Lista de obras - Walter Cabri - Dominio Público Uruguay

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

artículo científico publicado en 2014

A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase.

artículo científico publicado en 2010

A translation of the twelve principles of green chemistry to guide the development of cross-coupling reactions

artículo científico publicado en 2022

Application of Af4-Multidetection to Liraglutide in Its Formulation: Preserving and Representing Native Aggregation

artículo científico publicado en 2022

Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors

artículo científico publicado en 2009

Benefits of a Mixed-Mode Stationary Phase to Address the Challenging Purification of an Industrially Relevant Peptide: A Proof-of-Concept Study

artículo científico publicado en 2022

Biotechnological lycopene production by mated fermentation of Blakeslea trispora

artículo científico publicado en 2004

Biotransformation of colchicinoids into their corresponding 3-O-glucosyl derivatives by selected strains of Bacillus megaterium

artículo científico publicado en 2014

Camptothecins in tumor homing via an RGD sequence mimetic.

artículo científico publicado en 2012

Cefdinir: A comparative study of anhydrous vs. monohydrate form. Microstructure and tabletting behaviour

artículo científico publicado en 2006

Combination of HPLC "inverted chirality columns approach" and MS/MS detection for extreme enantiomeric excess determination even in absence of reference samples. Application to camptothecin derivatives

scientific article published on 29 June 2007

Derivatives of R-aminocarnitine without ammonium moiety as liver carnitine palmitoyltransferase I (L-CPT I) inhibitors

scientific article published on 10 August 2011

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

artículo científico publicado en 2010

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

artículo científico publicado en 2012

Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.

artículo científico publicado en 2012

Effect of SAMITAL® in the treatment of chemotherapy-induced mucositis in adult oncohematological patients

artículo científico publicado en 2013

Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry

artículo científico publicado en 2011

Enol carbamates as inhibitors of fatty acid amide hydrolase (FAAH) endowed with high selectivity for FAAH over the other targets of the endocannabinoid system

artículo científico publicado en 2010

Evolution of an acylase active on cephalosporin C

artículo científico publicado en 2005

Extending the use of "Inverted Chirality Columns Approach" for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative.

artículo científico publicado en 2009

Fast Heck-Cassar-Sonogashira (HCS) Reactions in Green Solvents

artículo científico publicado en 2020

Ganoderma lucidum Ethanol Extracts Enhance Re-Epithelialization and Prevent Keratinocytes from Free-Radical Injury

scientific article published on 29 August 2020

Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives.

artículo científico

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

artículo científico publicado en 2012

Identification of impurities in artemisinin, their behavior in high performance liquid chromatography and implications for the quality of derived anti-malarial drugs

artículo científico publicado en 2011

Innovative chemical synthesis and conformational hints on the lipopeptide liraglutide.

artículo científico publicado en 2016

Investigating the Neuroprotective Effects of Turmeric Extract: Structural Interactions of β-Amyloid Peptide with Single Curcuminoids.

artículo científico publicado en 2016

Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors

artículo científico publicado en 2012

Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors

artículo científico publicado en 2013

Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography

artículo científico publicado en 2019

N-Hydroxy-(4-oxime)-cinnamide: a versatile scaffold for the synthesis of novel histone deacetylase [correction of deacetilase] (HDAC) inhibitors

artículo científico publicado en 2009

Natural Occurring and Engineered Enzymes for Peptide Ligation and Cyclization

artículo científico publicado en 2019

New retinoid derivatives as back-ups of Adarotene

artículo científico publicado en 2012

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

artículo científico publicado en 2010

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

artículo científico publicado el 23 de noviembre de 2011

Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study

artículo científico publicado en 2019

Novel substituted aminoalkylguanidines as potential antihyperglycemic and food intake-reducing agents

artículo científico publicado en 2008

Omega-alkoxy analogues of SAHA (vorinostat) as inhibitors of HDAC: a study of chain-length and stereochemical dependence.

artículo científico publicado en 2007

On-column epimerization of dihydroartemisinin: an effective analytical approach to overcome the shortcomings of the International Pharmacopoeia monograph.

artículo científico publicado en 2008

Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation.

artículo científico publicado en 2011

Polymorphisms and Patent, Market, and Legal Battles: Cefdinir Case Study

artículo científico publicado en 2007

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands

scientific article published on 07 May 2015

Production of peptides as generic drugs: a patent landscape of octreotide

artículo científico publicado en 2016

Protective effect of Panax ginseng in cisplatin-induced cachexia in rats.

artículo científico publicado en 2014

Reducing effect of the Chinese medicinal herb, Salvia miltiorrhiza, on alcohol self-administration in Sardinian alcohol-preferring rats

artículo científico publicado en 2014

SAMITAL®: a new botanical drug for the treatment of mucositis induced by oncological therapies.

artículo científico publicado en 2013

ST7612AA1, a thioacetate-ω(γ-lactam carboxamide) derivative selected from a novel generation of oral HDAC inhibitors

artículo científico publicado en 2014

Stereodynamic investigation of labile stereogenic centres in dihydroartemisinin.

artículo científico publicado en 2010

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive kinetic investigation. Part 2.

artículo científico publicado en 2011

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive thermodynamic investigation. Part 1.

artículo científico publicado en 2011

Synthesis and biological activity of fluorinated combretastatin analogues

artículo científico publicado en 2008

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

artículo científico publicado en 2013

Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.

artículo científico publicado en 2014

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

artículo científico publicado en 2013

Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties

scientific article published on 13 April 2014

Vorinostat-like molecules as structural, stereochemical, and pharmacological tools

artículo científico publicado en 2010

Lista de obras de Walter Cabri

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors

A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase.

