Lista de obras - Benoit Crousse - Dominio Público Uruguay

(19)F NMR monitoring of the eukaryotic 20S proteasome chymotrypsin-like activity: an investigative tool for studying allosteric regulation

artículo científico publicado en 2014

A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime.

artículo científico publicado en 2013

Access to novel amino trifluoromethyl cyclopropane carboxylic acid derivatives

Access to novel functionalized trifluoromethyl β-lactams by ring expansion of aziridines

Aminocyclopropanes as precursors of endoperoxides with antimalarial activity ⬇️

artículo científico publicado el 11 de octubre de 2010

Analogues of key precursors of aspartyl protease inhibitors: synthesis of trifluoromethyl amino epoxides

artículo científico publicado en 2005

Benefits of a Dual Chemical and Physical Activation: Direct aza-Michael Addition of Anilines Promoted by Solvent Effect under High Pressure

article

Bisulfate Salt-Catalyzed Friedel-Crafts Benzylation of Arenes with Benzylic Alcohols

artículo científico publicado en 2018

Carbonylhydrazide-based molecular tongs inhibit wild-type and mutated HIV-1 protease dimerization

artículo científico publicado en 2012

Designed Glycopeptidomimetics Disrupt Protein-Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability.

artículo científico publicado en 2016

Electrophilic amination of fluoroalkyl groups on azodicarboxylate derivatives.

artículo científico publicado en 2015

Facile ring opening of oxiranes with aromatic amines in fluoro alcohols

scientific article published on 01 October 2000

First synthesis of 10 alpha-(trifluoromethyl)deoxoartemisinin

scientific article published on 01 March 2002

Fluorinated Alcohols: A New Medium for Selective and Clean Reaction

Fluoro artemisinins: difluoromethylene ketones

artículo científico publicado en 2001

Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.

artículo científico publicado en 2004

Fluorous 4-N,N-dimethylaminopyridine (DMAP) salts as simple recyclable acylation catalysts

artículo científico publicado en 2010

Fluorous tagging of DABCO through halogen bonding: recyclable catalyst for the Morita-Baylis-Hillman reaction

artículo científico publicado en 2011

In vitro antileishmanial activity of fluoro-artemisinin derivatives against Leishmania donovani

artículo científico publicado en 2008

Influence of the structure of polyfluorinated alcohols on Brønsted acidity/hydrogen-bond donor ability and consequences on the promoter effect

artículo científico publicado en 2011

Intramolecular Pd-catalyzed carbocyclization, Heck reactions, and aryl-radical cyclizations with planar chiral arene tricarbonyl chromium complexes

artículo científico publicado en 2001

N-Difluoromethyl-triazole as a constrained scaffold in peptidomimetics

artículo científico publicado en 2017

Non Lewis acid catalysed epoxide ring opening with amino acid esters.

artículo científico publicado en 2009

Nonmetal catalyzed insertion reactions of diazocarbonyls to acid derivatives in fluorinated alcohols

artículo científico publicado en 2011

Novel [1,2]- and [2,3]-Wittig rearrangements of alpha-benzyloxy beta-CF(3)-beta-lactam enolates

scientific article published on 01 August 2001

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin

artículo científico publicado en 2004

Preparation of 10-trifluoromethyl artemether and artesunate. Influence of hexafluoropropan-2-ol on substitution reaction

artículo científico publicado en 2003

Reactivity of carbon dioxide in hydrofluoroethers: a facile access to cyclic carbonates

artículo científico publicado en 2015

Regioselective Halogenation of Arenes and Heterocycles in Hexafluoroisopropanol

artículo científico publicado en 2017

S(N)/S(N)' competition: selective access to new 10-fluoro artemisinins.

artículo científico publicado en 2006

Solubility switch of gold nanoparticles through hydrogen bond association

artículo científico publicado en 2008

Solvent-promoted and -controlled aza-Michael reaction with aromatic amines.

