Lista de obras - Jordi Teixidó - Dominio Público Uruguay

2-Methoxy-6-oxo-1,4,5,6-tetrahydropyridine-3-carbonitriles: versatile starting materials for the synthesis of libraries with diverse heterocyclic scaffolds

artículo científico publicado en 2005

4-Amino-2-arylamino-6-(2,6-dichlorophenyl)-pyrido[2,3-d]pyrimidin-7-(8H)-ones as BCR kinase inhibitors for B lymphoid malignancies.

artículo científico publicado en 2014

A captured room temperature stable Wheland intermediate as a key structure for the orthogonal decoration of 4-amino-pyrido[2,3-d]pyrimidin-7(8H)-ones

artículo científico publicado en 2020

A diversity oriented, microwave assisted synthesis of N-substituted 2-hydro-4-amino-pyrido[2,3-d]pyrimidin-7(8H)-ones

artículo científico publicado en 2008

A diversity-oriented synthesis of 3-(2-amino-1,6-dihydro-6-oxo-pyrimidin-5-yl)propanoic esters

artículo científico publicado en 2010

A new and practical method for the synthesis of 6-aryl-5,6-dihydropyrido[2,3-[Formula: see text]]pyrimidine-4,7(3[Formula: see text],8[Formula: see text])-diones.

artículo científico publicado en 2013

A one-pot microwave-assisted synthesis of pyrido[2,3-d]pyrimidines

artículo científico publicado en 2003

A regiospecific synthesis of both positional isomers of 4,6-disubstituted 2-dicyanomethylene-1, 2-dihydropyridin-3-carbonitriles

artículo científico publicado en 2010

ALK and ROS1 as a joint target for the treatment of lung cancer: a review

artículo científico publicado en 2013

APIF: a new interaction fingerprint based on atom pairs and its application to virtual screening.

artículo científico publicado en 2009

An unusual Michael addition of 3,3-dimethoxypropanenitrile to 2-aryl acrylates: a convenient route to 4-unsubstituted 5,6-dihydropyrido[2,3-d]pyrimidines

artículo científico publicado en 2010

C4-C5 fused pyrazol-3-amines: when the degree of unsaturation and electronic characteristics of the fused ring controls regioselectivity in Ullmann and acylation reactions

artículo científico publicado en 2020

Cell-integral-diversity criterion: a proposal for minimizing cluster artifact in cell-based selections

artículo científico publicado en 2007

Clustering and classifying diverse HIV entry inhibitors using a novel consensus shape-based virtual screening approach: further evidence for multiple binding sites within the CCR5 extracellular pocket.

artículo científico publicado en 2008

Comparative study of neural networks and least mean square algorithm applied to the optimization of cosmetic formulations

artículo científico publicado en 2010

Comparison of ligand-based and receptor-based virtual screening of HIV entry inhibitors for the CXCR4 and CCR5 receptors using 3D ligand shape matching and ligand-receptor docking

artículos científicos

Design and analysis of a combinatorial library of HEPT analogues: comparison of selection methodologies and inspection of the actually covered chemical space

artículo científico publicado en 2003

Design and synthesis of two pyrazole libraries based on o-hydroxyacetophenones

artículo científico publicado en 2004

Design, synthesis and biological activity of acyl substituted 3-amino-5-methyl-1,4,5,7-tetrahydropyrazolo[3,4-b]pyridin-6-ones as potential hypnotic drugs

artículo científico publicado en 2005

Design, synthesis and biological evaluation of pyrido[2,3-d]pyrimidin-7-(8H)-ones as HCV inhibitors

artículo científico publicado en 2016

Diethyl 2,7-dibromo-4H,5H- thieno[3,2-b:4,5-b']dipyrrole-3,6- dicarboxylate: a key intermediate for a diversity oriented synthesis of 2,7,12,17-tetraarylporphycenes

artículo científico publicado en 2006

Discovery of novel HIV entry inhibitors for the CXCR4 receptor by prospective virtual screening.

artículo científico publicado en 2009

Discovery of novel non-cyclam polynitrogenated CXCR4 coreceptor inhibitors

artículo científico publicado en 2008

Diverse combinatorial design, synthesis and in vitro evaluation of new HEPT analogues as potential non-nucleoside HIV-1 reverse transcription inhibitors

artículo científico publicado en 2012

Dose-dependent progressive sunscreens. A new strategy for photoprotection?

artículo científico publicado en 2010

Effect of aza substitution on the photophysical and electrochemical properties of porphycenes: Characterization of the near-IR-absorbing photosensitizers 2,7,12,17-tetrakis(p-substituted phenyl)-3,6,13,16-tetraazaporphycenes.

artículo científico publicado en 2006

Highly specific and sensitive pharmacophore model for identifying CXCR4 antagonists. Comparison with docking and shape-matching virtual screening performance.

