Lista de obras - Eelco Ruijter - Dominio Público Uruguay

1-Azadienes in cycloaddition and multicomponent reactions towards N-heterocycles

artículo científico publicado en 2008

2-Bromo-6-isocyanopyridine as a Universal Convertible Isocyanide for Multicomponent Chemistry

artículo científico publicado en 2016

A New Route to Protected Acyloins and Their Enzymatic Resolution with Lipases

A flexible six-component reaction to access constrained depsipeptides based on a dihydropyridinone core

artículo científico publicado en 2007

A highly efficient synthesis of telaprevir by strategic use of biocatalysis and multicomponent reactions

artículo científico publicado en 2010

A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation.

artículo científico publicado en 2011

A multicomponent reaction towards N-(cyanomethyl)amides

artículo científico publicado en 2009

A multicomponent synthesis of triazinane diones.

artículo científico publicado en 2007

A novel three-component reaction toward dihydrooxazolopyridines

scientific article published on 01 January 2009

A resource-efficient and highly flexible procedure for a three-component synthesis of 2-imidazolines

artículo científico publicado en 2007

Asymmetric Synthesis of Tetracyclic Pyrroloindolines and Constrained Tryptamines by a Switchable Cascade Reaction

artículo científico publicado en 2015

Asymmetric synthesis of synthetic alkaloids by a tandem biocatalysis/Ugi/Pictet–Spengler-type cyclization sequence

scientific article published on 27 September 2010

Brønsted Acid-Catalyzed Cyanotritylation of Aldehydes by Trityl Isocyanide

scientific article published on 12 July 2016

Catalytic Asymmetric Synthesis of Diketopiperazines by Intramolecular Tsuji-Trost Allylation

scientific article published on 10 September 2019

Chemoselective addition of isocyanides to N-tert-butanesulfinimines

scientific article published in 2014

Copper(i) catalyzed oxidative hydrolysis of Ugi 3-component and Ugi-azide reaction products towards 2° α-ketoamides and α-ketotetrazoles.

artículo científico publicado en 2017

Development of a novel chemical probe for the selective enrichment of phosphorylated serine- and threonine-containing peptides

artículo científico publicado en 2005

Diastereoselective One-Pot Synthesis of Tetrafunctionalized 2-Imidazolines

artículo científico publicado en 2014

Finding Furfural Hydrogenation Catalysts via Predictive Modelling.

artículo científico publicado en 2010

Generation of molecular diversity using a complexity-generating MCR-platform towards triazinane diones

scientific article published on 03 July 2008

Hexafluoroisopropanol as the Acid Component in the Passerini Reaction: One-Pot Access to β-Amino Alcohols.

artículo científico publicado en 2018

Highly Stereoselective Synthesis of Substituted Prolyl Peptides Using a Combination of Biocatalytic Desymmetrization and Multicomponent Reactions

artículo científico publicado en 2010

IBX-mediated oxidation of unactivated cyclic amines: application in highly diastereoselective oxidative Ugi-type and aza-Friedel-Crafts reactions.

artículo científico publicado en 2015

Integrative Theory/Experiment-Driven Exploration of a Multicomponent Reaction towards Imidazoline-2-(thi)ones

Iodide-Catalyzed Synthesis of Secondary Thiocarbamates from Isocyanides and Thiosulfonates

artículo científico publicado en 2016

Iodospirocyclization of Tryptamine-Derived Isocyanides: Formal Total Synthesis of Aspidofractinine

artículo científico publicado en 2018

Isocyanide-based multicomponent reactions towards cyclic constrained peptidomimetics.

artículo científico

Metal-free one-pot α-carboxylation of primary alcohols.

artículo científico publicado en 2016

Mild and Practical Indole C2 Allylation by Allylboration of in situ Generated 3-Chloroindolenines

artículo científico publicado en 2019

Modular Three-Component Synthesis of 4-Aminoquinolines via an Imidoylative Sonogashira/Cyclization Cascade

artículo científico publicado en 2017

Multicomponent Reaction Design in the Quest for Molecular Complexity and Diversity ⬇️

artículo científico publicado el 27 de junio de 2011

Multicomponent reactions - opportunities for the pharmaceutical industry.

