Lista de obras - Dong Guo - Dominio Público Uruguay

5′-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A2A Receptor

artículo científico publicado en 2016

A two-state model for the kinetics of competitive radioligand binding.

artículo científico publicado en 2018

Agonists for the adenosine A1 receptor with tunable residence time. A Case for nonribose 4-amino-6-aryl-5-cyano-2-thiopyrimidines

artículo científico publicado en 2014

Biased and constitutive signaling in the CC-chemokine receptor CCR5 by manipulating the interface between transmembrane helices 6 and 7.

artículo científico publicado en 2013

Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor

artículo científico publicado en 2014

Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge Strength

artículo científico publicado en 2016

Drug-Target Association Kinetics in Drug Discovery

artículo científico publicado en 2019

Drug-target residence time--a case for G protein-coupled receptors

artículo científico publicado en 2014

Dual-point competition association assay: a fast and high-throughput kinetic screening method for assessing ligand-receptor binding kinetics

artículo científico publicado en 2012

Equilibrium and kinetic selectivity profiling on the human adenosine receptors

artículo científico publicado en 2016

Exploring chemical substructures essential for HERG k(+) channel blockade by synthesis and biological evaluation of dofetilide analogues

artículo científico publicado en 2009

Functional efficacy of adenosine A₂A receptor agonists is positively correlated to their receptor residence time

artículo científico publicado en 2012

GPCR structure and activation: an essential role for the first extracellular loop in activating the adenosine A2B receptor

scholarly article published February 2011

Gating function of isoleucine-116 in TM-3 (position III:16/3.40) for the activity state of the CC-chemokine receptor 5 (CCR5).

artículo científico publicado en 2014

Kinetic Aspects of the Interaction between Ligand and G Protein-Coupled Receptor: The Case of the Adenosine Receptors

artículo científico publicado en 2016

Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors.

artículo científico publicado en 2015

Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor.

artículo científico publicado en 2016

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor

artículo científico publicado en 2014

Structure-Activity Relationships of the Sustained Effects of Adenosine A2A Receptor Agonists Driven by Slow Dissociation Kinetics.

artículo científico publicado en 2016

Structure-kinetics relationships of Capadenoson derivatives as adenosine A 1 receptor agonists

artículo científico publicado en 2015

The Added Value of Assessing Ligand-Receptor Binding Kinetics in Drug Discovery

artículo científico publicado en 2016

The Role of Target Binding Kinetics in Drug Discovery

artículo científico publicado en 2015

Lista de obras de Dong Guo

5′-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A2A Receptor

A two-state model for the kinetics of competitive radioligand binding.

Agonists for the adenosine A1 receptor with tunable residence time. A Case for nonribose 4-amino-6-aryl-5-cyano-2-thiopyrimidines

Biased and constitutive signaling in the CC-chemokine receptor CCR5 by manipulating the interface between transmembrane helices 6 and 7.

Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor

Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge Strength

Drug-Target Association Kinetics in Drug Discovery

Drug-target residence time--a case for G protein-coupled receptors

Dual-point competition association assay: a fast and high-throughput kinetic screening method for assessing ligand-receptor binding kinetics

Equilibrium and kinetic selectivity profiling on the human adenosine receptors

Exploring chemical substructures essential for HERG k(+) channel blockade by synthesis and biological evaluation of dofetilide analogues

Functional efficacy of adenosine A₂A receptor agonists is positively correlated to their receptor residence time

GPCR structure and activation: an essential role for the first extracellular loop in activating the adenosine A2B receptor

Gating function of isoleucine-116 in TM-3 (position III:16/3.40) for the activity state of the CC-chemokine receptor 5 (CCR5).

Kinetic Aspects of the Interaction between Ligand and G Protein-Coupled Receptor: The Case of the Adenosine Receptors

Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors.

Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor.

Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor

Structure-Activity Relationships of the Sustained Effects of Adenosine A2A Receptor Agonists Driven by Slow Dissociation Kinetics.

Structure-kinetics relationships of Capadenoson derivatives as adenosine A 1 receptor agonists

The Added Value of Assessing Ligand-Receptor Binding Kinetics in Drug Discovery

The Role of Target Binding Kinetics in Drug Discovery