Lista de obras - Roland J. Pieters - Dominio Público Uruguay

A New Chemical Probe for Proteomics of Carbohydrate-Binding Proteins

artículo científico publicado en 2005

A facile synthesis of the GalNAcbeta1-->4Gal target sequence of respiratory pathogens.

artículo científico publicado en 2005

A hybrid polymer to target blood group dependence of cholera toxin

scientific article published on 01 December 2019

A new chemical probe for the detection of the cancer-linked galectin-3

scientific article published on 30 October 2006

A proteinaceous fraction of wheat bran may interfere in the attachment of enterotoxigenic E. coli K88 (F4+) to porcine epithelial cells

artículo científico publicado en 2014

Activity Based High-Throughput Screening for Novel O-GlcNAc Transferase Substrates Using a Dynamic Peptide Microarray

artículo científico publicado en 2016

Adhesion inhibition of F1C-fimbriated Escherichia coli and Pseudomonas aeruginosa PAK and PAO by multivalent carbohydrate ligands.

artículo científico publicado en 2003

Bacterial Adhesion of Streptococcus suis to Host Cells and Its Inhibition by Carbohydrate Ligands.

artículo científico publicado en 2013

Cross-platform comparison of glycan microarray formats.

artículo científico publicado en 2014

Demystifying O-GlcNAcylation: hints from peptide substrates

artículo científico publicado en 2018

Detection of galectin-3 by novel peptidic photoprobes

artículo científico publicado en 2006

Detection of pathogenic Streptococcus suis bacteria using magnetic glycoparticles.

artículo científico publicado en 2010

Efficient microwave-assisted synthesis of multivalent dendrimeric peptides using cycloaddition reaction (click) chemistry

artículo científico publicado en 2005

Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors.

artículo científico publicado en 2013

Enhanced Inhibition of Influenza A Virus Adhesion by Di- and Trivalent Hemagglutinin Inhibitors

scientific article published on 28 June 2019

Enhanced membrane pore formation by multimeric/oligomeric antimicrobial peptides

scientific article published on 18 October 2007

Enhancing membrane disruption by targeting and multivalent presentation of antimicrobial peptides.

artículo científico publicado en 2012

Functional Characterization of Cholera Toxin Inhibitors Using Human Intestinal Organoids

artículo científico publicado en 2016

Functional assay for shiga-like toxin via detection by antibody capture and multivalent galabiose binding.

artículo científico publicado en 2012

Functionalization of a Rigid Divalent Ligand for LecA, a Bacterial Adhesion Lectin

artículo científico publicado en 2015

Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition

artículo científico publicado en 2016

Homodimeric galectin-7 (p53-induced gene 1) is a negative growth regulator for human neuroblastoma cells

artículo científico publicado en 2003

ITAM-derived phosphopeptide-containing dendrimers as multivalent ligands for Syk tandem SH2 domain.

artículo científico publicado en 2009

Identification of laminin-binding motifs of Yersinia pestis plasminogen activator by phage display

artículo científico publicado en 2005

Identification of peptide ligands for malignancy- and growth-regulating galectins using random phage-display and designed combinatorial peptide libraries.

artículo científico publicado en 2005

Inhibition and detection of galectins.

artículo científico publicado en 2006

Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids

scientific article published on 18 April 2018

Inhibition of P-fimbriated Escherichia coli adhesion by multivalent galabiose derivatives studied by a live-bacteria application of surface plasmon resonance.

artículo científico

Inhibition of Streptococcus suis adhesion by dendritic galabiose compounds at low nanomolar concentration.

artículo científico publicado en 2004

Interference of the galactose-dependent binding of lectins by novel pentapeptide ligands

artículo científico publicado en 2004

Intervention with bacterial adhesion by multivalent carbohydrates.

