Lista de obras - Gerd K. Wagner - Dominio Público Uruguay

2'-deoxy cyclic adenosine 5'-diphosphate ribose derivatives: importance of the 2'-hydroxyl motif for the antagonistic activity of 8-substituted cADPR derivatives

artículo científico publicado en 2008

5-Phenyluridine trihydrate

artículo científico publicado en 2008

A facile two-step synthesis of 8-arylated guanosine mono- and triphosphates (8-aryl GXPs)

artículo científico publicado en 2006

A fast synthetic route to GDP-sugars modified at the nucleobase

artículo científico publicado en 2007

A novel fluorescent probe for NAD-consuming enzymes

artículo científico publicado en 2011

A novel fluorescent probe for retaining galactosyltransferases

artículo científico publicado en 2010

A survey of chemical methods for sugar-nucleotide synthesis.

artículo científico publicado en 2009

Base-modified Donor Analogues Reveal Novel Dynamic Features of a Glycosyltransferase

artículo científico publicado en 2013

Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases.

artículo científico publicado en 2015

CD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose Template

artículo científico publicado en 2013

Cellular effects and metabolic stability of N1-cyclic inosine diphosphoribose and its derivatives

artículo científico publicado en 2006

Conjugation to 4-aminoquinoline improves the anti-trypanosomal activity of Deferiprone-type iron chelators

artículo científico publicado en 2012

Development of fluorescent aryltryptophans by Pd mediated cross-coupling of unprotected halotryptophans in water

artículo científico publicado en 2008

Enzymatic synthesis of nucleobase-modified UDP-sugars: scope and limitations

artículo científico publicado en 2014

Exploring the role of the 5-substituent for the intrinsic fluorescence of 5-aryl and 5-heteroaryl uracil nucleotides: a systematic study

artículo científico publicado en 2013

From imidazoles to pyrimidines: new inhibitors of cytokine release

artículo científico publicado en 2002

Glycosyltransferases and their Assays ⬇️

artículo científico publicado el 24 de septiembre de 2010

Identification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits

scientific article published on 29 November 2017

Identification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.

artículo científico publicado en 2003

Imidazole inhibitors of cytokine release: probing substituents in the 2 position.

artículo científico publicado en 2002

Inhibition of galactosyltransferases by a novel class of donor analogues

artículo científico publicado en 2012

New approaches to the treatment of inflammatory disorders small molecule inhibitors of p38 MAP kinase.

artículo científico publicado en 2006

Novel UDP-GalNAc Derivative Structures Provide Insight into the Donor Specificity of Human Blood Group Glycosyltransferase.

artículo científico publicado en 2015

Novel derivatives of UDP-glucose: concise synthesis and fluorescent properties

artículo científico publicado en 2008

Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes

artículo científico publicado en 2003

One-step synthesis of novel glycosyltransferase inhibitors

scientific article published on 01 December 2012

Ones, thiones, and N-oxides: an exercise in imidazole chemistry

artículo científico publicado en 2002

Optimised chemical synthesis of 5-substituted UDP-sugars and their evaluation as glycosyltransferase inhibitors

artículo científico publicado en 2012

Profiling of <i>Haemophilus influenzae</i> strain R2866 with carbohydrate-based covalent probes

artículo científico publicado en 2020

Rapid synthetic route toward structurally modified derivatives of cyclic adenosine 5'-diphosphate ribose

artículo científico publicado en 2005

Rationally designed squaryldiamides – a novel class of sugar-nucleotide mimics?

artículo científico publicado en 2010

Small molecular anti-cytokine agents.

artículo científico publicado en 2006

Structural determinants for N1/N7 cyclization of nicotinamide hypoxanthine 5'-dinucleotide (NHD+) derivatives by ADP-ribosyl cyclase from aplysia californica: Ca2+-mobilizing activity of 8-substituted cyclic inosine 5'-diphosphoribose analogues in T

scientific article published on 01 August 2006

Studies on the anti-inflammatory activity of phytopharmaceuticals prepared from Arnica flowers

artículo científico publicado en 2002

The first C-glycosidic analogue of a novel galactosyltransferase inhibitor.

