Lista de obras - Bård Helge Hoff - Dominio Público Uruguay

(1)H and (13)C NMR data of methyl tetra-O-benzoyl-D-pyranosides in acetone-d(6).

artículo científico publicado en 2009

(1)H,(13)C and (19)F NMR data of N-substituted 6-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amines in DMSO-d(6).

artículo científico publicado en 2010

Activity of 6-aryl-pyrrolo[2,3-d]pyrimidine-4-amines to Tetrahymena

artículo científico publicado en 2012

Balancing potency, metabolic stability and permeability in pyrrolopyrimidine-based EGFR inhibitors

artículo científico publicado en 2016

Benzoylated uronic acid building blocks and synthesis of N-uronate conjugates of lamotrigine

artículo científico publicado en 2012

Changes in cellular signaling proteins in extracts from A549, H460, and U2OS cells treated with cisplatin or docetaxel

artículo científico publicado en 2017

Chemo-enzymatic synthesis of the antidepressant duloxetine and its enantiomer

Chiral 6-aryl-furo[2,3-d]pyrimidin-4-amines as EGFR inhibitors

artículo científico publicado en 2016

Chiral N-benzyl-N-methyl-1-(naphthalen-1-yl)ethanamines and their in vitro antifungal activity against Cryptococcus neoformans, Trichophyton mentagrophytes and Trichophyton rubrum

artículo científico publicado en 2013

Economical synthesis of 13C-labeled opiates, cocaine derivatives and selected urinary metabolites by derivatization of the natural products

artículo científico publicado en 2015

Effect of Auxiliary Donors on 3,8-Phenothiazine Dyes for Dye-Sensitized Solar Cells

scientific article published on 07 December 2019

Enantiopure derivatives of 1,2-alkanediols: substrate requirements of lipase B from Candida antarctica

Enantioselectivity, swelling and stability of 4-hydroxyprolinol containing acrylic polymer beads in the asymmetric reduction of ketones

Extended structure-activity study of thienopyrimidine-based EGFR inhibitors with evaluation of drug-like properties.

artículo científico publicado en 2015

Gas chromatographic enantiomer separation of C-3 and C-4 synthons: prediction of absolute configuration from elution order and enzymatic resolution

Identification of fused pyrimidines as interleukin 17 secretion inhibitors

scientific article published on 15 June 2018

Identification of new 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines as highly potent EGFR-TK inhibitors with Src-family activity

artículo científico publicado en 2014

In vitro baselining of new pyrrolopyrimidine EGFR-TK inhibitors with Erlotinib

artículo científico publicado en 2015

Is literature data useful for identifying enzyme catalysts for new substrates? A case study on reduction of 1-aryl-2-alkanoates

artículo científico publicado en 2017

On-column trypsinization allows for re-use of matrix in modified multiplexed inhibitor beads assay

artículo científico publicado en 2017

Optical Rotation Calculations for Fluorinated Alcohols, Amines, Amides and Esters

artículo científico publicado en 2016

Preparation of pharmaceutical important fluorinated 1-arylethanols using isolated enzymes

artículo científico publicado en 2013

Resolution of derivatives of 1,2-propanediol with lipase B from Candida antarctica. Effect of substrate structure, medium, water activity and acyl donor on enantiomeric ratio

artículo científico publicado en 1998

Single-step microwave-assisted hot water extraction of hemicelluloses from selected lignocellulosic materials - A biorefinery approach.

artículo científico publicado en 2017

Solvent Effects on Optical Rotation: On the Balance between Hydrogen Bonding and Shifts in Dihedral Angles.

artículo científico publicado en 2017

Structure-activity study leading to identification of a highly active thienopyrimidine based EGFR inhibitor

artículo científico publicado en 2014

Synthesis and in vitro EGFR (ErbB1) tyrosine kinase inhibitory activity of 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines

artículo científico publicado en 2011

Synthesis of 1,3-dithianes and 1,3-dithiolanes. Baker's yeast reduction and lipase-catalyzed resolution for synthesis of enantiopure derivatives

artículo científico publicado en 1999

Synthesis of Novel 3,6-Dithienyl Diketopyrrolopyrrole Dyes by Direct C‒H Arylation

scientific article published on 18 May 2020

Synthesis of [13C4]-labeled ∆9-tetrahydrocannabinol and 11-nor-9-carboxy-∆9-tetrahydrocannabinol as internal standards for reducing ion suppressing/alteration effects in LC/MS-MS quantification.

artículo científico publicado en 2014

Synthesis of [13C6]-labelled phenethylamine derivatives for drug quantification in biological samples

artículo científico publicado en 2014

Synthesis of the antistroke drug lubeluzole and its enantiomer. Lipase-catalyzed resolution of chiral building block

artículo científico publicado en 2001

Truncated structures used in search for new lead compounds and in a retrospective analysis of thienopyrimidine-based EGFR inhibitors

artículo científico publicado en 2015

Lista de obras de Bård Helge Hoff

(1)H and (13)C NMR data of methyl tetra-O-benzoyl-D-pyranosides in acetone-d(6).