artículo científico publicado en 2013

Multicomponent reactions in drug discovery and medicinal chemistry

artículo científico publicado en 2018

Multicomponent synthesis of 3,6-dihydro-2H-1,3-thiazine-2-thiones.

artículo científico publicado en 2012

Multicomponent synthesis of 4-aminophthalazin-1(2H)-ones by palladium-catalyzed isocyanide insertion

artículo científico publicado en 2013

New scavenger resin for the reversible linking and monoprotection of functionalized aromatic aldehydes.

artículo científico publicado en 2004

One-Pot Synthesis of N-Substituted β-Amino Alcohols from Aldehydes and Isocyanides

artículo científico publicado en 2015

Palladium-catalyzed migratory insertion of isocyanides: an emerging platform in cross-coupling chemistry

artículo científico publicado en 2013

Palladium-catalyzed synthesis of 2-aminobenzoxazinones by aerobic oxidative coupling of anthranilic acids and isocyanides.

artículo científico publicado en 2013

Palladium-catalyzed synthesis of 4-aminophthalazin-1(2H)-ones by isocyanide insertion

scientific article published on 15 November 2011

Photocrosslinking and click chemistry enable the specific detection of proteins interacting with phospholipids at the membrane interface

artículo científico publicado en 2009

Recent Advances in Palladium-Catalyzed Isocyanide Insertions

artículo científico publicado en 2020

Recent developments in asymmetric multicomponent reactions.

artículo científico publicado en 2012

Scope and limitations of an efficient four-component reaction for dihydropyridin-2-ones.

artículo científico publicado en 2010

Selective enrichment of Ser-/Thr-phosphorylated peptides in the presence of Ser-/Thr-glycosylated peptides

artículo científico publicado en 2006

Selective formation of 2-imidazolines and 2-substituted oxazoles by using a three-component reaction

scientific article published on 01 January 2008

Sequential Multicomponent Strategy for the Diastereoselective Synthesis of Densely Functionalized Spirooxindole-Fused Thiazolidines.

artículo científico publicado en 2018

Stereoselective Synthesis of Functionalized Bicyclic Scaffolds by Passerini 3-Center-2-Component Reactions of Cyclic Ketoacids.

artículo científico publicado en 2017

Stereoselective Synthesis of Fused Vinylcyclopropanes by Intramolecular Tsuji-Trost Cascade Cyclization

artículo científico publicado en 2018

Stereoselective synthesis of N-aryl proline amides by biotransformation–Ugi-Smiles sequence

artículo científico publicado en 2011

Stereoselective synthesis of fluorinated aminoglycosyl phosphonates

artículo científico publicado en 2015

Sustainable synthesis of diverse privileged heterocycles by palladium-catalyzed aerobic oxidative isocyanide insertion

artículo científico publicado en 2012

Sustainable three-component synthesis of isothioureas from isocyanides, thiosulfonates, and amines

scientific article published on 15 September 2014

Synthesis and photophysics of a red-light absorbing supramolecular chromophore system

artículo científico publicado en 2014

Synthesis and resolution of a key building block for epothilones: a comparison of asymmetric synthesis, chemical and enzymatic resolution

article

Synthesis of 3′-Deoxyribolactones using a Hydrolysis-Induced Lactonization Cascade Reaction of Epoxy Cyanohydrins

Synthesis of 4-aminoquinazolines by palladium-catalyzed intramolecular imidoylation of N-(2-bromoaryl)amidines.

artículo científico publicado en 2011

Synthesis of Densely Functionalized Pyrimidouracils by Nickel(II)-Catalyzed Isocyanide Insertion

scientific article published on 16 January 2020

Synthesis of Imidazolidine-2-(thi)ones via C2-Selective Oxidation and Thionation of 2-Imidazolinium Halides