artículo científico publicado en 2009

Stereoselective Barbier-type allylation reaction of trifluoromethyl aldimines

artículo científico publicado en 2003

Structure-activity relationships of sugar-based peptidomimetics as modulators of amyloid β-peptide early oligomerization and fibrillization

artículo científico publicado en 2014

Synthesis of 2-CF(3)-tetrahydroquinoline and quinoline derivatives from CF(3)-N-aryl-aldimine

scientific article published on 01 August 2000

Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach

scientific article published on 18 October 2010

The fluorous effect in biomolecular applications ⬇️

artículo científico publicado el 20 de junio de 2011

The use of 4,4,4-trifluorothreonine to stabilize extended peptide structures and mimic β-strands.

artículo científico publicado en 2017

Trifluoromethyl nitrones: from fluoral to optically active hydroxylamines

artículo científico publicado en 2010

α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome.

artículo científico publicado en 2013

Lista de obras de Benoit Crousse

(19)F NMR monitoring of the eukaryotic 20S proteasome chymotrypsin-like activity: an investigative tool for studying allosteric regulation

A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime.

Access to novel amino trifluoromethyl cyclopropane carboxylic acid derivatives

Access to novel functionalized trifluoromethyl β-lactams by ring expansion of aziridines

Aminocyclopropanes as precursors of endoperoxides with antimalarial activity ⬇️

Analogues of key precursors of aspartyl protease inhibitors: synthesis of trifluoromethyl amino epoxides

Benefits of a Dual Chemical and Physical Activation: Direct aza-Michael Addition of Anilines Promoted by Solvent Effect under High Pressure

Bisulfate Salt-Catalyzed Friedel-Crafts Benzylation of Arenes with Benzylic Alcohols

Carbonylhydrazide-based molecular tongs inhibit wild-type and mutated HIV-1 protease dimerization

Designed Glycopeptidomimetics Disrupt Protein-Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability.

Electrophilic amination of fluoroalkyl groups on azodicarboxylate derivatives.

Facile ring opening of oxiranes with aromatic amines in fluoro alcohols

First synthesis of 10 alpha-(trifluoromethyl)deoxoartemisinin

Fluorinated Alcohols: A New Medium for Selective and Clean Reaction

Fluoro artemisinins: difluoromethylene ketones

Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.

Fluorous 4-N,N-dimethylaminopyridine (DMAP) salts as simple recyclable acylation catalysts

Fluorous tagging of DABCO through halogen bonding: recyclable catalyst for the Morita-Baylis-Hillman reaction

In vitro antileishmanial activity of fluoro-artemisinin derivatives against Leishmania donovani

Influence of the structure of polyfluorinated alcohols on Brønsted acidity/hydrogen-bond donor ability and consequences on the promoter effect

Intramolecular Pd-catalyzed carbocyclization, Heck reactions, and aryl-radical cyclizations with planar chiral arene tricarbonyl chromium complexes

N-Difluoromethyl-triazole as a constrained scaffold in peptidomimetics

Non Lewis acid catalysed epoxide ring opening with amino acid esters.

Nonmetal catalyzed insertion reactions of diazocarbonyls to acid derivatives in fluorinated alcohols

Novel [1,2]- and [2,3]-Wittig rearrangements of alpha-benzyloxy beta-CF(3)-beta-lactam enolates

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin

Preparation of 10-trifluoromethyl artemether and artesunate. Influence of hexafluoropropan-2-ol on substitution reaction

Reactivity of carbon dioxide in hydrofluoroethers: a facile access to cyclic carbonates

Regioselective Halogenation of Arenes and Heterocycles in Hexafluoroisopropanol

S(N)/S(N)' competition: selective access to new 10-fluoro artemisinins.

Solubility switch of gold nanoparticles through hydrogen bond association

Solvent-promoted and -controlled aza-Michael reaction with aromatic amines.

Stereoselective Barbier-type allylation reaction of trifluoromethyl aldimines

Structure-activity relationships of sugar-based peptidomimetics as modulators of amyloid β-peptide early oligomerization and fibrillization

Synthesis of 2-CF(3)-tetrahydroquinoline and quinoline derivatives from CF(3)-N-aryl-aldimine

Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach

The fluorous effect in biomolecular applications ⬇️

The use of 4,4,4-trifluorothreonine to stabilize extended peptide structures and mimic β-strands.

Trifluoromethyl nitrones: from fluoral to optically active hydroxylamines

α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome.