Lista de obras - Louis Gendron - Dominio Público Uruguay

A Ras-dependent chloride current activated by adrenocorticotropin in rat adrenal zona glomerulosa cells

scientific article published on 01 February 2000

A role for p21ras in the angiotensin II AT2 receptor transduction pathway

scientific article published on 01 August 1998

Activation of spinal mu- and delta-opioid receptors potently inhibits substance P release induced by peripheral noxious stimuli

artículo científico publicado en 2011

Adeno-associated virus 2/9 delivery of Cre recombinase in mouse primary afferents.

artículo científico publicado en 2018

Alleviating pain with delta opioid receptor agonists: evidence from experimental models

artículo científico publicado en 2020

Altered morphine-induced analgesia in neurotensin type 1 receptor null mice.

artículo científico publicado en 2010

Behavioral, medical imaging and histopathological features of a new rat model of bone cancer pain

artículo científico publicado en 2010

Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.

artículo científico publicado en 2018

Coexpression of somatostatin receptor subtype 5 affects internalization and trafficking of somatostatin receptor subtype 2.

artículo científico publicado en 2007

Corrigendum to "Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings" [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320-2323]

scientific article published on 05 September 2018

Delta Opioid Receptor Signaling Promotes Resilience to Stress Under the Repeated Social Defeat Paradigm in Mice

artículo científico publicado en 2018

Delta opioid receptor-mediated analgesia is not altered in preprotachykinin A knockout mice

artículo científico publicado en 2010

Delta opioid receptors recycle to the membrane after sorting to the degradation path

artículo científico publicado en 2017

Differential noxious and motor tolerance of chronic delta opioid receptor agonists in rodents

artículo científico publicado en 2009

Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists

artículo científico publicado en 2019

Enkephalins: Endogenous Analgesics with an Emerging Role in Stress Resilience

artículo científico publicado en 2017

Essential role of mu opioid receptor in the regulation of delta opioid receptor-mediated antihyperalgesia

artículo científico publicado en 2007

Experimental Autoimmune Encephalomyelitis Potentiates Mouse Mast Cell Protease 4-Dependent Pressor Responses to Centrally or Systemically Administered Big Endothelin-1

scientific article published on 27 June 2019

Exploring the Backbone of Enkephalins To Adjust Their Pharmacological Profile for the δ-Opioid Receptor.

artículo científico publicado en 2010

Identification and functional characterization of a 5-transmembrane domain variant isoform of the NTS2 neurotensin receptor in rat central nervous system.

artículo científico publicado en 2005

Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound

artículo científico publicado en 2014

Identification of N-[(5-{[(4-methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine (NTRC-824), a neurotensin-like nonpeptide compound selective for the neurotensin receptor type 2

artículo científico publicado en 2014

Implication of delta opioid receptor subtype 2 but not delta opioid receptor subtype 1 in the development of morphine analgesic tolerance in a rat model of chronic inflammatory pain

artículo científico publicado en 2015

In vivo mapping of a GPCR interactome using knockin mice

scientific article published on 26 May 2020

Increased anxiety-like behaviors in rats experiencing chronic inflammatory pain.

artículo científico publicado en 2012

Increased radiosensitivity of colorectal tumors with intra-tumoral injection of low dose of gold nanoparticles.

artículo científico publicado en 2016

Involvement of cannabinoid receptors in peripheral and spinal morphine analgesia

artículo científico publicado en 2013

Involvement of the coatomer protein complex I in the intracellular traffic of the delta opioid receptor

artículo científico publicado en 2016

Label-free monitoring of apoptosis by surface plasmon resonance detection of morphological changes

artículo científico publicado en 2012

Label-free monitoring of μ-opioid receptor-mediated signaling.

artículo científico publicado en 2014

Low-affinity neurotensin receptor (NTS2) signaling: internalization-dependent activation of extracellular signal-regulated kinases 1/2.

artículo científico publicado en 2004

Molecular Pharmacology of δ-Opioid Receptors

artículo científico publicado en 2016

Molecular aspects of delta opioid receptors ⬇️

scientific article published on 08 July 2019

Monitoring the Aggregation of GPCRs by Fluorescence Microscopy

scientific article published on 01 January 2019

Morphine and pain-related stimuli enhance cell surface availability of somatic delta-opioid receptors in rat dorsal root ganglia.

artículo científico publicado en 2006

Morphine priming in rats with chronic inflammation reveals a dichotomy between antihyperalgesic and antinociceptive properties of deltorphin.

