Lista de obras - James A. Bull - Dominio Público Uruguay

2-(Aryl-sulfonyl)oxetanes as designer 3-dimensional fragments for fragment screening: synthesis and strategies for functionalisation.

artículo científico publicado en 2013

A molecular rotor for measuring viscosity in plasma membranes of live cells.

artículo científico publicado en 2013

Acid-Mediated Ring Expansion of 2,2-Disubstituted Azetidine Carbamates to 6,6-Disubstituted 1,3-Oxazinan-2-ones

artículo científico publicado en 2019

Catalytic enantioselective synthesis of secondary alkylboronate building blocks with and without metals

artículo científico publicado en 2012

Chemical and structural investigation of the paroxetine-human serotonin transporter complex

artículo científico publicado en 2020

Copper catalysed oxidative α-sulfonylation of branched aldehydes using the acid enhanced reactivity of manganese(iv) oxide

scientific article published on 24 March 2020

Copper-catalyzed N-arylation of 2-imidazolines with aryl iodides

artículo científico publicado en 2013

Copper-catalyzed direct alkenylation of N-iminopyridinium ylides

artículo científico publicado en 2010

Diazo-Transfer Reagent 2-Azido-4,6-dimethoxy-1,3,5-triazine Displays Highly Exothermic Decomposition Comparable to Tosyl Azide

scientific article published on 17 April 2019

Divergent Synthesis of Cyclopropane-Containing Lead-Like Compounds, Fragments and Building Blocks through a Cobalt Catalyzed Cyclopropanation of Phenyl Vinyl Sulfide

artículo científico publicado en 2017

Highly Chemoselective NH- and O-Transfer to Thiols Using Hypervalent Iodine Reagents: Synthesis of Sulfonimidates and Sulfonamides.

artículo científico publicado en 2018

Highly cis-selective synthesis of iodo-aziridines using diiodomethyllithium and in situ generated N-Boc-imines

artículo científico publicado en 2012

Imaging phase separation in model lipid membranes through the use of BODIPY based molecular rotors

artículo científico publicado en 2015

Imaging tumor microscopic viscosity in vivo using molecular rotors

artículo científico publicado en 2017

Intramolecular Simmons-Smith cyclopropanation. Studies into the reactivity of alkyl-substituted zinc carbenoids, effect of directing groups and synthesis of bicyclo[n.1.0]alkanes

artículo científico publicado en 2010

Intramolecular palladium(ii)/(iv) catalysed C(sp3)-H arylation of tertiary aldehydes using a transient imine directing group

scientific article published on 01 July 2019

Lithium-Catalyzed Thiol Alkylation with Tertiary and Secondary Alcohols: Synthesis of 3-Sulfanyl-Oxetanes as Bioisosteres.

artículo científico publicado en 2017

Methylene C(sp3)-H β,β'-Diarylation of Cyclohexanecarbaldehydes Promoted by a Transient Directing Group and Pyridone Ligand

artículo científico publicado en 2020

N-4-Pyrimidinyl-1H-indazol-4-amine inhibitors of Lck: indazoles as phenol isosteres with improved pharmacokinetics

artículo científico publicado en 2007

On the Use of Differential Scanning Calorimetry for Thermal Hazard Assessment of New Chemistry: Avoiding Explosive Mistakes

artículo científico publicado en 2020

Oxetanes: Recent Advances in Synthesis, Reactivity, and Medicinal Chemistry.

artículo científico publicado en 2016

Palladium-Catalyzed C(sp3 )-H Arylation of Primary Amines Using a Catalytic Alkyl Acetal to Form a Transient Directing Group

artículo científico publicado en 2018

Palladium-catalyzed cross-coupling of aziridinylmetal species, generated by sulfinyl-magnesium exchange, with aryl bromides: reaction optimization, scope, and kinetic investigations

artículo científico publicado en 2013

Probing supramolecular protein assembly using covalently attached fluorescent molecular rotors.

artículo científico publicado en 2017

Rapid Assembly of Saturated Nitrogen Heterocycles in One-Pot: Diazo-Heterocycle "Stitching" by N-H Insertion and Cyclization

artículo científico publicado en 2018

Regio- and Stereoselective Palladium-Catalyzed C(sp3)-H Arylation of Pyrrolidines and Piperidines with C(3) Directing Groups

artículo científico publicado en 2018

Regio- and stereospecific synthesis of C-3 functionalized proline derivatives by palladium catalyzed directed C(sp3)-H arylation

scientific article published on 05 September 2014

Single operation palladium catalysed C(sp3)-H functionalisation of tertiary aldehydes: investigations into transient imine directing groups

artículo científico publicado en 2017

Stereocontrolled total synthesis of bengazole a: a marine bisoxazole natural product displaying potent antifungal properties

artículo científico publicado en 2006

Stereospecific functionalization of iodoaziridines via unstabilized aziridinyllithiums generated by iodine-lithium exchange

artículo científico publicado en 2014

Structurally Divergent Lithium Catalyzed Friedel-Crafts Reactions on Oxetan-3-ols: Synthesis of 3,3-Diaryloxetanes and 2,3-Dihydrobenzofurans

scientific article published on 10 October 2016

Studies on the synthesis, stability and conformation of 2-sulfonyl-oxetane fragments.

