Lista de obras - Giuseppe Caliendo - Dominio Público Uruguay

5-Amino-2-hydroxybenzoic Acid 4-(5-Thioxo-5H-[1,2]dithiol-3yl)-phenyl Ester (ATB-429), a Hydrogen Sulfide-Releasing Derivative of Mesalamine, Exerts Antinociceptive Effects in a Model of Postinflammatory Hypersensitivity

artículo científico publicado en 2006

5-HT(1A) receptor: an old target as a new attractive tool in drug discovery from central nervous system to cancer

artículo científico publicado en 2013

A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold

A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT(1A) receptor ligands.

artículo científico publicado en 2002

A convenient synthesis of N-Fmoc-N,N′-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N′-bis-Boc-7-guanyl-Tic-OH, GTIC)

A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.

artículo científico publicado en 2009

A suitable 1,2,4-oxadiazoles synthesis by microwave irradiation

artículo científico publicado en 2004

Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies.

artículo científico publicado en 2004

Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs

artículo científico publicado en 2007

Conformational analysis of three NK1 tripeptide antagonists: a proton nuclear magnetic resonance study

artículo científico publicado en 1997

Derivatives as 5HT1A receptor ligands--past and present.

artículo científico publicado en 2005

Design of Inhibitors for Human Tissue Kallikrein Using Non-Natural Aromatic and Basic Amino Acids

artículo científico publicado en 2002

Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents.

artículo científico publicado en 2017

Efficient microwave combinatorial parallel and nonparallel synthesis of N-alkylated glycine methyl esters as peptide building blocks.

artículo científico publicado en 2005

Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands.

artículo científico publicado en 2009

Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis

artículo científico publicado en 2007

Evidence for a protective role played by the Na+/Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats

artículo científico publicado en 2004

Gastrointestinal Safety and Anti-Inflammatory Effects of a Hydrogen Sulfide–Releasing Diclofenac Derivative in the Rat

artículo científico publicado en 2006

Identification of a pepducin acting as S1P3 receptor antagonist.

artículo científico publicado en 2013

In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives

artículo científico publicado en 2006

Kallikrein protease activated receptor (PAR) axis: an attractive target for drug development

artículo científico publicado en 2012

Markedly reduced toxicity of a hydrogen sulphide-releasing derivative of naproxen (ATB-346).

artículo científico publicado en 2010

Minimal structural requirements for agonist activity of PAR-2 activating peptides.

artículo científico publicado en 2002

Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage

artículo científico publicado en 2012

Nevirapine quantification in human plasma by high-performance liquid chromatography coupled to electrospray tandem mass spectrometry. Application to bioequivalence study.

artículo científico publicado en 2002

New 5-HT(1A) receptor ligands containing a N'-cyanoisonicotinamidine nucleus: synthesis and in vitro pharmacological evaluation

artículo científico publicado en 2010

New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: synthesis and in vitro pharmacological evaluation.

artículo científico publicado en 2005

New potent 5-HT2A receptor ligands containing an N′-cyanopicolinamidine nucleus: Synthesis and in vitro pharmacological evaluation

artículo científico publicado en 2011

Nitric Oxide Related Therapeutic Phenomenon: A Challenging Task

artículo científico publicado en 2002

PAR1 antagonism protects against experimental liver fibrosis. Role of proteinase receptors in stellate cell activation

artículo científico publicado en 2004

Peptide T revisited: conformational mimicry of epitopes of anti-HIV proteins

artículo científico publicado en 2001

Perfusion of rat colon with sennosides, rhein and rheinanthrone. Concentration-related histamine release

artículo científico publicado en 1990

Pharmacokinetics of dihydroergocristine and its major metabolite 8'-hydroxy-dihydroergocristine in human plasma

artículo científico publicado en 2005

Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists.

artículo científico publicado en 2001

Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity

artículo científico publicado en 1999

S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids

artículo científico publicado en 2001

Specificity studies on Kallikrein-related peptidase 7 (KLK7) and effects of osmolytes and glycosaminoglycans on its peptidase activity.

artículo científico publicado en 2014

Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes

Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation

artículo científico publicado en 2019

Synthesis and antiinflammatory—analgesic profile of 1-methyl-2-(4-X-benzoyl) imidazole-5-carboxylic acids

article published in 1995

Synthesis and antimicrobial activities of 5-amidobenzotriazole derivatives

Synthesis and antinociceptive activity of peptides related to interleukin-1 beta 193-195 Lys-Pro-Thr

scientific article published on 01 January 1996

Synthesis and biological activity of benzotriazole derivatives structurally related to trazodone

Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.

artículo científico publicado en 1999

Synthesis and biological activity of tripeptide FR113680 analogues containing unconventional amino acids.

