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Lista de obras de Andrew S Murkin

A beta-fluoroamine inhibitor of purine nucleoside phosphorylase

artículo científico publicado en 2008

Alteration of the Flexible Loop in 1-Deoxy- d -xylulose-5-phosphate Reductoisomerase Boosts Enthalpy-Driven Inhibition by Fosmidomycin

artículo científico publicado en 2014

Arsenate and phosphate as nucleophiles at the transition states of human purine nucleoside phosphorylase

artículo científico publicado en 2011

Azetidine based transition state analogue inhibitors of N-ribosyl hydrolases and phosphorylases

artículo científico publicado en 2008

Commentary: Ohm's law as an analogy for enzyme kinetics

artículo científico publicado en 2015

Cysteine is the general base that serves in catalysis by isocitrate lyase and in mechanism-based inhibition by 3-nitropropionate

artículo científico publicado en 2013

DXP Reductoisomerase: Reaction of the Substrate in Pieces Reveals a Catalytic Role for the Nonreacting Phosphodianion Group

artículo científico publicado el 20 de marzo de 2013

Dehydroalanine-based inhibition of a peptide epimerase from spider venom

artículo científico publicado en 2002

Femtosecond dynamics coupled to chemical barrier crossing in a Born-Oppenheimer enzyme

artículo científico publicado en 2011

Highly precise measurement of kinetic isotope effects using 1H-detected 2D [13C,1H]-HSQC NMR spectroscopy

scientific article published in 2012

Identification of three classes of heteroaromatic compounds with activity against intracellular Trypanosoma cruzi by chemical library screening

artículo científico publicado en 2009

Immucillins in custom catalytic-site cavities

artículo científico publicado en 2008

Inverse Solvent Isotope Effects in Enzyme-Catalyzed Reactions

scientific article published on 21 April 2020

Mechanism and inhibition of 1-deoxy-D-xylulose-5-phosphate reductoisomerase

artículo científico

Mechanism-based inactivator of isocitrate lyases 1 and 2 from Mycobacterium tuberculosis.

artículo científico publicado en 2017

Neighboring Group Participation in the Transition State of Human Purine Nucleoside Phosphorylase †

artículo científico publicado en 2007

New Electrophiles and Strategies for Mechanism-Based and Targeted Covalent Inhibitor Design

artículo científico publicado en 2019

Phosphate activation in the ground state of purine nucleoside phosphorylase.

artículo científico publicado en 2006

Plasmodium falciparum parasites are killed by a transition state analogue of purine nucleoside phosphorylase in a primate animal model

artículo científico publicado en 2011

Pre-steady-state kinetic analysis of 1-deoxy-D-xylulose-5-phosphate reductoisomerase from Mycobacterium tuberculosis reveals partially rate-limiting product release by parallel pathways.

artículo científico publicado en 2012

Ribocation transition state capture and rebound in human purine nucleoside phosphorylase

artículo científico publicado en 2009

The Nitro Group as a Masked Electrophile in Covalent Enzyme Inhibition

scientific article published on 23 May 2018

The role of phosphate in a multistep enzymatic reaction: reactions of the substrate and intermediate in pieces

artículo científico publicado en 2015

Third-generation immucillins: syntheses and bioactivities of acyclic immucillin inhibitors of human purine nucleoside phosphorylase

artículo científico publicado en 2009

Transition state analogue discrimination by related purine nucleoside phosphorylases

artículo científico publicado en 2006

Transition-state interactions revealed in purine nucleoside phosphorylase by binding isotope effects

artículo científico publicado en 2008

l -Enantiomers of Transition State Analogue Inhibitors Bound to Human Purine Nucleoside Phosphorylase

artículo científico publicado en 2008