Synthesis of Secondary Amides from Thiocarbamates

artículo científico publicado en 2018

Synthesis of conformationally constrained peptidomimetics using multicomponent reactions

artículo científico publicado en 2009

Synthesis of heterocycles by formal cycloadditions of isocyanides.

artículo científico publicado en 2014

Synthesis of polycyclic spiroindolines by highly diastereoselective interrupted Ugi cascade reactions of 3-(2-isocyanoethyl)indoles.

artículo científico publicado en 2016

The efficient one-pot reaction of up to eight components by the union of multicomponent reactions

artículo científico publicado en 2009

Thiazine-2-thiones as Masked 1-Azadienes in Cascade Dimerization Reactions).

artículo científico publicado en 2017

Trityl Isocyanide as a Mechanistic Probe in Multicomponent Chemistry: Walking the Line between Ugi- and Strecker-type Reactions.

artículo científico publicado en 2016

What can a chemist learn from nature's macrocycles?--a brief, conceptual view.

artículo científico publicado en 2005

YidC is involved in the biogenesis of the secreted autotransporter hemoglobin protease.

artículo científico publicado en 2010

Lista de obras de Eelco Ruijter

1-Azadienes in cycloaddition and multicomponent reactions towards N-heterocycles

2-Bromo-6-isocyanopyridine as a Universal Convertible Isocyanide for Multicomponent Chemistry

A New Route to Protected Acyloins and Their Enzymatic Resolution with Lipases

A flexible six-component reaction to access constrained depsipeptides based on a dihydropyridinone core

A highly efficient synthesis of telaprevir by strategic use of biocatalysis and multicomponent reactions

A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation.

A multicomponent reaction towards N-(cyanomethyl)amides

A multicomponent synthesis of triazinane diones.

A novel three-component reaction toward dihydrooxazolopyridines

A resource-efficient and highly flexible procedure for a three-component synthesis of 2-imidazolines

Asymmetric Synthesis of Tetracyclic Pyrroloindolines and Constrained Tryptamines by a Switchable Cascade Reaction

Asymmetric synthesis of synthetic alkaloids by a tandem biocatalysis/Ugi/Pictet–Spengler-type cyclization sequence

Brønsted Acid-Catalyzed Cyanotritylation of Aldehydes by Trityl Isocyanide

Catalytic Asymmetric Synthesis of Diketopiperazines by Intramolecular Tsuji-Trost Allylation

Chemoselective addition of isocyanides to N-tert-butanesulfinimines

Copper(i) catalyzed oxidative hydrolysis of Ugi 3-component and Ugi-azide reaction products towards 2° α-ketoamides and α-ketotetrazoles.

Development of a novel chemical probe for the selective enrichment of phosphorylated serine- and threonine-containing peptides

Diastereoselective One-Pot Synthesis of Tetrafunctionalized 2-Imidazolines

Finding Furfural Hydrogenation Catalysts via Predictive Modelling.

Generation of molecular diversity using a complexity-generating MCR-platform towards triazinane diones

Hexafluoroisopropanol as the Acid Component in the Passerini Reaction: One-Pot Access to β-Amino Alcohols.

Highly Stereoselective Synthesis of Substituted Prolyl Peptides Using a Combination of Biocatalytic Desymmetrization and Multicomponent Reactions

IBX-mediated oxidation of unactivated cyclic amines: application in highly diastereoselective oxidative Ugi-type and aza-Friedel-Crafts reactions.

Integrative Theory/Experiment-Driven Exploration of a Multicomponent Reaction towards Imidazoline-2-(thi)ones

Iodide-Catalyzed Synthesis of Secondary Thiocarbamates from Isocyanides and Thiosulfonates

Iodospirocyclization of Tryptamine-Derived Isocyanides: Formal Total Synthesis of Aspidofractinine

Isocyanide-based multicomponent reactions towards cyclic constrained peptidomimetics.

Metal-free one-pot α-carboxylation of primary alcohols.