artículo científico publicado en 1995

Synthesis and biological effects of hydrogen sulfide (H2S): development of H2S-releasing drugs as pharmaceuticals

artículo científico publicado en 2010

Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with the general structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X.

artículo científico publicado en 2001

Synthesis and in vitro pharmacological evaluation of novel 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands

artículo científico publicado en 2014

Synthesis and in-vitro pharmacological evaluation of new 5-HT1A receptor ligands containing a benzotriazinone nucleus.

artículo científico publicado en 2008

Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides.

artículo científico publicado en 1997

Synthesis and pharmacological evaluation of a set of N-[2-(alkylamino)ethyl]benzotriazol-X-yl isobutyramides acting as local anesthetics

scholarly article by Giuseppe Caliendo et al published January 1996 in European Journal of Medicinal Chemistry

Synthesis and pharmacological evaluation of peptide-mimetic protease-activated receptor-1 antagonists containing novel heterocyclic scaffolds.

artículo científico publicado en 2008

Synthesis and pharmacological evaluations of sildenafil analogues for treatment of erectile dysfunction.

artículo científico publicado en 2008

Synthesis and structure-activity relationships of antiinflammatory 1-methyl-2-(4-X-benzoyl)imidazole-5-acetic acids

Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers

artículo científico publicado en 2002

Synthesis by microwave irradiation and antidiarrhoeal activity of benzotriazinone and saccharine derivatives

artículo científico publicado en 2005

Synthesis by microwave irradiation and binding properties of novel 5-HT(1A) receptor ligands

artículo científico publicado en 2001

Synthesis of 1-naphtylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents

scientific article published on 08 March 2011

Synthesis of 2-Methyl-3-indolylacetic Derivatives as Anti-Inflammatory Agents That Inhibit Preferentially Cyclooxygenase 1 without Gastric Damage

artículo científico publicado en 2006

Synthesis of benzamide derivatives and their evaluation as antiprion agents

artículo científico publicado en 2012

Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands

scientific article published on 01 March 2000

Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV.

artículo científico publicado en 2001

Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage

artículo científico publicado en 2001

Synthesis ofN α-FmocN,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC)

article

Synthesis, antimicrobial data and correlation analysis in a set of 2-alkyl-5-amidobenzotriazoles

Synthesis, biological evaluation, and docking studies of PAR2-AP-derived pseudopeptides as inhibitors of kallikrein 5 and 6

artículo científico publicado en 2015

Synthesis, local anesthetic activity and QSAR studies for a set of N-[2-(alkylamino)ethyl]benzotriazol-x-yl acetamides

Synthesis, pharmacological evaluation, and molecular modeling studies of novel peptidic CAAX analogues as farnesyl-protein-transferase inhibitors

artículo científico publicado en 2006

Lista de obras de Giuseppe Caliendo

5-Amino-2-hydroxybenzoic Acid 4-(5-Thioxo-5H-[1,2]dithiol-3yl)-phenyl Ester (ATB-429), a Hydrogen Sulfide-Releasing Derivative of Mesalamine, Exerts Antinociceptive Effects in a Model of Postinflammatory Hypersensitivity

5-HT(1A) receptor: an old target as a new attractive tool in drug discovery from central nervous system to cancer

A convenient strategy of dimerization by microwave heating and using 2,5-diketopiperazine as scaffold

A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT(1A) receptor ligands.

A convenient synthesis of N-Fmoc-N,N′-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N′-bis-Boc-7-guanyl-Tic-OH, GTIC)

A nitro-arginine derivative of trimebutine (NO2-Arg-Trim) attenuates pain induced by colorectal distension in conscious rats.

A suitable 1,2,4-oxadiazoles synthesis by microwave irradiation

Bromazepam determination in human plasma by high-performance liquid chromatography coupled to tandem mass spectrometry: a highly sensitive and specific tool for bioequivalence studies.

Conformation-activity relationship of peptide T and new pseudocyclic hexapeptide analogs

Conformational analysis of three NK1 tripeptide antagonists: a proton nuclear magnetic resonance study

Derivatives as 5HT1A receptor ligands--past and present.

Design of Inhibitors for Human Tissue Kallikrein Using Non-Natural Aromatic and Basic Amino Acids

Development of 1,2,3-Triazole-Based Sphingosine Kinase Inhibitors and Their Evaluation as Antiproliferative Agents.

Efficient microwave combinatorial parallel and nonparallel synthesis of N-alkylated glycine methyl esters as peptide building blocks.

Efficient microwave combinatorial synthesis of novel indolic arylpiperazine derivatives as serotoninergic ligands.

Enhanced activity of a hydrogen sulphide-releasing derivative of mesalamine (ATB-429) in a mouse model of colitis

Evidence for a protective role played by the Na+/Ca2+ exchanger in cerebral ischemia induced by middle cerebral artery occlusion in male rats

Gastrointestinal Safety and Anti-Inflammatory Effects of a Hydrogen Sulfide–Releasing Diclofenac Derivative in the Rat

Identification of a pepducin acting as S1P3 receptor antagonist.

In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives

Kallikrein protease activated receptor (PAR) axis: an attractive target for drug development

Markedly reduced toxicity of a hydrogen sulphide-releasing derivative of naproxen (ATB-346).

Minimal structural requirements for agonist activity of PAR-2 activating peptides.

Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage

Nevirapine quantification in human plasma by high-performance liquid chromatography coupled to electrospray tandem mass spectrometry. Application to bioequivalence study.

New 5-HT(1A) receptor ligands containing a N'-cyanoisonicotinamidine nucleus: synthesis and in vitro pharmacological evaluation

New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: synthesis and in vitro pharmacological evaluation.

New potent 5-HT2A receptor ligands containing an N′-cyanopicolinamidine nucleus: Synthesis and in vitro pharmacological evaluation

Nitric Oxide Related Therapeutic Phenomenon: A Challenging Task

PAR1 antagonism protects against experimental liver fibrosis. Role of proteinase receptors in stellate cell activation

Peptide T revisited: conformational mimicry of epitopes of anti-HIV proteins

Perfusion of rat colon with sennosides, rhein and rheinanthrone. Concentration-related histamine release

Pharmacokinetics of dihydroergocristine and its major metabolite 8'-hydroxy-dihydroergocristine in human plasma

Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists.

Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity

S1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids

Specificity studies on Kallikrein-related peptidase 7 (KLK7) and effects of osmolytes and glycosaminoglycans on its peptidase activity.

Structure—affinity relationship studies on benzotriazole derivatives binding to 5-HT receptor subtypes

Synthesis and Pharmacological Screening of Pyridopyrimidines as Effective Anti-Diarrheal Agents through the Suppression of Cyclic Nucleotide Accumulation

Synthesis and antiinflammatory—analgesic profile of 1-methyl-2-(4-X-benzoyl) imidazole-5-carboxylic acids

Synthesis and antimicrobial activities of 5-amidobenzotriazole derivatives

Synthesis and antinociceptive activity of peptides related to interleukin-1 beta 193-195 Lys-Pro-Thr

Synthesis and biological activity of benzotriazole derivatives structurally related to trazodone

Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids.

Synthesis and biological activity of tripeptide FR113680 analogues containing unconventional amino acids.

Synthesis and biological effects of hydrogen sulfide (H2S): development of H2S-releasing drugs as pharmaceuticals

Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with the general structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X.

Synthesis and in vitro pharmacological evaluation of novel 2-hydroxypropyl-4-arylpiperazine derivatives as serotoninergic ligands

Synthesis and in-vitro pharmacological evaluation of new 5-HT1A receptor ligands containing a benzotriazinone nucleus.

Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides.

Synthesis and pharmacological evaluation of a set of N-[2-(alkylamino)ethyl]benzotriazol-X-yl isobutyramides acting as local anesthetics

Synthesis and pharmacological evaluation of peptide-mimetic protease-activated receptor-1 antagonists containing novel heterocyclic scaffolds.

Synthesis and pharmacological evaluations of sildenafil analogues for treatment of erectile dysfunction.

Synthesis and structure-activity relationships of antiinflammatory 1-methyl-2-(4-X-benzoyl)imidazole-5-acetic acids

Synthesis and vasorelaxant activity of new 1,4-benzoxazine derivatives potassium channel openers

Synthesis by microwave irradiation and antidiarrhoeal activity of benzotriazinone and saccharine derivatives

Synthesis by microwave irradiation and binding properties of novel 5-HT(1A) receptor ligands

Synthesis of 1-naphtylpiperazine derivatives as serotoninergic ligands and their evaluation as antiproliferative agents

Synthesis of 2-Methyl-3-indolylacetic Derivatives as Anti-Inflammatory Agents That Inhibit Preferentially Cyclooxygenase 1 without Gastric Damage

Synthesis of benzamide derivatives and their evaluation as antiprion agents

Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands

Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV.

Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage

Synthesis ofN α-FmocN,N′-bis-Boc-5-, 6- and 8-guanyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic Acid (5-GTIC, 6-GTIC and 8-GTIC)

Synthesis, antimicrobial data and correlation analysis in a set of 2-alkyl-5-amidobenzotriazoles

Synthesis, biological evaluation, and docking studies of PAR2-AP-derived pseudopeptides as inhibitors of kallikrein 5 and 6

Synthesis, local anesthetic activity and QSAR studies for a set of N-[2-(alkylamino)ethyl]benzotriazol-x-yl acetamides

Synthesis, pharmacological evaluation, and molecular modeling studies of novel peptidic CAAX analogues as farnesyl-protein-transferase inhibitors