Lista de obras - Akihiro Sugawara - Dominio Público Uruguay

5-O-Mycaminosyltylonolide antibacterial derivatives: design, synthesis and bioactivity

artículo científico publicado en 2017

An inducible cell-cell fusion system with integrated ability to measure the efficiency and specificity of HIV-1 entry inhibitors

artículo científico publicado en 2011

Argifin; efficient solid phase total synthesis and evaluation of analogues of acyclic peptide

artículo científico publicado en 2009

Associating HIV-1 envelope glycoprotein structures with states on the virus observed by smFRET

scientific article published on 10 April 2019

Asymmetric Total Synthesis of Indole Alkaloids Containing an Indoline Spiroaminal Framework

artículo científico publicado en 2015

Asymmetric total synthesis of neoxaline

artículo científico publicado en 2013

Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A(H1N1)pdm09 virus infection by interfering with virus internalization process

artículo científico publicado en 2019

Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites

artículo científico publicado en 2013

Cinatrins D and E, and virgaricin B, three novel compounds produced by a fungus, Virgaria boninensis FKI-4958. ⬇️

artículo científico publicado en 2015

Computational analysis of the binding affinities of the natural-product cyclopentapeptides argifin and argadin to chitinase B from Serratia marcescens

artículo científico publicado en 2008

Computer-aided rational molecular design of argifin-derivatives with increased inhibitory activity against chitinase B from Serratia marcescens.

artículo científico publicado en 2009

Creation of Customized Bioactivity within a 14-Membered Macrolide Scaffold: Design, Synthesis, and Biological Evaluation Using a Family-18 Chitinase

artículo científico publicado en 2015

Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site

artículo científico publicado en 2014

Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity

artículo científico publicado en 2007

Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening

artículo científico publicado en 2010

Human acidic mammalian chitinase as a novel target for anti-asthma drug design using in silico screening

artículo científico publicado en 2013

Jietacins, azoxy antibiotics with potent nematocidal activity: Design, synthesis, and biological evaluation against parasitic nematodes

artículo científico publicado en 2017

Jietacins, azoxy natural products, as novel NF-κB inhibitors: Discovery, synthesis, biological activity, and mode of action

artículo científico publicado en 2019

Leucomycin A3, a 16-membered macrolide antibiotic, inhibits influenza A virus infection and disease progression.

artículo científico publicado en 2014

Macrolides Promote CCL2-Mediated Macrophage Recruitment and Clearance of Nasopharyngeal Pneumococcal Colonization in Mice

artículo científico publicado en 2015

Macrolides sensitize EGFR-TKI-induced non-apoptotic cell death via blocking autophagy flux in pancreatic cancer cell lines.

artículo científico publicado en 2015

Macrolides with promotive activity of monocyte to macrophage differentiation

artículo científico publicado en 2005

Molecular modeling of human acidic mammalian chitinase in complex with the natural-product cyclopentapeptide chitinase inhibitor argifin

artículo científico publicado en 2009

NMR spectroscopy and computational analysis of interaction between Serratia marcescens chitinase B and a dipeptide derived from natural-product cyclopentapeptide chitinase inhibitor argifin ⬇️

artículo científico publicado el 15 de agosto de 2010

Non-antibiotic 12-membered macrolides: design, synthesis and biological evaluation in a cigarette-smoking model

artículo científico publicado en 2015

Novel 12-membered non-antibiotic macrolides from erythromycin A; EM900 series as novel leads for anti-inflammatory and/or immunomodulatory agents

scientific article published on 07 April 2011

Novel 12-membered non-antibiotic macrolides, EM900 series with anti-inflammatory and/or immunomodulatory activity; synthesis, structure-activity relationships and in vivo study

artículo científico publicado en 2012

Solid-phase total synthesis of the chitinase inhibitor Argadin using a supported acetal resin.