artículo científico publicado en 2013

Impact of the CXCR4 structure on docking-based virtual screening of HIV entry inhibitors.

artículo científico publicado en 2012

Improving VEGFR-2 Docking-Based Screening by Pharmacophore Postfiltering and Similarity Search Postprocessing ⬇️

artículo científico publicado el 18 de marzo de 2011

Nitrogen positional scanning in tetramines active against HIV-1 as potential CXCR4 inhibitors.

artículo científico publicado en 2015

Noncyclam tetraamines inhibit CXC chemokine receptor type 4 and target glioma-initiating cells

artículo científico publicado en 2012

Novel monocyclam derivatives as HIV entry inhibitors: Design, synthesis, anti-HIV evaluation, and their interaction with the CXCR4 co-receptor.

artículo científico publicado en 2010

On the Applicability of Elastic Network Models for the Study of RNA CUG Trinucleotide Repeat Overexpansion

artículo científico publicado en 2016

Photochemical production and characterisation of the radical ions of tetraphenylporphycenes

artículo científico publicado en 2006

Porphycenes: facts and prospects in photodynamic therapy of cancer.

artículo científico publicado en 2007

Preparative-scale synthesis of two metabolites isolated from soil treated with zoxium fungicide and kerb herbicide

artículo científico publicado en 2002

Pyrido[2,3-d]pyrimidin-7(8H)-ones: Synthesis and Biomedical Applications

scientific article published on 16 November 2019

Quantitative structure-retention relationships applied to liquid chromatography gradient elution method for the determination of carbonyl-2,4-dinitrophenylhydrazone compounds

artículo científico publicado en 2012

Selective hydrolysis of 2,4-diaminopyrimidine systems: a theoretical and experimental insight into an old rule

artículo científico publicado en 2001

Solid phase vs. solution phase differential behavior: formation of a salicylate structure from a malondialdehyde moiety

scientific article published on 01 January 2000

Solid-phase synthesis of 2-substituted 4-amino-7-oxo-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidines: an example of cyclization-assisted cleavage.

artículo científico publicado en 2003

Solid-phase synthesis of a combinatorial library of dihydroceramide analogues and its activity in human alveolar epithelial cells

artículo científico publicado en 2006

Structure-based virtual screening of FGFR inhibitors: cross-decoys and induced-fit effect.

artículo científico publicado en 2007

Studying the binding interactions of allosteric agonists and antagonists of the CXCR4 receptor.

artículo científico publicado en 2015

Synthesis and biological activity of 4-amino-7-oxo-substituted analogues of 5-deaza-5,6,7,8-tetrahydrofolic acid and 5,10-dideaza-5, 6,7,8-tetrahydrofolic acid

artículo científico publicado en 1998

Synthesis and biological activity of 7-oxo substituted analogues of 5-deaza-5,6,7,8-tetrahydrofolic acid (5-DATHF) and 5,10-dideaza-5,6,7,8-tetrahydrofolic acid (DDATHF).

artículo científico publicado en 2001

Synthesis of 2-arylamino substituted 5,6-dihydropyrido[2,3-d]pyrimidine-7(8H)-ones from arylguanidines

artículo científico publicado en 2012

Lista de obras de Jordi Teixidó

2-Methoxy-6-oxo-1,4,5,6-tetrahydropyridine-3-carbonitriles: versatile starting materials for the synthesis of libraries with diverse heterocyclic scaffolds

4-Amino-2-arylamino-6-(2,6-dichlorophenyl)-pyrido[2,3-d]pyrimidin-7-(8H)-ones as BCR kinase inhibitors for B lymphoid malignancies.

A captured room temperature stable Wheland intermediate as a key structure for the orthogonal decoration of 4-amino-pyrido[2,3-d]pyrimidin-7(8H)-ones

A diversity oriented, microwave assisted synthesis of N-substituted 2-hydro-4-amino-pyrido[2,3-d]pyrimidin-7(8H)-ones

A diversity-oriented synthesis of 3-(2-amino-1,6-dihydro-6-oxo-pyrimidin-5-yl)propanoic esters

A new and practical method for the synthesis of 6-aryl-5,6-dihydropyrido[2,3-[Formula: see text]]pyrimidine-4,7(3[Formula: see text],8[Formula: see text])-diones.

A one-pot microwave-assisted synthesis of pyrido[2,3-d]pyrimidines

A regiospecific synthesis of both positional isomers of 4,6-disubstituted 2-dicyanomethylene-1, 2-dihydropyridin-3-carbonitriles

ALK and ROS1 as a joint target for the treatment of lung cancer: a review

APIF: a new interaction fingerprint based on atom pairs and its application to virtual screening.

