril formation and toxicity

Superbugs but no drugs: steps in averting a post-antibiotic era

Synthesis and antimicrobial activity of cholic acid hydrazone analogues

Synthesis of a new series of heterocyclic scaffolds for medicinal purposes

Tandem Achmatowicz-Knoevenagel protocol: diastereoselective synthesis and anticancer evaluation of cyclopenta[b]pyrane derivatives ⬇️

Tandem multicomponent reactions toward the design and synthesis of novel antibacterial and cytotoxic motifs.