(1)H,(13)C and (19)F NMR data of N-substituted 6-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amines in DMSO-d(6).

Activity of 6-aryl-pyrrolo[2,3-d]pyrimidine-4-amines to Tetrahymena

Balancing potency, metabolic stability and permeability in pyrrolopyrimidine-based EGFR inhibitors

Benzoylated uronic acid building blocks and synthesis of N-uronate conjugates of lamotrigine

Changes in cellular signaling proteins in extracts from A549, H460, and U2OS cells treated with cisplatin or docetaxel

Chemo-enzymatic synthesis of the antidepressant duloxetine and its enantiomer

Chiral 6-aryl-furo[2,3-d]pyrimidin-4-amines as EGFR inhibitors

Chiral N-benzyl-N-methyl-1-(naphthalen-1-yl)ethanamines and their in vitro antifungal activity against Cryptococcus neoformans, Trichophyton mentagrophytes and Trichophyton rubrum

Economical synthesis of 13C-labeled opiates, cocaine derivatives and selected urinary metabolites by derivatization of the natural products

Effect of Auxiliary Donors on 3,8-Phenothiazine Dyes for Dye-Sensitized Solar Cells

Enantiopure derivatives of 1,2-alkanediols: substrate requirements of lipase B from Candida antarctica

Enantioselectivity, swelling and stability of 4-hydroxyprolinol containing acrylic polymer beads in the asymmetric reduction of ketones

Extended structure-activity study of thienopyrimidine-based EGFR inhibitors with evaluation of drug-like properties.

Gas chromatographic enantiomer separation of C-3 and C-4 synthons: prediction of absolute configuration from elution order and enzymatic resolution

Identification of fused pyrimidines as interleukin 17 secretion inhibitors

Identification of new 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines as highly potent EGFR-TK inhibitors with Src-family activity

In vitro baselining of new pyrrolopyrimidine EGFR-TK inhibitors with Erlotinib

Is literature data useful for identifying enzyme catalysts for new substrates? A case study on reduction of 1-aryl-2-alkanoates

On-column trypsinization allows for re-use of matrix in modified multiplexed inhibitor beads assay

Optical Rotation Calculations for Fluorinated Alcohols, Amines, Amides and Esters

Preparation of pharmaceutical important fluorinated 1-arylethanols using isolated enzymes

Resolution of derivatives of 1,2-propanediol with lipase B from Candida antarctica. Effect of substrate structure, medium, water activity and acyl donor on enantiomeric ratio

Single-step microwave-assisted hot water extraction of hemicelluloses from selected lignocellulosic materials - A biorefinery approach.

Solvent Effects on Optical Rotation: On the Balance between Hydrogen Bonding and Shifts in Dihedral Angles.

Structure-activity study leading to identification of a highly active thienopyrimidine based EGFR inhibitor

Synthesis and in vitro EGFR (ErbB1) tyrosine kinase inhibitory activity of 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines

Synthesis of 1,3-dithianes and 1,3-dithiolanes. Baker's yeast reduction and lipase-catalyzed resolution for synthesis of enantiopure derivatives

Synthesis of Novel 3,6-Dithienyl Diketopyrrolopyrrole Dyes by Direct C‒H Arylation

Synthesis of [13C4]-labeled ∆9-tetrahydrocannabinol and 11-nor-9-carboxy-∆9-tetrahydrocannabinol as internal standards for reducing ion suppressing/alteration effects in LC/MS-MS quantification.

Synthesis of [13C6]-labelled phenethylamine derivatives for drug quantification in biological samples

Synthesis of the antistroke drug lubeluzole and its enantiomer. Lipase-catalyzed resolution of chiral building block

Truncated structures used in search for new lead compounds and in a retrospective analysis of thienopyrimidine-based EGFR inhibitors