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Lista de obras de Laurence Goossens

1-[4-(Methylsulfonyl)phenyl]-5-phenyl-1H-pyrazole derivatives

artículo científico publicado en 2004

A new synthesis of pyrrolo[3,2-b]quinolines by a tandem electrocyclization–oxidation process

Antiproliferative effects of isopentenylated coumarins isolated from Phellolophium madagascariense Baker

artículo científico publicado en 2006

Antispasmodic and antioxidant activities of fractions and bioactive constituent davidigenin isolated from Mascarenhasia arborescens.

artículo científico publicado en 2010

COX-2/5-LOX dual acting anti-inflammatory drugs in cancer chemotherapy.

artículo científico publicado en 2007

Chemotaxonomic interest of iridoids isolated from a Malagasy species: Perichlaena richardii

artículo científico publicado en 2011

Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance

artículo científico publicado en 2017

DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge

artículo científico publicado en 2017

Discovery of orally bioavailable NK1 receptor antagonists

artículo científico publicado en 2003

Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors

artículo científico publicado en 2011

Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitors.

artículo científico publicado en 2014

New NSAIDs-NO hybrid molecules with antiproliferative properties on human prostatic cancer cell lines.

artículo científico publicado en 2008

Quinazoline derivatives as anticancer drugs: a patent review (2011 - present).

artículo científico

Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer.

artículo científico publicado en 2010

Synthesis and activity of a new methoxytetrahydropyran derivative as dual cyclooxygenase-2/5-lipoxygenase inhibitor

artículo científico publicado en 2002

Synthesis and biological evaluation of a new family of anti-benzylanilinosulfonamides as CA IX inhibitors

artículo científico publicado en 2008

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

artículo científico publicado en 2015

Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.

artículo científico publicado en 2012

[4-(6,7-Disubstituted quinazolin-4-ylamino)phenyl] carbamic acid esters: a novel series of dual EGFR/VEGFR-2 tyrosine kinase inhibitors