Lista de obras - Tom D. Sheppard - Dominio Público Uruguay

A general procedure for the synthesis of enones via gold-catalyzed Meyer-Schuster rearrangement of propargylic alcohols at room temperature

scientific article published on 25 January 2011

A lactate-derived chiral aldehyde for determining the enantiopurity of enantioenriched primary amines

artículo científico publicado en 2015

A rapid route to aminocyclopropanes via carbamatoorganozinc carbenoids.

artículo científico publicado en 2013

A series of α7 nicotinic acetylcholine receptor allosteric modulators with close chemical similarity but diverse pharmacological properties

artículo científico publicado en 2012

Aminopolyols from Carbohydrates: Amination of Sugars and Sugar-Derived Tetrahydrofurans with Transaminases

artículo científico publicado el 14 de febrero de 2019

An Accessible Method for DFT Calculation of 11B NMR Shifts of Organoboron Compounds

artículo científico publicado en 2018

An alternative approach to aldol reactions: gold-catalyzed formation of boron enolates from alkynes

artículo científico publicado en 2010

B(OCH2CF3)3-mediated direct amidation of pharmaceutically relevant building blocks in cyclopentyl methyl ether

scientific article published on 14 September 2015

Borate esters as convenient reagents for direct amidation of carboxylic acids and transamidation of primary amides

scientific article published on 06 January 2011

Borate esters: Simple catalysts for the sustainable synthesis of complex amides

artículo científico publicado en 2017

Catalytic direct amidations in tert-butyl acetate using B(OCH2CF3)3

artículo científico publicado en 2019

Chiral Glycolate Equivalents for the Asymmetric Synthesis of α-Hydroxycarbonyl Compounds

article

Data on a thermostable enzymatic one-pot reaction for the production of a high-value compound from l-arabinose

artículo científico publicado en 2018

Dihalohydration of Alkynols: A Versatile Approach to Diverse Halogenated Molecules

artículo científico publicado en 2018

Direct amidation of unprotected amino acids using B(OCH2CF3)3.

artículo científico publicado en 2016

Direct synthesis of amides from carboxylic acids and amines using B(OCH2CF3)3.

artículo científico publicado en 2013

Diversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural Model.

artículo científico publicado en 2017

Functionalised tetrahydrofuran fragments from carbohydrates or sugar beet pulp biomass

article by Laure Benhamou et al published 2019 in Green Chemistry

Gold catalysed synthesis of 3-alkoxyfurans at room temperature

artículo científico publicado en 2014

Gold- and silver-catalyzed reactions of propargylic alcohols in the presence of protic additives

scientific article published on 28 February 2012

Gold-Catalyzed Hydroamination of Propargylic Alcohols: Controlling Divergent Catalytic Reaction Pathways To Access 1,3-Amino Alcohols, 3-Hydroxyketones, or 3-Aminoketones

scientific article published on 28 August 2019

Gold-Catalyzed Hydrophenoxylation of Propargylic Alcohols and Amines: Synthesis of Phenyl Enol Ethers

artículo científico publicado en 2019

HBF4-Catalysed Nucleophilic Substitutions of Propargylic Alcohols

artículo científico publicado en 2015

Highly Diastereoselective Lithium Enolate Aldol Reactions of Butane-2,3-diacetal Desymmetrized Glycolic Acid and Deprotection to Enantiopureanti-2,3-Dihydroxy Esters

artículo científico publicado en 2001

Highly Regioselective Synthesis of Substituted Isoindolinones via Ruthenium-Catalyzed Alkyne Cyclotrimerizations.

artículo científico publicado en 2013

Identification by virtual screening and functional characterisation of novel positive and negative allosteric modulators of the α7 nicotinic acetylcholine receptor

scientific article published on 20 July 2018

Intercepting the Gold-Catalysed Meyer-Schuster Rearrangement by Controlled Protodemetallation: A Regioselective Hydration of Propargylic Alcohols

artículo científico publicado en 2016

Irreversible endo-selective diels-alder reactions of substituted alkoxyfurans: a general synthesis of endo-cantharimides

artículo científico publicado en 2015

Mechanistic insights into boron-catalysed direct amidation reactions.

