Lista de obras - Salvatore Ferla - Dominio Público Uruguay

3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization

scholarly article by Romeo Romagnoli published in October 2018

A new antiviral scaffold for human norovirus identified with computer-aided approaches on the viral polymerase

scientific article published on 05 December 2019

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

artículo científico publicado en 2019

Broad-spectrum non-nucleoside inhibitors for caliciviruses.

artículo científico publicado en 2017

Combining bioinformatics, cheminformatics, functional genomics and whole organism approaches for identifying epigenetic drug targets in Schistosoma mansoni

scientific article published on 13 November 2018

Computational Studies towards the Identification of Novel Rhodopsin-Binding Compounds as Chemical Chaperones for Misfolded Opsins

artículo científico publicado en 2020

Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3',4',5'-Trimethoxyphenyl)-2-Aryl-1H-Imidazole

artículo científico publicado en 2016

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

artículo científico publicado en 2016

Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors

scientific article published on 01 August 2019

Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication

artículo científico publicado en 2016

In silico screening for human norovirus antivirals reveals a novel non-nucleoside inhibitor of the viral polymerase.

artículo científico publicado en 2018

Networks of enzymatically oxidized membrane lipids support calcium-dependent coagulation factor binding to maintain hemostasis.

artículo científico publicado en 2017

Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation

artículo científico publicado en 2014

Novel symmetrical phenylenediamines as potential anti-hepatitis C virus agents.

artículo científico publicado en 2016

Polyfluorinated groups in medicinal chemistry.

artículo científico

Quercetin derivatives as novel antihypertensive agents: Synthesis and physiological characterization

artículo científico publicado en 2015

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

artículo científico publicado en 2016

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

artículo científico publicado en 2017

Small-molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): synthesis and biological evaluation

artículo científico publicado en 2014

Structure-activity relationship study of itraconazole, a broad-range inhibitor of picornavirus replication that targets oxysterol-binding protein (OSBP)

artículo científico publicado en 2018

Synthesis and biological evaluation of 6-substituted-5-fluorouridine ProTides

artículo científico publicado en 2017

Lista de obras de Salvatore Ferla

3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization

A new antiviral scaffold for human norovirus identified with computer-aided approaches on the viral polymerase

A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative agents against prostate cancer

Broad-spectrum non-nucleoside inhibitors for caliciviruses.

Combining bioinformatics, cheminformatics, functional genomics and whole organism approaches for identifying epigenetic drug targets in Schistosoma mansoni

Computational Studies towards the Identification of Novel Rhodopsin-Binding Compounds as Chemical Chaperones for Misfolded Opsins

Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3',4',5'-Trimethoxyphenyl)-2-Aryl-1H-Imidazole

Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer

Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors

Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication

In silico screening for human norovirus antivirals reveals a novel non-nucleoside inhibitor of the viral polymerase.

Networks of enzymatically oxidized membrane lipids support calcium-dependent coagulation factor binding to maintain hemostasis.

Novel styryl-indoles as small molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): Synthesis and biological evaluation

Novel symmetrical phenylenediamines as potential anti-hepatitis C virus agents.

Polyfluorinated groups in medicinal chemistry.

Quercetin derivatives as novel antihypertensive agents: Synthesis and physiological characterization

Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety

Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents.

Small-molecule inhibitors of 25-hydroxyvitamin D-24-hydroxylase (CYP24A1): synthesis and biological evaluation

Structure-activity relationship study of itraconazole, a broad-range inhibitor of picornavirus replication that targets oxysterol-binding protein (OSBP)

Synthesis and biological evaluation of 6-substituted-5-fluorouridine ProTides