Lista de obras - Gerardo Burton - Dominio Público Uruguay

13C NMR studies of glycolysis in intra- and extra-erythrocytic Babesia microti

artículo científico publicado en 1984

18,20-Hemiacetal-type and Other Withanolides fromDunaliabrachyacantha

artículo científico publicado en 1999

27-Nor-Δ(4)-dafachronic acid is a synthetic ligand of Caenorhabditis elegans DAF-12 receptor

artículo científico publicado en 2013

6,19-Sulfur-bridged progesterone analogues with antiimmunosuppressive activity

artículo científico publicado en 2005

6,19-carbon-bridged steroids. Synthesis of 6,19-methanoprogesterone

artículo científico publicado en 2003

7-Hydroxywithanolides from datura ferox

scientific article published on 01 July 1999

A highly lipophilic form of aldosterone. Isolation and characterization of an aldosterone dimer

artículo científico publicado en 1985

A rapid direct assay for uroporphyrinogen III cosynthetase

scientific article published on 01 June 1980

Allopregnanolone (3alpha-hydroxy-5alpha-pregnan-20-one) derivatives with a polar chain in position 16alpha: synthesis and activity

artículo científico publicado en 2009

Antifeedant activity of withanolides from Salpichroa origanifolia on Musca domestica

artículo científico publicado en 2000

Antioxidant properties in a non-polar environment of difluoromethyl bioisosteres of methyl hydroxycinnamates.

artículo científico publicado en 2016

Biological activity and ligand binding mode to the progesterone receptor of A-homo analogues of progesterone

artículo científico publicado en 2011

C(16)-C(22) oxygen-bridged analogues of ceDAF-12 and LXR ligands.

artículo científico publicado en 2016

Destabilization of the torsioned conformation of a ligand side chain inverts the LXRβ activity.

artículo científico publicado en 2015

Development of beta-lapachone prodrugs for therapy against human cancer cells with elevated NAD(P)H:quinone oxidoreductase 1 levels.

artículo científico publicado en 2005

Dissociation of glucocorticoid effects of C-21 steroids at high concentrations in thymocytes

scientific article published on 01 June 1983

Effect of synthetic steroids on GABAA receptor binding in rat brain

artículo científico publicado en 2015

Eighteen-deoxyaldosterone and other less polar forms of 18-hydroxycorticosterone as aldosterone precursors in rat adrenals

article by E N Cozza et al published 1 May 1985 in The Journal of Steroid Biochemistry

Exploring the molecular basis of action of ring D aromatic steroidal antiestrogens.

artículo científico publicado en 2015

Features of the shuttle pair 11 beta-hydroxyprogesterone-11-ketoprogesterone

scientific article published on 01 April 1997

Fluorinated oxysterol analogues: Synthesis, molecular modelling and LXRβ activity.

artículo científico publicado en 2016

Hemisuccinate of 21-hydroxy-6,19-epoxyprogesterone: a tissue-specific modulator of the glucocorticoid receptor

artículo científico publicado en 2008

Induction of quinone reductase by withanolides.

artículo científico publicado en 2002

Influence of calf serum on glucocorticoid-responses of certain progesterone derivatives

artículo científico publicado en 1998

Inhibition of thymocyte RNA synthesis by natural adrenal steroids and their 1,4-diene analogs. Structure-activity correlations using 13C-n.m.r. spectroscopy

scientific article published on 01 December 1981

Insights on glucocorticoid receptor activity modulation through the binding of rigid steroids

artículo científico publicado en 2010

Intramolecular PhI=O mediated copper-catalyzed aziridination of unsaturated sulfamates: a new direct access to polysubstituted amines from simple homoallylic alcohols

scientific article published on 01 July 2002

Live cell imaging unveils multiple domain requirements for in vivo dimerization of the glucocorticoid receptor

artículo científico publicado en 2014

Mapping the Dynamics of the Glucocorticoid Receptor within the Nuclear Landscape.

artículo científico publicado en 2017

Microwave assisted preparation of C1-C11 oxygen-bridged pregnanes

artículo científico publicado en 2011

Modification of an essential amino group in the mineralocorticoid receptor evidences a differential conformational change of the receptor protein upon binding of antagonists, natural agonists and the synthetic agonist 11,19-oxidoprogesterone.

artículo científico publicado en 2002

Neuroprotective action of synthetic steroids with oxygen bridge. Activity on GABAA receptor.

artículo científico publicado en 2013

New Hydroxylated Withanolides from Salpichroa origanifolia

scientific article published on 01 March 1998

New lead compounds in the search for pure antiglucocorticoids and the dissociation of antiglucocorticoid effects.