A translation of the twelve principles of green chemistry to guide the development of cross-coupling reactions

Application of Af4-Multidetection to Liraglutide in Its Formulation: Preserving and Representing Native Aggregation

Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors

Benefits of a Mixed-Mode Stationary Phase to Address the Challenging Purification of an Industrially Relevant Peptide: A Proof-of-Concept Study

Biotechnological lycopene production by mated fermentation of Blakeslea trispora

Biotransformation of colchicinoids into their corresponding 3-O-glucosyl derivatives by selected strains of Bacillus megaterium

Camptothecins in tumor homing via an RGD sequence mimetic.

Cefdinir: A comparative study of anhydrous vs. monohydrate form. Microstructure and tabletting behaviour

Combination of HPLC "inverted chirality columns approach" and MS/MS detection for extreme enantiomeric excess determination even in absence of reference samples. Application to camptothecin derivatives

Derivatives of R-aminocarnitine without ammonium moiety as liver carnitine palmitoyltransferase I (L-CPT I) inhibitors

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.

Effect of SAMITAL® in the treatment of chemotherapy-induced mucositis in adult oncohematological patients

Efficient organic monoliths prepared by γ-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry

Enol carbamates as inhibitors of fatty acid amide hydrolase (FAAH) endowed with high selectivity for FAAH over the other targets of the endocannabinoid system

Evolution of an acylase active on cephalosporin C

Extending the use of "Inverted Chirality Columns Approach" for enantiomeric excess determination in absence of reference samples: Application to a water-soluble camptothecin derivative.

Fast Heck-Cassar-Sonogashira (HCS) Reactions in Green Solvents

Ganoderma lucidum Ethanol Extracts Enhance Re-Epithelialization and Prevent Keratinocytes from Free-Radical Injury

Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives.

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

Identification of impurities in artemisinin, their behavior in high performance liquid chromatography and implications for the quality of derived anti-malarial drugs

Innovative chemical synthesis and conformational hints on the lipopeptide liraglutide.

Investigating the Neuroprotective Effects of Turmeric Extract: Structural Interactions of β-Amyloid Peptide with Single Curcuminoids.

Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors

Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors

Modeling the nonlinear behavior of a bioactive peptide in reversed-phase gradient elution chromatography

N-Hydroxy-(4-oxime)-cinnamide: a versatile scaffold for the synthesis of novel histone deacetylase [correction of deacetilase] (HDAC) inhibitors

Natural Occurring and Engineered Enzymes for Peptide Ligation and Cyclization

New retinoid derivatives as back-ups of Adarotene

Non-natural macrocyclic inhibitors of histone deacetylases: design, synthesis, and activity.

Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90 ⬇️

Novel insights into the chemistry of an old medicine: A general degradative pathway for penicillins from a piperacillin/tazobactam stability study

Novel substituted aminoalkylguanidines as potential antihyperglycemic and food intake-reducing agents

Omega-alkoxy analogues of SAHA (vorinostat) as inhibitors of HDAC: a study of chain-length and stereochemical dependence.

On-column epimerization of dihydroartemisinin: an effective analytical approach to overcome the shortcomings of the International Pharmacopoeia monograph.

Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation.

Polymorphisms and Patent, Market, and Legal Battles: Cefdinir Case Study

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands

Production of peptides as generic drugs: a patent landscape of octreotide

Protective effect of Panax ginseng in cisplatin-induced cachexia in rats.

Reducing effect of the Chinese medicinal herb, Salvia miltiorrhiza, on alcohol self-administration in Sardinian alcohol-preferring rats

SAMITAL®: a new botanical drug for the treatment of mucositis induced by oncological therapies.

ST7612AA1, a thioacetate-ω(γ-lactam carboxamide) derivative selected from a novel generation of oral HDAC inhibitors

Stereodynamic investigation of labile stereogenic centres in dihydroartemisinin.

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive kinetic investigation. Part 2.

Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive thermodynamic investigation. Part 1.

Synthesis and biological activity of fluorinated combretastatin analogues

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

Synthesis and evaluation of new Hsp90 inhibitors based on a 1,4,5-trisubstituted 1,2,3-triazole scaffold.

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties

Vorinostat-like molecules as structural, stereochemical, and pharmacological tools