artículo científico publicado en 2006

N-Guanidyl and C-Tetrazole Leu-Enkephalin Derivatives: Efficient Mu and Delta Opioid Receptor Agonists with Improved Pharmacological Properties

artículo científico publicado en 2019

NLRX1 inhibits the early stages of CNS inflammation and prevents the onset of spontaneous autoimmunity

artículo científico publicado en 2019

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

artículo científico publicado en 2019

Nitric oxide and cyclic GMP are involved in angiotensin II AT(2) receptor effects on neurite outgrowth in NG108-15 cells

artículo científico publicado en 2002

Pain after discontinuation of morphine treatment is associated with synaptic increase of GluA4-containing AMPAR in the dorsal horn of the spinal cord.

artículo científico publicado en 2013

Pharmacology and functional properties of NTS2 neurotensin receptors in cerebellar granule cells

scientific journal article

Preparation and evaluation at the delta opioid receptor of a series of linear leu-enkephalin analogues obtained by systematic replacement of the amides

artículo científico publicado en 2013

Presence of task-1 channel in the laryngeal mucosa in the newborn lamb

artículo científico publicado en 2011

Prolonged morphine treatment selectively increases membrane recruitment of delta-opioid receptors in mouse basal ganglia

artículo científico publicado en 2005

Recent advances on the δ opioid receptor: from trafficking to function

artículo científico publicado en 2014

Regulation of μ and δ opioid receptor functions: involvement of cyclin-dependent kinase 5.

artículo científico publicado en 2015

Sciatic nerve ligation-induced proliferation of spinal cord astrocytes is mediated by kappa opioid activation of p38 mitogen-activated protein kinase

artículo científico publicado en 2007

Spinal activation of delta opioid receptors alleviates cancer-related bone pain

artículo científico publicado en 2011

Spinal μ and δ opioids inhibit both thermal and mechanical pain in rats.

artículo científico publicado en 2013

Synthesis and Evaluation of a 64Cu-Conjugate, a Selective δ-Opioid Receptor Positron Emission Tomography Imaging Agent.

artículo científico publicado en 2017

Synthesis of Gly-ψ[(Z)CF═CH]-Phe, a Fluoroalkene Dipeptide Isostere, and Its Incorporation into a Leu-enkephalin Peptidomimetic.

artículo científico publicado en 2016

Systematic replacement of amides by 1,4-disubstituted[1,2,3]triazoles in Leu-enkephalin and the impact on the delta opioid receptor activity

artículo científico publicado en 2013

The Delta Opioid Receptor in Pain Control.

artículo científico publicado en 2017

The PAR2 inhibitor I-287 selectively targets Gαq and Gα12/13 signaling and has anti-inflammatory effects

artículo científico publicado en 2020

The angiotensin type 2 receptor of angiotensin II and neuronal differentiation: from observations to mechanisms

scientific journal article

The combination of opioid and neurotensin receptor agonists improves their analgesic/adverse effect ratio

artículo científico publicado en 2019

Use of a non-invasive brain penetrating peptide-drug conjugate strategy to improve the delivery of opioid pain relief medications to the brain

artículo científico publicado en 2020

iRAGE as a novel carboxymethylated peptide that prevents advanced glycation end product-induced apoptosis and endoplasmic reticulum stress in vascular smooth muscle cells

artículo científico publicado en 2015

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.

artículo científico publicado en 2017

Lista de obras de Louis Gendron

A Ras-dependent chloride current activated by adrenocorticotropin in rat adrenal zona glomerulosa cells

A role for p21ras in the angiotensin II AT2 receptor transduction pathway

Activation of spinal mu- and delta-opioid receptors potently inhibits substance P release induced by peripheral noxious stimuli

Adeno-associated virus 2/9 delivery of Cre recombinase in mouse primary afferents.

Alleviating pain with delta opioid receptor agonists: evidence from experimental models

Altered morphine-induced analgesia in neurotensin type 1 receptor null mice.

Behavioral, medical imaging and histopathological features of a new rat model of bone cancer pain

Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.

Coexpression of somatostatin receptor subtype 5 affects internalization and trafficking of somatostatin receptor subtype 2.

Corrigendum to "Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings" [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320-2323]

Delta Opioid Receptor Signaling Promotes Resilience to Stress Under the Repeated Social Defeat Paradigm in Mice

Delta opioid receptor-mediated analgesia is not altered in preprotachykinin A knockout mice

Delta opioid receptors recycle to the membrane after sorting to the degradation path

Differential noxious and motor tolerance of chronic delta opioid receptor agonists in rodents

Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists

Enkephalins: Endogenous Analgesics with an Emerging Role in Stress Resilience

Essential role of mu opioid receptor in the regulation of delta opioid receptor-mediated antihyperalgesia

Experimental Autoimmune Encephalomyelitis Potentiates Mouse Mast Cell Protease 4-Dependent Pressor Responses to Centrally or Systemically Administered Big Endothelin-1

Exploring the Backbone of Enkephalins To Adjust Their Pharmacological Profile for the δ-Opioid Receptor.

