Lista de obras - Marco Pallavicini - Dominio Público Uruguay

4-Oxystilbene compounds are selective ligands for neuronal nicotinic alphaBungarotoxin receptors.

artículo científico publicado en 1998

5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity

artículo científico publicado en 2008

6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist.

artículo científico publicado en 2013

Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.

artículo científico publicado en 2012

An investigation into the influence of counterion on the RS-propranolol and S-propranolol skin permeability.

artículo científico publicado en 2010

Benzodioxane-benzamides as new bacterial cell division inhibitors

artículo científico publicado en 2014

Cardiovascular and pulmonary activity of platelet-activating factor (PAF-acether) and its derivatives.

artículo científico publicado en 1986

Characterization of in vitro metabolites of JWH-018, JWH-073 and their 4-methyl derivatives, markers of the abuse of these synthetic cannabinoids

artículo científico publicado en 2014

Construction of human ghrelin receptor (hGHS-R1a) model using a fragmental prediction approach and validation through docking analysis

artículo científico publicado en 2006

Corrigendum to “Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes” [Bioorg. Med. Chem. Lett. 16 (2006) 5610–5615]

scholarly article published in Bioorganic & Medicinal Chemistry Letters

Design, synthesis and binding affinity of acetylcholine carbamoyl analogues

artículo científico publicado en 2013

Exploring the space of histidine containing dipeptides in search of novel efficient RCS sequestering agents

artículo científico publicado en 2013

Farnesyltransferase inhibitors: CAAX mimetics based on different biaryl scaffolds

scientific article published on 30 April 2014

From 2-aminomethyl-1,4-benzodioxane enantiomers to unichiral 2-cyano- and 2-carbonyl-substituted benzodioxanes via dichloroamine

artículo científico publicado en 2014

Identification of 1-butyl-3-(1-(4-methyl)naphtoyl)indole detected for the first time in “herbal high” products on the Italian market

article

Modelling of full-length human alpha4beta2 nicotinic receptor by fragmental approach and analysis of its binding modes

artículo científico publicado en 2008

Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

artículo científico publicado en 2020

New Ras CAAX mimetics: design, synthesis, antiproliferative activity, and RAS prenylation inhibition

artículo científico publicado en 2009

Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency

artículo científico publicado en 2007

Potent anti-glioblastoma agents by hybridizing the onium-alkyloxy-stilbene based structures of an alpha7-, alpha9-nAChR antagonist and of a pro-oxidant mitocan

artículo científico publicado en 2018

Predicting the physicochemical profile of diastereoisomeric histidine-containing dipeptides by property space analysis

artículo científico publicado en 2012

QSAR study for a novel series of ortho disubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

artículo científico publicado en 2006

QSAR study for a novel series of ortho monosubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

artículo científico publicado en 2005

Structure-affinity studies for a novel series of homochiral naphtho and tetrahydronaphtho analogues of alpha 1 antagonist WB-4101.

artículo científico publicado en 2004

Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers

artículo científico publicado en 2004

Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes

artículo científico publicado en 2006

Synthesis of homochiral 5- and 8-substituted 2-[((2-(2,6-dimethoxyphenoxy)-ethyl)amino)methyl]-1,4-benzodioxanes and electrophoretic determination of their enantiomeric excess

scientific article published on 01 February 2001

Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase

artículo científico publicado en 2011

Unichiral 2-(2'-pyrrolidinyl)-1,4-benzodioxanes: the 2R,2'S diastereomer of the N-methyl-7-hydroxy analogue is a potent α4β2- and α6β2-nicotinic acetylcholine receptor partial agonist

artículo científico publicado en 2011

WB4101-related compounds: new, subtype-selective alpha1-adrenoreceptor antagonists (or inverse agonists?).

artículo científico publicado en 2006

Lista de obras de Marco Pallavicini

4-Oxystilbene compounds are selective ligands for neuronal nicotinic alphaBungarotoxin receptors.

5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity

6-methoxy-7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of 2-[2-(2,6-Dimethoxyphenoxy)ethyl]aminomethyl-1,4-benzodioxane (WB4101):1 discovery of a potent and selective α1D-adrenoceptor antagonist.

Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist.

An investigation into the influence of counterion on the RS-propranolol and S-propranolol skin permeability.

Benzodioxane-benzamides as new bacterial cell division inhibitors

Cardiovascular and pulmonary activity of platelet-activating factor (PAF-acether) and its derivatives.

Characterization of in vitro metabolites of JWH-018, JWH-073 and their 4-methyl derivatives, markers of the abuse of these synthetic cannabinoids

Construction of human ghrelin receptor (hGHS-R1a) model using a fragmental prediction approach and validation through docking analysis

Corrigendum to “Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes” [Bioorg. Med. Chem. Lett. 16 (2006) 5610–5615]

Design, synthesis and binding affinity of acetylcholine carbamoyl analogues

Exploring the space of histidine containing dipeptides in search of novel efficient RCS sequestering agents

Farnesyltransferase inhibitors: CAAX mimetics based on different biaryl scaffolds

From 2-aminomethyl-1,4-benzodioxane enantiomers to unichiral 2-cyano- and 2-carbonyl-substituted benzodioxanes via dichloroamine

Identification of 1-butyl-3-(1-(4-methyl)naphtoyl)indole detected for the first time in “herbal high” products on the Italian market

Modelling of full-length human alpha4beta2 nicotinic receptor by fragmental approach and analysis of its binding modes

Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

New Ras CAAX mimetics: design, synthesis, antiproliferative activity, and RAS prenylation inhibition

Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency

Potent anti-glioblastoma agents by hybridizing the onium-alkyloxy-stilbene based structures of an alpha7-, alpha9-nAChR antagonist and of a pro-oxidant mitocan

Predicting the physicochemical profile of diastereoisomeric histidine-containing dipeptides by property space analysis

QSAR study for a novel series of ortho disubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

QSAR study for a novel series of ortho monosubstituted phenoxy analogues of alpha1-adrenoceptor antagonist WB4101.

Structure-affinity studies for a novel series of homochiral naphtho and tetrahydronaphtho analogues of alpha 1 antagonist WB-4101.

Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers

Synthesis and α4β2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes

Synthesis of homochiral 5- and 8-substituted 2-[((2-(2,6-dimethoxyphenoxy)-ethyl)amino)methyl]-1,4-benzodioxanes and electrophoretic determination of their enantiomeric excess

Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase

Unichiral 2-(2'-pyrrolidinyl)-1,4-benzodioxanes: the 2R,2'S diastereomer of the N-methyl-7-hydroxy analogue is a potent α4β2- and α6β2-nicotinic acetylcholine receptor partial agonist

WB4101-related compounds: new, subtype-selective alpha1-adrenoreceptor antagonists (or inverse agonists?).