An unusual Michael addition of 3,3-dimethoxypropanenitrile to 2-aryl acrylates: a convenient route to 4-unsubstituted 5,6-dihydropyrido[2,3-d]pyrimidines

C4-C5 fused pyrazol-3-amines: when the degree of unsaturation and electronic characteristics of the fused ring controls regioselectivity in Ullmann and acylation reactions

Cell-integral-diversity criterion: a proposal for minimizing cluster artifact in cell-based selections

Clustering and classifying diverse HIV entry inhibitors using a novel consensus shape-based virtual screening approach: further evidence for multiple binding sites within the CCR5 extracellular pocket.

Comparative study of neural networks and least mean square algorithm applied to the optimization of cosmetic formulations

Comparison of ligand-based and receptor-based virtual screening of HIV entry inhibitors for the CXCR4 and CCR5 receptors using 3D ligand shape matching and ligand-receptor docking

Design and analysis of a combinatorial library of HEPT analogues: comparison of selection methodologies and inspection of the actually covered chemical space

Design and synthesis of two pyrazole libraries based on o-hydroxyacetophenones

Design, synthesis and biological activity of acyl substituted 3-amino-5-methyl-1,4,5,7-tetrahydropyrazolo[3,4-b]pyridin-6-ones as potential hypnotic drugs

Design, synthesis and biological evaluation of pyrido[2,3-d]pyrimidin-7-(8H)-ones as HCV inhibitors

Diethyl 2,7-dibromo-4H,5H- thieno[3,2-b:4,5-b']dipyrrole-3,6- dicarboxylate: a key intermediate for a diversity oriented synthesis of 2,7,12,17-tetraarylporphycenes

Discovery of novel HIV entry inhibitors for the CXCR4 receptor by prospective virtual screening.

Discovery of novel non-cyclam polynitrogenated CXCR4 coreceptor inhibitors

Diverse combinatorial design, synthesis and in vitro evaluation of new HEPT analogues as potential non-nucleoside HIV-1 reverse transcription inhibitors

Dose-dependent progressive sunscreens. A new strategy for photoprotection?

Effect of aza substitution on the photophysical and electrochemical properties of porphycenes: Characterization of the near-IR-absorbing photosensitizers 2,7,12,17-tetrakis(p-substituted phenyl)-3,6,13,16-tetraazaporphycenes.

Highly specific and sensitive pharmacophore model for identifying CXCR4 antagonists. Comparison with docking and shape-matching virtual screening performance.

Impact of the CXCR4 structure on docking-based virtual screening of HIV entry inhibitors.

Improving VEGFR-2 Docking-Based Screening by Pharmacophore Postfiltering and Similarity Search Postprocessing ⬇️

Nitrogen positional scanning in tetramines active against HIV-1 as potential CXCR4 inhibitors.

Noncyclam tetraamines inhibit CXC chemokine receptor type 4 and target glioma-initiating cells

Novel monocyclam derivatives as HIV entry inhibitors: Design, synthesis, anti-HIV evaluation, and their interaction with the CXCR4 co-receptor.

On the Applicability of Elastic Network Models for the Study of RNA CUG Trinucleotide Repeat Overexpansion

Photochemical production and characterisation of the radical ions of tetraphenylporphycenes

Porphycenes: facts and prospects in photodynamic therapy of cancer.

Preparative-scale synthesis of two metabolites isolated from soil treated with zoxium fungicide and kerb herbicide

Pyrido[2,3-d]pyrimidin-7(8H)-ones: Synthesis and Biomedical Applications

Quantitative structure-retention relationships applied to liquid chromatography gradient elution method for the determination of carbonyl-2,4-dinitrophenylhydrazone compounds

Selective hydrolysis of 2,4-diaminopyrimidine systems: a theoretical and experimental insight into an old rule

Solid phase vs. solution phase differential behavior: formation of a salicylate structure from a malondialdehyde moiety

Solid-phase synthesis of 2-substituted 4-amino-7-oxo-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidines: an example of cyclization-assisted cleavage.

Solid-phase synthesis of a combinatorial library of dihydroceramide analogues and its activity in human alveolar epithelial cells

Structure-based virtual screening of FGFR inhibitors: cross-decoys and induced-fit effect.

Studying the binding interactions of allosteric agonists and antagonists of the CXCR4 receptor.

Synthesis and biological activity of 4-amino-7-oxo-substituted analogues of 5-deaza-5,6,7,8-tetrahydrofolic acid and 5,10-dideaza-5, 6,7,8-tetrahydrofolic acid

Synthesis and biological activity of 7-oxo substituted analogues of 5-deaza-5,6,7,8-tetrahydrofolic acid (5-DATHF) and 5,10-dideaza-5,6,7,8-tetrahydrofolic acid (DDATHF).

Synthesis of 2-arylamino substituted 5,6-dihydropyrido[2,3-d]pyrimidine-7(8H)-ones from arylguanidines