Identification and functional characterization of a 5-transmembrane domain variant isoform of the NTS2 neurotensin receptor in rat central nervous system.

Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound

Identification of N-[(5-{[(4-methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine (NTRC-824), a neurotensin-like nonpeptide compound selective for the neurotensin receptor type 2

Implication of delta opioid receptor subtype 2 but not delta opioid receptor subtype 1 in the development of morphine analgesic tolerance in a rat model of chronic inflammatory pain

In vivo mapping of a GPCR interactome using knockin mice

Increased anxiety-like behaviors in rats experiencing chronic inflammatory pain.

Increased radiosensitivity of colorectal tumors with intra-tumoral injection of low dose of gold nanoparticles.

Involvement of cannabinoid receptors in peripheral and spinal morphine analgesia

Involvement of the coatomer protein complex I in the intracellular traffic of the delta opioid receptor

Label-free monitoring of apoptosis by surface plasmon resonance detection of morphological changes

Label-free monitoring of μ-opioid receptor-mediated signaling.

Low-affinity neurotensin receptor (NTS2) signaling: internalization-dependent activation of extracellular signal-regulated kinases 1/2.

Molecular Pharmacology of δ-Opioid Receptors

Molecular aspects of delta opioid receptors ⬇️

Monitoring the Aggregation of GPCRs by Fluorescence Microscopy

Morphine and pain-related stimuli enhance cell surface availability of somatic delta-opioid receptors in rat dorsal root ganglia.

Morphine priming in rats with chronic inflammation reveals a dichotomy between antihyperalgesic and antinociceptive properties of deltorphin.

N-Guanidyl and C-Tetrazole Leu-Enkephalin Derivatives: Efficient Mu and Delta Opioid Receptor Agonists with Improved Pharmacological Properties

NLRX1 inhibits the early stages of CNS inflammation and prevents the onset of spontaneous autoimmunity

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

Nitric oxide and cyclic GMP are involved in angiotensin II AT(2) receptor effects on neurite outgrowth in NG108-15 cells

Pain after discontinuation of morphine treatment is associated with synaptic increase of GluA4-containing AMPAR in the dorsal horn of the spinal cord.

Pharmacology and functional properties of NTS2 neurotensin receptors in cerebellar granule cells

Preparation and evaluation at the delta opioid receptor of a series of linear leu-enkephalin analogues obtained by systematic replacement of the amides

Presence of task-1 channel in the laryngeal mucosa in the newborn lamb

Prolonged morphine treatment selectively increases membrane recruitment of delta-opioid receptors in mouse basal ganglia

Recent advances on the δ opioid receptor: from trafficking to function

Regulation of μ and δ opioid receptor functions: involvement of cyclin-dependent kinase 5.

Sciatic nerve ligation-induced proliferation of spinal cord astrocytes is mediated by kappa opioid activation of p38 mitogen-activated protein kinase

Spinal activation of delta opioid receptors alleviates cancer-related bone pain

Spinal μ and δ opioids inhibit both thermal and mechanical pain in rats.

Synthesis and Evaluation of a 64Cu-Conjugate, a Selective δ-Opioid Receptor Positron Emission Tomography Imaging Agent.

Synthesis of Gly-ψ[(Z)CF═CH]-Phe, a Fluoroalkene Dipeptide Isostere, and Its Incorporation into a Leu-enkephalin Peptidomimetic.

Systematic replacement of amides by 1,4-disubstituted[1,2,3]triazoles in Leu-enkephalin and the impact on the delta opioid receptor activity

The Delta Opioid Receptor in Pain Control.

The PAR2 inhibitor I-287 selectively targets Gαq and Gα12/13 signaling and has anti-inflammatory effects

The angiotensin type 2 receptor of angiotensin II and neuronal differentiation: from observations to mechanisms

The combination of opioid and neurotensin receptor agonists improves their analgesic/adverse effect ratio

Use of a non-invasive brain penetrating peptide-drug conjugate strategy to improve the delivery of opioid pain relief medications to the brain

iRAGE as a novel carboxymethylated peptide that prevents advanced glycation end product-induced apoptosis and endoplasmic reticulum stress in vascular smooth muscle cells

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.