artículo científico publicado en 2018

Metal-catalysed halogen exchange reactions of aryl halides

artículo científico publicado en 2009

Michael, Michael-aldol and Michael-Michael reactions of enolate equivalents of butane-2,3-diacetal protected glycolic acid derivatives

artículo científico publicado en 2005

Motional timescale predictions by molecular dynamics simulations: case study using proline and hydroxyproline sidechain dynamics.

artículo científico publicado en 2013

One-pot, two-step transaminase and transketolase synthesis of l-gluco-heptulose from l-arabinose

artículo científico publicado en 2018

Prebiotic synthesis of cysteine peptides that catalyze peptide ligation in neutral water

artículo científico publicado en 2020

Preparation of enantiopure butane-2,3-diacetals of glycolic acid and alkylation reactions leading to α-hydroxyacid and amide derivatives

Protecting-Group-Free Amidation of Amino Acids using Lewis Acid Catalysts.

artículo científico publicado en 2018

Rapid assembly of functionalised spirocyclic indolines by palladium-catalysed dearomatising diallylation of indoles with allyl acetate.

artículo científico publicado en 2014

Rapid synthesis of highly functionalised α-amino amides and medium ring lactones using multicomponent reactions of amino alcohols and isocyanides

scientific article published on 10 November 2011

Regioselective dihalohydration reactions of propargylic alcohols: gold-catalyzed and noncatalyzed reactions

artículo científico publicado en 2014

Silver-Free Palladium-Catalyzed C(sp3)-H Arylation of Saturated Bicyclic Amine Scaffolds

artículo científico publicado en 2017

Structurally similar allosteric modulators of α7 nicotinic acetylcholine receptors exhibit five distinct pharmacological effects.

artículo científico publicado en 2014

Studies on the generation of enolate anions from butane-2,3-diacetal protected glycolic acid derivatives and subsequent highly diastereoselective coupling reactions with aldehydes and acid chlorides

Sustainable Synthesis of Chiral Tetrahydrofurans through the Selective Dehydration of Pentoses.

artículo científico publicado en 2015

Synthesis of a Ceramide Sphingolipid as a Potential Sex Pheromone of the Hair CrabErimacrus isenbeckiiUsing Butane-2,3-diacetal Desymmetrised Glycolic Acid Building Blocks

Synthesis of substituted benzooxaborinin-1-ols via palladium-catalysed cyclisation of alkenyl- and alkynyl-boronic acids

scientific article published on 10 August 2016

The application of design of experiments (DoE) reaction optimisation and solvent selection in the development of new synthetic chemistry

artículo científico publicado en 2015

The development and application of synthetic affinity ligands for the purification of ferritin-based influenza antigens.

artículo científico publicado en 2017

The influence of allosteric modulators and transmembrane mutations on desensitisation and activation of α7 nicotinic acetylcholine receptors

artículo científico publicado en 2015

Lista de obras de Tom D. Sheppard

A general procedure for the synthesis of enones via gold-catalyzed Meyer-Schuster rearrangement of propargylic alcohols at room temperature

A lactate-derived chiral aldehyde for determining the enantiopurity of enantioenriched primary amines

A rapid route to aminocyclopropanes via carbamatoorganozinc carbenoids.

A series of α7 nicotinic acetylcholine receptor allosteric modulators with close chemical similarity but diverse pharmacological properties

Aminopolyols from Carbohydrates: Amination of Sugars and Sugar-Derived Tetrahydrofurans with Transaminases

An Accessible Method for DFT Calculation of 11B NMR Shifts of Organoboron Compounds

An alternative approach to aldol reactions: gold-catalyzed formation of boron enolates from alkynes

B(OCH2CF3)3-mediated direct amidation of pharmaceutically relevant building blocks in cyclopentyl methyl ether

Borate esters as convenient reagents for direct amidation of carboxylic acids and transamidation of primary amides

Borate esters: Simple catalysts for the sustainable synthesis of complex amides

Catalytic direct amidations in tert-butyl acetate using B(OCH2CF3)3

Chiral Glycolate Equivalents for the Asymmetric Synthesis of α-Hydroxycarbonyl Compounds

Data on a thermostable enzymatic one-pot reaction for the production of a high-value compound from l-arabinose

Dihalohydration of Alkynols: A Versatile Approach to Diverse Halogenated Molecules

Direct amidation of unprotected amino acids using B(OCH2CF3)3.