artículo científico publicado en 2009

Oxidative Cyclization of Iodo Ketones. Synthesis of 6-Oxa-5alpha-pregnane-3,20-dione

scientific article published on 01 September 1996

Phytotoxic withanolides from Jaborosa rotacea ⬇️

scientific article published on 01 May 2006

Preparation and cytotoxicity toward cancer cells of mono(arylimino) derivatives of beta-lapachone

artículo científico publicado en 2001

QSAR on antiproliferative naphthoquinones based on a conformation-independent approach

artículo científico publicado en 2014

Response of Tribolium castaneum (Coleoptera, Tenebrionidae) to Salpichroa origanifolia Withanolides

artículo científico publicado en 2002

Sesquiterpene lactone variability in Parthenium hysterophorus L ⬇️

artículo científico publicado en 2000

Spiranoid withanolides from Jaborosa odonelliana

artículo científico publicado en 2002

Structure of the glucocorticoid receptor, a flexible protein that can adapt to different ligands.

scientific article published on May 2010

Synthesis and GABA(A) receptor activity of 2,19-sulfamoyl analogues of allopregnanolone

artículo científico publicado en 2009

Synthesis and GABA(A) receptor activity of 6-oxa-analogs of neurosteroids

scientific article published on 01 June 2000

Synthesis and GABA(A) receptor activity of a 6,19-oxido analogue of pregnanolone

artículo científico publicado en 2003

Synthesis and GABA(A) receptor activity of oxygen-bridged neurosteroid analogs

artículo científico publicado en 2008

Synthesis and GABAA receptor activity of A-homo analogues of neuroactive steroids.

artículo científico publicado en 2010

Synthesis and activity evaluation of a series of cholanamides as modulators of the liver X receptors.

artículo científico publicado en 2018

Synthesis and antifungal activity of C-21 steroids with an aromatic D ring

artículo científico publicado en 2013

Synthesis and biological evaluation of salpichrolide analogs as antiestrogenic agents.

artículo científico publicado en 2014

Synthesis of 21-hydroxy-11,19-oxidopregn-4-ene-3,20-dione and 21-hydroxy-6,19-oxidopregn-4-ene-3,20-dione

artículo científico publicado en 1995

Synthesis of 3beta-hydroxy-5-cholenic acid from 3beta-hydroxy-5-pregnen-20-one aimed at the preparation of lebelled steroid compounds

artículo científico publicado en 1977

Synthesis of 6,19-cyclopregnanes. Constrained analogues of steroid hormones

artículo científico publicado en 2007

Synthesis of 6,19-sulfamidate bridged pregnanes

artículo científico publicado en 2005

Synthesis of 6-azaprogesterone and 19-hydroxy-6-azasteroids

scientific article published on 02 November 2012

Synthesis of oxido-bridged analogs of 18-hydroxyprogesterone

artículo científico publicado en 1996

Synthetic DAF-12 modulators with potential use in controlling the nematode life cycle

artículo científico publicado en 2015

The Caenorhabditis elegans DAF-12 nuclear receptor: structure, dynamics, and interaction with ligands

scientific article published on 10 May 2012

The glucocorticoid properties of the synthetic steroid pregna-1,4-diene-11beta-ol-3,20-dione (deltaHOP) are not entirely correlated with the steroid binding to the glucocorticoid receptor

artículo científico publicado en 1999

The rigid steroid 21-hydroxy-6,19-epoxyprogesterone (21OH-6,19OP) is a dissociated glucocorticoid receptor modulator potentially useful as a novel coadjuvant in breast cancer chemotherapy.

artículo científico publicado en 2014

Withanolides and Related Steroids ⬇️

artículo científico publicado el 1 de enero de 2011

Withanolides from Jaborosa laciniata

artículo científico publicado en 2007

Withanolides from Salpichroa origanifolia

artículo científico publicado en 2001

Withanolides from Vassobia lorentzii ⬇️

artículo científico publicado en 2000

Withanolides with phytotoxic activity from Jaborosa caulescens var. caulescens and J. caulescens var. bipinnatifida 1

scientific article published on 12 April 2007

Lista de obras de Gerardo Burton

13C NMR studies of glycolysis in intra- and extra-erythrocytic Babesia microti

18,20-Hemiacetal-type and Other Withanolides fromDunaliabrachyacantha

27-Nor-Δ(4)-dafachronic acid is a synthetic ligand of Caenorhabditis elegans DAF-12 receptor

6,19-Sulfur-bridged progesterone analogues with antiimmunosuppressive activity

6,19-carbon-bridged steroids. Synthesis of 6,19-methanoprogesterone

7-Hydroxywithanolides from datura ferox

A highly lipophilic form of aldosterone. Isolation and characterization of an aldosterone dimer

A rapid direct assay for uroporphyrinogen III cosynthetase

Allopregnanolone (3alpha-hydroxy-5alpha-pregnan-20-one) derivatives with a polar chain in position 16alpha: synthesis and activity

Antifeedant activity of withanolides from Salpichroa origanifolia on Musca domestica

Antioxidant properties in a non-polar environment of difluoromethyl bioisosteres of methyl hydroxycinnamates.

Biological activity and ligand binding mode to the progesterone receptor of A-homo analogues of progesterone

C(16)-C(22) oxygen-bridged analogues of ceDAF-12 and LXR ligands.

Destabilization of the torsioned conformation of a ligand side chain inverts the LXRβ activity.