artículo científico publicado en 2007

Intracellular Hydrolysis of Small-Molecule O-Linked N-Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition

artículo científico publicado en 2020

Lactulose synergizes with CpG-ODN to modulate epithelial and immune cells cross talk

scientific article published on 01 January 2019

Maximising multivalency effects in protein-carbohydrate interactions

artículo científico publicado en 2009

Measuring O-GlcNAc cleavage by OGA and cell lysates on a peptide microarray

artículo científico publicado en 2017

Microwave-assisted, tin-mediated, regioselective 3-O-alkylation of galactosides

Multivalent carbohydrate recognition on a glycodendrimer-functionalized flow-through chip.

artículo científico publicado en 2008

Multivalent glycoconjugates as anti-pathogenic agents ⬇️

artículo científico publicado en 2012

N-Guanidino Derivatives of 1,5-Dideoxy-1,5-imino-d-xylitol are Potent, Selective, and Stable Inhibitors of β-Glucocerebrosidase

artículo científico publicado en 2017

Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase

artículo científico publicado en 2009

New properties of wheat bran: anti-biofilm activity and interference with bacteria quorum-sensing systems

artículo científico publicado en 2014

Optimizing divalent inhibitors of Pseudomonas aeruginosa lectin LecA by using a rigid spacer.

artículo científico publicado en 2013

Orthoester functionalized N-guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase

artículo científico publicado en 2017

Peptide microarray analysis of the cross-talk between O-GlcNAcylation and tyrosine phosphorylation

artículo científico publicado en 2017

PhoX - an IMAC-enrichable Crosslinking Reagent

PhoX: An IMAC-Enrichable Cross-Linking Reagent

artículo científico publicado en 2019

Potent divalent inhibitors with rigid glucose click spacers for Pseudomonas aeruginosa lectin LecA

artículo científico publicado en 2012

Potential scorpionate antibiotics: targeted hydrolysis of lipid II containing model membranes by vancomycin-TACzyme conjugates and modulation of their antibacterial activity by Zn-ions.

artículo científico publicado en 2009

Probing the Inhibitor versus Chaperone Properties of sp2-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease

artículo científico publicado en 2018

Rapid screening of lectins for multivalency effects with a glycodendrimer microarray

artículo científico publicado en 2010

Rationally Designed Chemically Modified Glycodendrimer Inhibits Streptococcus suis Adhesin SadP at Picomolar Concentrations.

artículo científico publicado en 2017

Rigidified multivalent lactose molecules and their interactions with mammalian galectins: a route to selective inhibitors.

artículo científico publicado en 2003

Site-specific conjugation of single domain antibodies to liposomes enhances photosensitizer uptake and photodynamic therapy efficacy.

artículo científico publicado en 2016

Strong Inhibition of Cholera Toxin B Subunit by Affordable, Polymer-Based Multivalent Inhibitors

artículo científico publicado en 2019

Strong Inhibition of Cholera Toxin by Multivalent GM1 Derivatives

artículo científico publicado en 2007

Strong inhibition of cholera toxin binding by galactose dendrimers.

artículo científico publicado en 2007

Structural Insight into Multivalent Galactoside Binding to Pseudomonas aeruginosa Lectin LecA

artículo científico publicado en 2015

Study of cross talk between phosphatases and OGA on a ZO-3-derived peptide

scientific article published on 06 February 2019

Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics

artículo científico publicado en 2002

Synthesis and cholera toxin binding properties of multivalent GM1 mimics

artículo científico publicado en 2004

Synthesis and evaluation of TAC-based inhibitors of papain as mimics of cystatin B

artículo científico publicado en 2007

Synthesis and evaluation of new thiodigalactoside-based chemical probes to label galectin-3.

artículo científico publicado en 2009

Synthesis and evaluation of novel macrocyclic antifungal peptides

artículo científico publicado en 2011

Synthesis of multivalent Streptococcus suis adhesion inhibitors by enzymatic cleavage of polygalacturonic acid and 'click' conjugation.

artículo científico publicado en 2008

Tannic acid mimicking dendrimers as small intestine submucosa stabilizing nanomordants.

