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Lista de obras de Matthieu Desroses

Correction to Piperazin-1-ylpyridazine Derivatives Are a Novel Class of Human dCTP Pyrophosphatase 1 Inhibitors

artículo científico publicado en 2017

Corrigendum: MTH1 inhibition eradicates cancer by preventing sanitation of the dNTP pool

artículo científico publicado en 2017

Crystal structure of human MTH1 and the 8-oxo-dGMP product complex

artículo científico publicado en 2011

Crystal structure, biochemical and cellular activities demonstrate separate functions of MTH1 and MTH2

scientific journal article

DXR inhibition by potent mono- and disubstituted fosmidomycin analogues

artículo científico publicado en 2013

Derivatives of Iressa, a specific epidermal growth factor receptor inhibitor, are powerful apoptosis inducers in PC3 prostatic cancer cells

artículo científico publicado en 2007

Development of a chemical probe against NUDT15

artículo científico publicado en 2020

Discovery of novel N-phenylphenoxyacetamide derivatives as EthR inhibitors and ethionamide boosters by combining high-throughput screening and synthesis

artículo científico publicado en 2012

Ethionamide boosters. 2. Combining bioisosteric replacement and structure-based drug design to solve pharmacokinetic issues in a series of potent 1,2,4-oxadiazole EthR inhibitors

artículo científico publicado en 2012

Ethionamide boosters: synthesis, biological activity, and structure-activity relationships of a series of 1,2,4-oxadiazole EthR inhibitors

artículo científico publicado en 2011

Exploring drug target flexibility using in situ click chemistry: application to a mycobacterial transcriptional regulator

artículo científico publicado en 2010

MTH1 inhibition eradicates cancer by preventing sanitation of the dNTP pool

artículo científico publicado en 2014

Piperazin-1-ylpyridazine Derivatives Are a Novel Class of Human dCTP Pyrophosphatase 1 Inhibitors

artículo científico publicado en 2017

Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420.

artículo científico publicado en 2017

STAT3 differential scanning fluorimetry and differential scanning light scattering assays: Addressing a missing link in the characterization of STAT3 inhibitor interactions

artículo científico publicado en 2018

Structural analysis of the interaction between spiroisoxazoline SMARt-420 and the Mycobacterium tuberculosis repressor EthR2.

artículo científico publicado en 2017

Structure-metabolism-relationships in the microsomal clearance of piperazin-1-ylpyridazines

artículo científico publicado en 2017

Synthetic EthR inhibitors boost antituberculous activity of ethionamide

artículo científico publicado en 2009

The Next Step Forward in Ubiquitin-Specific Protease 7 Selective Inhibition

artículo científico publicado en 2017

Vinylic MIDA Boronates: New Building Blocks for the Synthesis of Aza-Heterocycles

artículo científico publicado en 2015

dUTPase inhibition augments replication defects of 5-Fluorouracil.

artículo científico publicado en 2017