Mild and Practical Indole C2 Allylation by Allylboration of in situ Generated 3-Chloroindolenines

Modular Three-Component Synthesis of 4-Aminoquinolines via an Imidoylative Sonogashira/Cyclization Cascade

Multicomponent Reaction Design in the Quest for Molecular Complexity and Diversity ⬇️

Multicomponent reactions - opportunities for the pharmaceutical industry.

Multicomponent reactions in drug discovery and medicinal chemistry

Multicomponent synthesis of 3,6-dihydro-2H-1,3-thiazine-2-thiones.

Multicomponent synthesis of 4-aminophthalazin-1(2H)-ones by palladium-catalyzed isocyanide insertion

New scavenger resin for the reversible linking and monoprotection of functionalized aromatic aldehydes.

One-Pot Synthesis of N-Substituted β-Amino Alcohols from Aldehydes and Isocyanides

Palladium-catalyzed migratory insertion of isocyanides: an emerging platform in cross-coupling chemistry

Palladium-catalyzed synthesis of 2-aminobenzoxazinones by aerobic oxidative coupling of anthranilic acids and isocyanides.

Palladium-catalyzed synthesis of 4-aminophthalazin-1(2H)-ones by isocyanide insertion

Photocrosslinking and click chemistry enable the specific detection of proteins interacting with phospholipids at the membrane interface

Recent Advances in Palladium-Catalyzed Isocyanide Insertions

Recent developments in asymmetric multicomponent reactions.

Scope and limitations of an efficient four-component reaction for dihydropyridin-2-ones.

Selective enrichment of Ser-/Thr-phosphorylated peptides in the presence of Ser-/Thr-glycosylated peptides

Selective formation of 2-imidazolines and 2-substituted oxazoles by using a three-component reaction

Sequential Multicomponent Strategy for the Diastereoselective Synthesis of Densely Functionalized Spirooxindole-Fused Thiazolidines.

Stereoselective Synthesis of Functionalized Bicyclic Scaffolds by Passerini 3-Center-2-Component Reactions of Cyclic Ketoacids.

Stereoselective Synthesis of Fused Vinylcyclopropanes by Intramolecular Tsuji-Trost Cascade Cyclization

Stereoselective synthesis of N-aryl proline amides by biotransformation–Ugi-Smiles sequence

Stereoselective synthesis of fluorinated aminoglycosyl phosphonates

Sustainable synthesis of diverse privileged heterocycles by palladium-catalyzed aerobic oxidative isocyanide insertion

Sustainable three-component synthesis of isothioureas from isocyanides, thiosulfonates, and amines

Synthesis and photophysics of a red-light absorbing supramolecular chromophore system

Synthesis and resolution of a key building block for epothilones: a comparison of asymmetric synthesis, chemical and enzymatic resolution

Synthesis of 3′-Deoxyribolactones using a Hydrolysis-Induced Lactonization Cascade Reaction of Epoxy Cyanohydrins

Synthesis of 4-aminoquinazolines by palladium-catalyzed intramolecular imidoylation of N-(2-bromoaryl)amidines.

Synthesis of Densely Functionalized Pyrimidouracils by Nickel(II)-Catalyzed Isocyanide Insertion

Synthesis of Imidazolidine-2-(thi)ones via C2-Selective Oxidation and Thionation of 2-Imidazolinium Halides

Synthesis of Secondary Amides from Thiocarbamates

Synthesis of conformationally constrained peptidomimetics using multicomponent reactions

Synthesis of heterocycles by formal cycloadditions of isocyanides.

Synthesis of polycyclic spiroindolines by highly diastereoselective interrupted Ugi cascade reactions of 3-(2-isocyanoethyl)indoles.

The efficient one-pot reaction of up to eight components by the union of multicomponent reactions

Thiazine-2-thiones as Masked 1-Azadienes in Cascade Dimerization Reactions).

Trityl Isocyanide as a Mechanistic Probe in Multicomponent Chemistry: Walking the Line between Ugi- and Strecker-type Reactions.

What can a chemist learn from nature's macrocycles?--a brief, conceptual view.

YidC is involved in the biogenesis of the secreted autotransporter hemoglobin protease.