artículo científico publicado en 2015

Surface functionalisation with viscosity-sensitive BODIPY molecular rotor.

artículo científico publicado en 2018

Synthesis and purification of iodoaziridines involving quantitative selection of the optimal stationary phase for chromatography

artículo científico publicado en 2014

Synthesis of 2- and 2,3-substituted pyrazolo[1,5-a]pyridines: scope and mechanistic considerations of a domino direct alkynylation and cyclization of N-iminopyridinium ylides using alkenyl bromides, alkenyl iodides, and alkynes

artículo científico publicado en 2011

Synthesis of 3,3-Diarylazetidines by Calcium(II)-Catalyzed Friedel-Crafts Reaction of Azetidinols with Unexpected Cbz Enhanced Reactivity

artículo científico publicado en 2018

Synthesis of 3-Aryl-3-Sulfanyl Azetidines by Iron-Catalyzed Thiol Alkylation with N-Cbz Azetidinols

scientific article published on 19 April 2019

Synthesis of NH-sulfoximines from sulfides by chemoselective one-pot N- and O-transfers.

artículo científico publicado en 2016

Synthesis of Selenoaziridines: A Study on Stereochemical Outcomes of the Reaction of Aziridine Radicals and Anions Generated from Iodoaziridines

artículo científico publicado en 2019

Synthesis of Substituted 1,4-Dioxenes through O-H Insertion and Cyclization Using Keto-Diazo Compounds

scientific article published on 17 October 2016

Synthesis of Sulfonimidamides from Sulfenamides via an Alkoxy-amino-λ6 -sulfanenitrile Intermediate

scientific article published on 28 August 2019

Synthesis of Sulfoximine Carbamates by Rhodium-Catalyzed Nitrene Transfer of Carbamates to Sulfoxides

artículo científico publicado en 2015

Synthesis of cis-C-iodo-N-tosyl-aziridines using diiodomethyllithium: reaction optimization, product scope and stability, and a protocol for selection of stationary phase for chromatography

artículo científico publicado en 2013

Synthesis of di-, tri-, and tetrasubstituted oxetanes by rhodium-catalyzed O-H insertion and C-C bond-forming cyclization

artículo científico publicado en 2014

Synthesis of diversely functionalised 2,2-disubstituted oxetanes: fragment motifs in new chemical space

artículo científico publicado en 2015

Synthesis of glycosyl sulfoximines by a highly chemo- and stereoselective NH- and O-transfer to thioglycosides

artículo científico publicado en 2020

Thermal Stability and Explosive Hazard Assessment of Diazo Compounds and Diazo Transfer Reagents

artículo científico publicado en 2019

Total Synthesis of Potent Antifungal Marine Bisoxazole Natural Products Bengazoles A and B

artículo científico publicado en 2007

Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides

artículo científico publicado en 2016

Transient imine directing groups for the C-H functionalisation of aldehydes, ketones and amines: an update 2018-2020

artículo científico publicado en 2020

Transient imines as 'next generation' directing groups for the catalytic functionalisation of C-H bonds in a single operation

scientific article published on 25 May 2018

Visualising the membrane viscosity of porcine eye lens cells using molecular rotors

artículo científico publicado en 2017

Lista de obras de James A. Bull

2-(Aryl-sulfonyl)oxetanes as designer 3-dimensional fragments for fragment screening: synthesis and strategies for functionalisation.

A molecular rotor for measuring viscosity in plasma membranes of live cells.

Acid-Mediated Ring Expansion of 2,2-Disubstituted Azetidine Carbamates to 6,6-Disubstituted 1,3-Oxazinan-2-ones

Catalytic enantioselective synthesis of secondary alkylboronate building blocks with and without metals

Chemical and structural investigation of the paroxetine-human serotonin transporter complex

Copper catalysed oxidative α-sulfonylation of branched aldehydes using the acid enhanced reactivity of manganese(iv) oxide

Copper-catalyzed N-arylation of 2-imidazolines with aryl iodides

Copper-catalyzed direct alkenylation of N-iminopyridinium ylides

Diazo-Transfer Reagent 2-Azido-4,6-dimethoxy-1,3,5-triazine Displays Highly Exothermic Decomposition Comparable to Tosyl Azide

Divergent Synthesis of Cyclopropane-Containing Lead-Like Compounds, Fragments and Building Blocks through a Cobalt Catalyzed Cyclopropanation of Phenyl Vinyl Sulfide

Highly Chemoselective NH- and O-Transfer to Thiols Using Hypervalent Iodine Reagents: Synthesis of Sulfonimidates and Sulfonamides.