artículo científico publicado en 2005

Tetra- versus Pentavalent Inhibitors of Cholera Toxin ⬇️

artículo científico

The influence of ligand valency on aggregation mechanisms for inhibiting bacterial toxins.

artículo científico publicado en 2009

The vancomycin-nisin(1-12) hybrid restores activity against vancomycin resistant Enterococci

artículo científico publicado en 2008

Thiodigalactoside-Bovine Serum Albumin Conjugates as High-Potency Inhibitors of Galectin-3: An Outstanding Example of Multivalent Presentation of Small Molecule Inhibitors.

artículo científico publicado en 2018

Thiourea-based spacers in potent divalent inhibitors of Pseudomonas aeruginosa virulence lectin LecA.

artículo científico publicado en 2015

Tuning the preference of thiodigalactoside- and lactosamine-based ligands to galectin-3 over galectin-1

scientific article published on 23 January 2013

Uptake and transport of superparamagnetic iron oxide nanoparticles through human brain capillary endothelial cells

scientific article published on 26 August 2013

Use of tetravalent galabiose for inhibition of streptococcus suis serotype 2 infection in a mouse model

artículo científico publicado en 2013

Lista de obras de Roland J. Pieters

A New Chemical Probe for Proteomics of Carbohydrate-Binding Proteins

A facile synthesis of the GalNAcbeta1-->4Gal target sequence of respiratory pathogens.

A hybrid polymer to target blood group dependence of cholera toxin

A new chemical probe for the detection of the cancer-linked galectin-3

A proteinaceous fraction of wheat bran may interfere in the attachment of enterotoxigenic E. coli K88 (F4+) to porcine epithelial cells

Activity Based High-Throughput Screening for Novel O-GlcNAc Transferase Substrates Using a Dynamic Peptide Microarray

Adhesion inhibition of F1C-fimbriated Escherichia coli and Pseudomonas aeruginosa PAK and PAO by multivalent carbohydrate ligands.

Bacterial Adhesion of Streptococcus suis to Host Cells and Its Inhibition by Carbohydrate Ligands.

Cross-platform comparison of glycan microarray formats.

Demystifying O-GlcNAcylation: hints from peptide substrates

Detection of galectin-3 by novel peptidic photoprobes

Detection of pathogenic Streptococcus suis bacteria using magnetic glycoparticles.

Efficient microwave-assisted synthesis of multivalent dendrimeric peptides using cycloaddition reaction (click) chemistry

Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors.

Enhanced Inhibition of Influenza A Virus Adhesion by Di- and Trivalent Hemagglutinin Inhibitors

Enhanced membrane pore formation by multimeric/oligomeric antimicrobial peptides

Enhancing membrane disruption by targeting and multivalent presentation of antimicrobial peptides.

Functional Characterization of Cholera Toxin Inhibitors Using Human Intestinal Organoids

Functional assay for shiga-like toxin via detection by antibody capture and multivalent galabiose binding.

Functionalization of a Rigid Divalent Ligand for LecA, a Bacterial Adhesion Lectin

Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition

Homodimeric galectin-7 (p53-induced gene 1) is a negative growth regulator for human neuroblastoma cells

ITAM-derived phosphopeptide-containing dendrimers as multivalent ligands for Syk tandem SH2 domain.

Identification of laminin-binding motifs of Yersinia pestis plasminogen activator by phage display

Identification of peptide ligands for malignancy- and growth-regulating galectins using random phage-display and designed combinatorial peptide libraries.

Inhibition and detection of galectins.

Inhibition of O-GlcNAc transferase (OGT) by peptidic hybrids

Inhibition of P-fimbriated Escherichia coli adhesion by multivalent galabiose derivatives studied by a live-bacteria application of surface plasmon resonance.

Inhibition of Streptococcus suis adhesion by dendritic galabiose compounds at low nanomolar concentration.

Interference of the galactose-dependent binding of lectins by novel pentapeptide ligands

Intervention with bacterial adhesion by multivalent carbohydrates.