Direct synthesis of amides from carboxylic acids and amines using B(OCH2CF3)3.

Diversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural Model.

Functionalised tetrahydrofuran fragments from carbohydrates or sugar beet pulp biomass

Gold catalysed synthesis of 3-alkoxyfurans at room temperature

Gold- and silver-catalyzed reactions of propargylic alcohols in the presence of protic additives

Gold-Catalyzed Hydroamination of Propargylic Alcohols: Controlling Divergent Catalytic Reaction Pathways To Access 1,3-Amino Alcohols, 3-Hydroxyketones, or 3-Aminoketones

Gold-Catalyzed Hydrophenoxylation of Propargylic Alcohols and Amines: Synthesis of Phenyl Enol Ethers

HBF4-Catalysed Nucleophilic Substitutions of Propargylic Alcohols

Highly Diastereoselective Lithium Enolate Aldol Reactions of Butane-2,3-diacetal Desymmetrized Glycolic Acid and Deprotection to Enantiopureanti-2,3-Dihydroxy Esters

Highly Regioselective Synthesis of Substituted Isoindolinones via Ruthenium-Catalyzed Alkyne Cyclotrimerizations.

Identification by virtual screening and functional characterisation of novel positive and negative allosteric modulators of the α7 nicotinic acetylcholine receptor

Intercepting the Gold-Catalysed Meyer-Schuster Rearrangement by Controlled Protodemetallation: A Regioselective Hydration of Propargylic Alcohols

Irreversible endo-selective diels-alder reactions of substituted alkoxyfurans: a general synthesis of endo-cantharimides

Mechanistic insights into boron-catalysed direct amidation reactions.

Metal-catalysed halogen exchange reactions of aryl halides

Michael, Michael-aldol and Michael-Michael reactions of enolate equivalents of butane-2,3-diacetal protected glycolic acid derivatives

Motional timescale predictions by molecular dynamics simulations: case study using proline and hydroxyproline sidechain dynamics.

One-pot, two-step transaminase and transketolase synthesis of l-gluco-heptulose from l-arabinose

Prebiotic synthesis of cysteine peptides that catalyze peptide ligation in neutral water

Preparation of enantiopure butane-2,3-diacetals of glycolic acid and alkylation reactions leading to α-hydroxyacid and amide derivatives

Protecting-Group-Free Amidation of Amino Acids using Lewis Acid Catalysts.

Rapid assembly of functionalised spirocyclic indolines by palladium-catalysed dearomatising diallylation of indoles with allyl acetate.

Rapid synthesis of highly functionalised α-amino amides and medium ring lactones using multicomponent reactions of amino alcohols and isocyanides

Regioselective dihalohydration reactions of propargylic alcohols: gold-catalyzed and noncatalyzed reactions

Silver-Free Palladium-Catalyzed C(sp3)-H Arylation of Saturated Bicyclic Amine Scaffolds

Structurally similar allosteric modulators of α7 nicotinic acetylcholine receptors exhibit five distinct pharmacological effects.

Studies on the generation of enolate anions from butane-2,3-diacetal protected glycolic acid derivatives and subsequent highly diastereoselective coupling reactions with aldehydes and acid chlorides

Sustainable Synthesis of Chiral Tetrahydrofurans through the Selective Dehydration of Pentoses.

Synthesis of a Ceramide Sphingolipid as a Potential Sex Pheromone of the Hair CrabErimacrus isenbeckiiUsing Butane-2,3-diacetal Desymmetrised Glycolic Acid Building Blocks

Synthesis of substituted benzooxaborinin-1-ols via palladium-catalysed cyclisation of alkenyl- and alkynyl-boronic acids

The application of design of experiments (DoE) reaction optimisation and solvent selection in the development of new synthetic chemistry

The development and application of synthetic affinity ligands for the purification of ferritin-based influenza antigens.

The influence of allosteric modulators and transmembrane mutations on desensitisation and activation of α7 nicotinic acetylcholine receptors