Highly cis-selective synthesis of iodo-aziridines using diiodomethyllithium and in situ generated N-Boc-imines

Imaging phase separation in model lipid membranes through the use of BODIPY based molecular rotors

Imaging tumor microscopic viscosity in vivo using molecular rotors

Intramolecular Simmons-Smith cyclopropanation. Studies into the reactivity of alkyl-substituted zinc carbenoids, effect of directing groups and synthesis of bicyclo[n.1.0]alkanes

Intramolecular palladium(ii)/(iv) catalysed C(sp3)-H arylation of tertiary aldehydes using a transient imine directing group

Lithium-Catalyzed Thiol Alkylation with Tertiary and Secondary Alcohols: Synthesis of 3-Sulfanyl-Oxetanes as Bioisosteres.

Methylene C(sp3)-H β,β'-Diarylation of Cyclohexanecarbaldehydes Promoted by a Transient Directing Group and Pyridone Ligand

N-4-Pyrimidinyl-1H-indazol-4-amine inhibitors of Lck: indazoles as phenol isosteres with improved pharmacokinetics

On the Use of Differential Scanning Calorimetry for Thermal Hazard Assessment of New Chemistry: Avoiding Explosive Mistakes

Oxetanes: Recent Advances in Synthesis, Reactivity, and Medicinal Chemistry.

Palladium-Catalyzed C(sp3 )-H Arylation of Primary Amines Using a Catalytic Alkyl Acetal to Form a Transient Directing Group

Palladium-catalyzed cross-coupling of aziridinylmetal species, generated by sulfinyl-magnesium exchange, with aryl bromides: reaction optimization, scope, and kinetic investigations

Probing supramolecular protein assembly using covalently attached fluorescent molecular rotors.

Rapid Assembly of Saturated Nitrogen Heterocycles in One-Pot: Diazo-Heterocycle "Stitching" by N-H Insertion and Cyclization

Regio- and Stereoselective Palladium-Catalyzed C(sp3)-H Arylation of Pyrrolidines and Piperidines with C(3) Directing Groups

Regio- and stereospecific synthesis of C-3 functionalized proline derivatives by palladium catalyzed directed C(sp3)-H arylation

Single operation palladium catalysed C(sp3)-H functionalisation of tertiary aldehydes: investigations into transient imine directing groups

Stereocontrolled total synthesis of bengazole a: a marine bisoxazole natural product displaying potent antifungal properties

Stereospecific functionalization of iodoaziridines via unstabilized aziridinyllithiums generated by iodine-lithium exchange

Structurally Divergent Lithium Catalyzed Friedel-Crafts Reactions on Oxetan-3-ols: Synthesis of 3,3-Diaryloxetanes and 2,3-Dihydrobenzofurans

Studies on the synthesis, stability and conformation of 2-sulfonyl-oxetane fragments.

Surface functionalisation with viscosity-sensitive BODIPY molecular rotor.

Synthesis and purification of iodoaziridines involving quantitative selection of the optimal stationary phase for chromatography

Synthesis of 2- and 2,3-substituted pyrazolo[1,5-a]pyridines: scope and mechanistic considerations of a domino direct alkynylation and cyclization of N-iminopyridinium ylides using alkenyl bromides, alkenyl iodides, and alkynes

Synthesis of 3,3-Diarylazetidines by Calcium(II)-Catalyzed Friedel-Crafts Reaction of Azetidinols with Unexpected Cbz Enhanced Reactivity

Synthesis of 3-Aryl-3-Sulfanyl Azetidines by Iron-Catalyzed Thiol Alkylation with N-Cbz Azetidinols

Synthesis of NH-sulfoximines from sulfides by chemoselective one-pot N- and O-transfers.

Synthesis of Selenoaziridines: A Study on Stereochemical Outcomes of the Reaction of Aziridine Radicals and Anions Generated from Iodoaziridines

Synthesis of Substituted 1,4-Dioxenes through O-H Insertion and Cyclization Using Keto-Diazo Compounds

Synthesis of Sulfonimidamides from Sulfenamides via an Alkoxy-amino-λ6 -sulfanenitrile Intermediate

Synthesis of Sulfoximine Carbamates by Rhodium-Catalyzed Nitrene Transfer of Carbamates to Sulfoxides

Synthesis of cis-C-iodo-N-tosyl-aziridines using diiodomethyllithium: reaction optimization, product scope and stability, and a protocol for selection of stationary phase for chromatography

Synthesis of di-, tri-, and tetrasubstituted oxetanes by rhodium-catalyzed O-H insertion and C-C bond-forming cyclization

Synthesis of diversely functionalised 2,2-disubstituted oxetanes: fragment motifs in new chemical space

Synthesis of glycosyl sulfoximines by a highly chemo- and stereoselective NH- and O-transfer to thioglycosides

Thermal Stability and Explosive Hazard Assessment of Diazo Compounds and Diazo Transfer Reagents

Total Synthesis of Potent Antifungal Marine Bisoxazole Natural Products Bengazoles A and B

Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides

Transient imine directing groups for the C-H functionalisation of aldehydes, ketones and amines: an update 2018-2020

Transient imines as 'next generation' directing groups for the catalytic functionalisation of C-H bonds in a single operation

Visualising the membrane viscosity of porcine eye lens cells using molecular rotors