Intracellular Hydrolysis of Small-Molecule O-Linked N-Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition

Lactulose synergizes with CpG-ODN to modulate epithelial and immune cells cross talk

Maximising multivalency effects in protein-carbohydrate interactions

Measuring O-GlcNAc cleavage by OGA and cell lysates on a peptide microarray

Microwave-assisted, tin-mediated, regioselective 3-O-alkylation of galactosides

Multivalent carbohydrate recognition on a glycodendrimer-functionalized flow-through chip.

Multivalent glycoconjugates as anti-pathogenic agents ⬇️

N-Guanidino Derivatives of 1,5-Dideoxy-1,5-imino-d-xylitol are Potent, Selective, and Stable Inhibitors of β-Glucocerebrosidase

Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase

New properties of wheat bran: anti-biofilm activity and interference with bacteria quorum-sensing systems

Optimizing divalent inhibitors of Pseudomonas aeruginosa lectin LecA by using a rigid spacer.

Orthoester functionalized N-guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase

Peptide microarray analysis of the cross-talk between O-GlcNAcylation and tyrosine phosphorylation

PhoX - an IMAC-enrichable Crosslinking Reagent

PhoX: An IMAC-Enrichable Cross-Linking Reagent

Potent divalent inhibitors with rigid glucose click spacers for Pseudomonas aeruginosa lectin LecA

Potential scorpionate antibiotics: targeted hydrolysis of lipid II containing model membranes by vancomycin-TACzyme conjugates and modulation of their antibacterial activity by Zn-ions.

Probing the Inhibitor versus Chaperone Properties of sp2-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease

Rapid screening of lectins for multivalency effects with a glycodendrimer microarray

Rationally Designed Chemically Modified Glycodendrimer Inhibits Streptococcus suis Adhesin SadP at Picomolar Concentrations.

Rigidified multivalent lactose molecules and their interactions with mammalian galectins: a route to selective inhibitors.

Site-specific conjugation of single domain antibodies to liposomes enhances photosensitizer uptake and photodynamic therapy efficacy.

Strong Inhibition of Cholera Toxin B Subunit by Affordable, Polymer-Based Multivalent Inhibitors

Strong Inhibition of Cholera Toxin by Multivalent GM1 Derivatives

Strong inhibition of cholera toxin binding by galactose dendrimers.

Structural Insight into Multivalent Galactoside Binding to Pseudomonas aeruginosa Lectin LecA

Study of cross talk between phosphatases and OGA on a ZO-3-derived peptide

Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics

Synthesis and cholera toxin binding properties of multivalent GM1 mimics

Synthesis and evaluation of TAC-based inhibitors of papain as mimics of cystatin B

Synthesis and evaluation of new thiodigalactoside-based chemical probes to label galectin-3.

Synthesis and evaluation of novel macrocyclic antifungal peptides

Synthesis of multivalent Streptococcus suis adhesion inhibitors by enzymatic cleavage of polygalacturonic acid and 'click' conjugation.

Tannic acid mimicking dendrimers as small intestine submucosa stabilizing nanomordants.

Tetra- versus Pentavalent Inhibitors of Cholera Toxin ⬇️

The influence of ligand valency on aggregation mechanisms for inhibiting bacterial toxins.

The vancomycin-nisin(1-12) hybrid restores activity against vancomycin resistant Enterococci

Thiodigalactoside-Bovine Serum Albumin Conjugates as High-Potency Inhibitors of Galectin-3: An Outstanding Example of Multivalent Presentation of Small Molecule Inhibitors.

Thiourea-based spacers in potent divalent inhibitors of Pseudomonas aeruginosa virulence lectin LecA.

Tuning the preference of thiodigalactoside- and lactosamine-based ligands to galectin-3 over galectin-1

Uptake and transport of superparamagnetic iron oxide nanoparticles through human brain capillary endothelial cells

Use of tetravalent galabiose for inhibition of streptococcus suis serotype 2 infection in a mouse model