artículo científico publicado en 2009

Three-Dimensional Solution Structure of Bottromycin A2: A Potent Antibiotic Active against Methicillin-Resistant Staphylococcus aureus and Vancomycin-Resistant Enterococci ⬇️

artículo científico publicado el 1 de enero de 2012

Three-dimensional solution structure of EM703 with potent promoting activity of monocyte-to-macrophage differentiation

artículo científico publicado en 2006

Total syntheses of the AChE inhibitors (-)-arisugacins F and G

scientific article published on 01 August 2003

Toward the total synthesis of luminamicin; an anaerobic antibiotic: construction of highly functionalized cis-decalin containing a bridged ether moiety

artículo científico publicado en 2017

Two New Terpenes Isolated from Dictyostelium Cellular Slime Molds

artículo científico publicado en 2020

Lista de obras de Akihiro Sugawara

5-O-Mycaminosyltylonolide antibacterial derivatives: design, synthesis and bioactivity

An inducible cell-cell fusion system with integrated ability to measure the efficiency and specificity of HIV-1 entry inhibitors

Argifin; efficient solid phase total synthesis and evaluation of analogues of acyclic peptide

Associating HIV-1 envelope glycoprotein structures with states on the virus observed by smFRET

Asymmetric Total Synthesis of Indole Alkaloids Containing an Indoline Spiroaminal Framework

Asymmetric total synthesis of neoxaline

Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A(H1N1)pdm09 virus infection by interfering with virus internalization process

Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites

Cinatrins D and E, and virgaricin B, three novel compounds produced by a fungus, Virgaria boninensis FKI-4958. ⬇️

Computational analysis of the binding affinities of the natural-product cyclopentapeptides argifin and argadin to chitinase B from Serratia marcescens

Computer-aided rational molecular design of argifin-derivatives with increased inhibitory activity against chitinase B from Serratia marcescens.

Creation of Customized Bioactivity within a 14-Membered Macrolide Scaffold: Design, Synthesis, and Biological Evaluation Using a Family-18 Chitinase

Crystal Structures of HIV-1 gp120 Envelope Glycoprotein in Complex with NBD Analogues That Target the CD4-Binding Site

Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity

Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening

Human acidic mammalian chitinase as a novel target for anti-asthma drug design using in silico screening

Jietacins, azoxy antibiotics with potent nematocidal activity: Design, synthesis, and biological evaluation against parasitic nematodes

Jietacins, azoxy natural products, as novel NF-κB inhibitors: Discovery, synthesis, biological activity, and mode of action

Leucomycin A3, a 16-membered macrolide antibiotic, inhibits influenza A virus infection and disease progression.

Macrolides Promote CCL2-Mediated Macrophage Recruitment and Clearance of Nasopharyngeal Pneumococcal Colonization in Mice

Macrolides sensitize EGFR-TKI-induced non-apoptotic cell death via blocking autophagy flux in pancreatic cancer cell lines.

Macrolides with promotive activity of monocyte to macrophage differentiation

Molecular modeling of human acidic mammalian chitinase in complex with the natural-product cyclopentapeptide chitinase inhibitor argifin

NMR spectroscopy and computational analysis of interaction between Serratia marcescens chitinase B and a dipeptide derived from natural-product cyclopentapeptide chitinase inhibitor argifin ⬇️

Non-antibiotic 12-membered macrolides: design, synthesis and biological evaluation in a cigarette-smoking model

Novel 12-membered non-antibiotic macrolides from erythromycin A; EM900 series as novel leads for anti-inflammatory and/or immunomodulatory agents

Novel 12-membered non-antibiotic macrolides, EM900 series with anti-inflammatory and/or immunomodulatory activity; synthesis, structure-activity relationships and in vivo study

Solid-phase total synthesis of the chitinase inhibitor Argadin using a supported acetal resin.

Three-Dimensional Solution Structure of Bottromycin A2: A Potent Antibiotic Active against Methicillin-Resistant Staphylococcus aureus and Vancomycin-Resistant Enterococci ⬇️

Three-dimensional solution structure of EM703 with potent promoting activity of monocyte-to-macrophage differentiation

Total syntheses of the AChE inhibitors (-)-arisugacins F and G

Toward the total synthesis of luminamicin; an anaerobic antibiotic: construction of highly functionalized cis-decalin containing a bridged ether moiety

Two New Terpenes Isolated from Dictyostelium Cellular Slime Molds