artículo científico publicado en 2011

Trypanosoma brucei: chemical evidence that cathepsin L is essential for survival and a relevant drug target

artículo científico publicado en 2012

Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)

artículo científico publicado en 2011

Uncharged nucleoside inhibitors of β-1,4-galactosyltransferase with activity in cells

artículo científico publicado en 2016

Lista de obras de Gerd K. Wagner

2'-deoxy cyclic adenosine 5'-diphosphate ribose derivatives: importance of the 2'-hydroxyl motif for the antagonistic activity of 8-substituted cADPR derivatives

5-Phenyluridine trihydrate

A facile two-step synthesis of 8-arylated guanosine mono- and triphosphates (8-aryl GXPs)

A fast synthetic route to GDP-sugars modified at the nucleobase

A novel fluorescent probe for NAD-consuming enzymes

A novel fluorescent probe for retaining galactosyltransferases

A survey of chemical methods for sugar-nucleotide synthesis.

Base-modified Donor Analogues Reveal Novel Dynamic Features of a Glycosyltransferase

Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases.

CD38 Structure-Based Inhibitor Design Using the N1-Cyclic Inosine 5'-Diphosphate Ribose Template

Cellular effects and metabolic stability of N1-cyclic inosine diphosphoribose and its derivatives

Conjugation to 4-aminoquinoline improves the anti-trypanosomal activity of Deferiprone-type iron chelators

Development of fluorescent aryltryptophans by Pd mediated cross-coupling of unprotected halotryptophans in water

Enzymatic synthesis of nucleobase-modified UDP-sugars: scope and limitations

Exploring the role of the 5-substituent for the intrinsic fluorescence of 5-aryl and 5-heteroaryl uracil nucleotides: a systematic study

From imidazoles to pyrimidines: new inhibitors of cytokine release

Glycosyltransferases and their Assays ⬇️

Identification of non-substrate-like glycosyltransferase inhibitors from library screening: pitfalls & hits

Identification of regioisomers in a series of N-substituted pyridin-4-yl imidazole derivatives by regiospecific synthesis, GC/MS, and 1H NMR.

Imidazole inhibitors of cytokine release: probing substituents in the 2 position.

Inhibition of galactosyltransferases by a novel class of donor analogues

New approaches to the treatment of inflammatory disorders small molecule inhibitors of p38 MAP kinase.

Novel UDP-GalNAc Derivative Structures Provide Insight into the Donor Specificity of Human Blood Group Glycosyltransferase.

Novel derivatives of UDP-glucose: concise synthesis and fluorescent properties

Novel substituted pyridinyl imidazoles as potent anticytokine agents with low activity against hepatic cytochrome P450 enzymes

One-step synthesis of novel glycosyltransferase inhibitors

Ones, thiones, and N-oxides: an exercise in imidazole chemistry

Optimised chemical synthesis of 5-substituted UDP-sugars and their evaluation as glycosyltransferase inhibitors

Profiling of <i>Haemophilus influenzae</i> strain R2866 with carbohydrate-based covalent probes

Rapid synthetic route toward structurally modified derivatives of cyclic adenosine 5'-diphosphate ribose

Rationally designed squaryldiamides – a novel class of sugar-nucleotide mimics?

Small molecular anti-cytokine agents.

Structural determinants for N1/N7 cyclization of nicotinamide hypoxanthine 5'-dinucleotide (NHD+) derivatives by ADP-ribosyl cyclase from aplysia californica: Ca2+-mobilizing activity of 8-substituted cyclic inosine 5'-diphosphoribose analogues in T

Studies on the anti-inflammatory activity of phytopharmaceuticals prepared from Arnica flowers

The first C-glycosidic analogue of a novel galactosyltransferase inhibitor.

Trypanosoma brucei: chemical evidence that cathepsin L is essential for survival and a relevant drug target

Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)

Uncharged nucleoside inhibitors of β-1,4-galactosyltransferase with activity in cells