Development of beta-lapachone prodrugs for therapy against human cancer cells with elevated NAD(P)H:quinone oxidoreductase 1 levels.

Dissociation of glucocorticoid effects of C-21 steroids at high concentrations in thymocytes

Effect of synthetic steroids on GABAA receptor binding in rat brain

Eighteen-deoxyaldosterone and other less polar forms of 18-hydroxycorticosterone as aldosterone precursors in rat adrenals

Exploring the molecular basis of action of ring D aromatic steroidal antiestrogens.

Features of the shuttle pair 11 beta-hydroxyprogesterone-11-ketoprogesterone

Fluorinated oxysterol analogues: Synthesis, molecular modelling and LXRβ activity.

Hemisuccinate of 21-hydroxy-6,19-epoxyprogesterone: a tissue-specific modulator of the glucocorticoid receptor

Induction of quinone reductase by withanolides.

Influence of calf serum on glucocorticoid-responses of certain progesterone derivatives

Inhibition of thymocyte RNA synthesis by natural adrenal steroids and their 1,4-diene analogs. Structure-activity correlations using 13C-n.m.r. spectroscopy

Insights on glucocorticoid receptor activity modulation through the binding of rigid steroids

Intramolecular PhI=O mediated copper-catalyzed aziridination of unsaturated sulfamates: a new direct access to polysubstituted amines from simple homoallylic alcohols

Live cell imaging unveils multiple domain requirements for in vivo dimerization of the glucocorticoid receptor

Mapping the Dynamics of the Glucocorticoid Receptor within the Nuclear Landscape.

Microwave assisted preparation of C1-C11 oxygen-bridged pregnanes

Modification of an essential amino group in the mineralocorticoid receptor evidences a differential conformational change of the receptor protein upon binding of antagonists, natural agonists and the synthetic agonist 11,19-oxidoprogesterone.

Neuroprotective action of synthetic steroids with oxygen bridge. Activity on GABAA receptor.

New Hydroxylated Withanolides from Salpichroa origanifolia

New lead compounds in the search for pure antiglucocorticoids and the dissociation of antiglucocorticoid effects.

Oxidative Cyclization of Iodo Ketones. Synthesis of 6-Oxa-5alpha-pregnane-3,20-dione

Phytotoxic withanolides from Jaborosa rotacea ⬇️

Preparation and cytotoxicity toward cancer cells of mono(arylimino) derivatives of beta-lapachone

QSAR on antiproliferative naphthoquinones based on a conformation-independent approach

Response of Tribolium castaneum (Coleoptera, Tenebrionidae) to Salpichroa origanifolia Withanolides

Sesquiterpene lactone variability in Parthenium hysterophorus L ⬇️

Spiranoid withanolides from Jaborosa odonelliana

Structure of the glucocorticoid receptor, a flexible protein that can adapt to different ligands.

Synthesis and GABA(A) receptor activity of 2,19-sulfamoyl analogues of allopregnanolone

Synthesis and GABA(A) receptor activity of 6-oxa-analogs of neurosteroids

Synthesis and GABA(A) receptor activity of a 6,19-oxido analogue of pregnanolone

Synthesis and GABA(A) receptor activity of oxygen-bridged neurosteroid analogs

Synthesis and GABAA receptor activity of A-homo analogues of neuroactive steroids.

Synthesis and activity evaluation of a series of cholanamides as modulators of the liver X receptors.

Synthesis and antifungal activity of C-21 steroids with an aromatic D ring

Synthesis and biological evaluation of salpichrolide analogs as antiestrogenic agents.

Synthesis of 21-hydroxy-11,19-oxidopregn-4-ene-3,20-dione and 21-hydroxy-6,19-oxidopregn-4-ene-3,20-dione

Synthesis of 3beta-hydroxy-5-cholenic acid from 3beta-hydroxy-5-pregnen-20-one aimed at the preparation of lebelled steroid compounds

Synthesis of 6,19-cyclopregnanes. Constrained analogues of steroid hormones

Synthesis of 6,19-sulfamidate bridged pregnanes

Synthesis of 6-azaprogesterone and 19-hydroxy-6-azasteroids

Synthesis of oxido-bridged analogs of 18-hydroxyprogesterone

Synthetic DAF-12 modulators with potential use in controlling the nematode life cycle

The Caenorhabditis elegans DAF-12 nuclear receptor: structure, dynamics, and interaction with ligands

The glucocorticoid properties of the synthetic steroid pregna-1,4-diene-11beta-ol-3,20-dione (deltaHOP) are not entirely correlated with the steroid binding to the glucocorticoid receptor

The rigid steroid 21-hydroxy-6,19-epoxyprogesterone (21OH-6,19OP) is a dissociated glucocorticoid receptor modulator potentially useful as a novel coadjuvant in breast cancer chemotherapy.

Withanolides and Related Steroids ⬇️

Withanolides from Jaborosa laciniata

Withanolides from Salpichroa origanifolia

Withanolides from Vassobia lorentzii ⬇️

Withanolides with phytotoxic activity from Jaborosa caulescens var. caulescens and J. caulescens var. bipinnatifida 1