Filtros de búsqueda

Lista de obras de Saeed Emami

(E)- and (Z)-1,2,4-triazolylchromanone oxime ethers as conformationally constrained antifungals

artículo científico publicado en 2004

1,2,3-Triazole-based kojic acid analogs as potent tyrosinase inhibitors: Design, synthesis and biological evaluation

scientific article published on 31 October 2018

1,2-Diaryl-2-hydroxyiminoethanones as dual COX-1 and β-amyloid aggregation inhibitors: biological evaluation and in silico study

scientific article published on 11 October 2014

1-[(2-arylthiazol-4-yl)methyl]azoles as a new class of anticonvulsants: design, synthesis, in vivo screening, and in silico drug-like properties.

artículo científico publicado en 2011

2-Amino-4-(nitroalkyl)-4H-chromene-3-carbonitriles as New Cytotoxic Agents

scientific article published on January 2013

2-Hydroxyphenacyl azoles and related azolium derivatives as antifungal agents

artículo científico publicado en 2007

2-Substituted-5-nitroheterocycles: in vitro anti-Helicobacter pylori activity and structure-activity relationship study

artículo científico publicado en 2009

2H-chromene derivatives bearing thiazolidine-2,4-dione, rhodanine or hydantoin moieties as potential anticancer agents.

artículo científico publicado en 2012

3-imidazolyl-substituted flavans as potential antifungal agents: synthesis, stereochemical properties, and antifungal activity.

artículo científico publicado en 2009

5,7-Dihydroxychromone-2-carboxylic acid and it's transition-metal (Mn and Zn) chelates as non-thiol radioprotective agents

artículo científico publicado en 2007

5-Nitroimidazole-based 1,3,4-thiadiazoles: heterocyclic analogs of metronidazole as anti-Helicobacter pylori agents

artículo científico publicado en 2010

9H-Carbazole Derivatives Containing the N-Benzyl-1,2,3-triazole Moiety as New Acetylcholinesterase Inhibitors.

artículo científico publicado en 2015

A new boronic acid fluorescent sensor based on fluorene for monosaccharides at physiological pH

artículo científico publicado en 2015

Acetophenone benzoylhydrazones as antioxidant agents: Synthesis, in vitro evaluation and structure-activity relationship studies

artículo científico publicado en 2018

An overview of azoles targeting sterol 14α-demethylase for antileishmanial therapy

artículo científico publicado en 2017

Anticonvulsant and antiepileptogenic effects of azolylchromanones on lithium-pilocarpine induced seizures and pentylenetetrazole-kindling model of epilepsy

artículo científico publicado en 2007

Antinociceptive properties of new coumarin derivatives bearing substituted 3,4-dihydro-2H-benzothiazines.

artículo científico publicado en 2014

Antituberculosis agents. V. Synthesis, evaluation of in vitro antituberculosis activity and cytotoxicity of some 2-(5-nitro-2-furyl)-1,3,4-thiadiazole derivatives

artículo científico publicado en 2002

Asymmetrical 2,6-bis(benzylidene)cyclohexanones: Synthesis, cytotoxic activity and QSAR study

artículo científico publicado en 2012

Azolylchromans as a novel scaffold for anticonvulsant activity

artículo científico publicado en 2006

Benzofuran-derived benzylpyridinium bromides as potent acetylcholinesterase inhibitors.

artículo científico publicado en 2015

Chromene-based synthetic chalcones as potent antileishmanial agents: synthesis and biological activity

artículo científico publicado en 2010

Complexes of 2-hydroxyacetophenone semicarbazones: A novel series of superoxide dismutase mimetics

artículo científico publicado en 2010

Conformationally constrained analogs of N-substituted piperazinylquinolones: synthesis and antibacterial activity of N-(2,3-dihydro-4-hydroxyimino-4H-1-benzopyran-3-yl)-piperazinylquinolones

artículo científico publicado en 2009

Coumarin-based bioactive compounds: facile synthesis and biological evaluation of coumarin-fused 1,4-thiazepines.

artículo científico publicado en 2011

Current developments of coumarin-based anti-cancer agents in medicinal chemistry.

artículo científico

Cytotoxic Activity and DNA Binding Property of New Aminopyrimidine Derivatives

artículo científico publicado en 2020

Cytotoxic activity evaluation and QSAR study of chromene-based chalcones.

artículo científico publicado en 2012

Design of conformationally constrained azole antifungals: efficient synthesis and antifungal activity of trans-3-imidazolylflavanones

artículo científico publicado en 2009

Design, synthesis and anticholinesterase activity of novel benzylidenechroman-4-ones bearing cyclic amine side chain

artículo científico publicado en 2015

Design, synthesis and biological evaluation of flexible and rigid analogs of 4H-1,2,4-triazoles bearing 3,4,5-trimethoxyphenyl moiety as new antiproliferative agents

artículo científico publicado en 2019

Design, synthesis and evaluation of novel multi-target-directed ligands for treatment of Alzheimer's disease based on coumarin and lipoic acid scaffolds

artículo científico publicado en 2018

Design, synthesis and in vitro study of 5,6-diaryl-1,2,4-triazine-3-ylthioacetate derivatives as COX-2 and β-amyloid aggregation inhibitors.

artículo científico publicado en 2015

Design, synthesis, biological evaluation and docking study of 5-oxo-4,5-dihydropyrano[3,2-c]chromene derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors

artículo científico publicado en 2013

Design, synthesis, in vivo and in silico evaluation of phenacyl triazole hydrazones as new anticonvulsant agents.

artículo científico publicado en 2018

Design, synthesis, pharmacological evaluation, and docking study of new acridone-based 1,2,4-oxadiazoles as potential anticonvulsant agents.

artículo científico publicado en 2016

Discovery of benzylthio analogs of fluconazole as potent antifungal agents.

artículo científico publicado en 2018

Down-regulation of peroxin synthesis by silencing RNA (siRNA): A novel hypothesis for treatment of leishmaniasis

artículo científico publicado en 2016

Experimental Study on the Reduction of Loratadine Particle Size through Confined Liquid Impinging Jets

scientific article published on 20 July 2020

Facile synthesis and antiproliferative activity of 7H-benzo[7,8]chromeno[2,3-d]pyrimidin-8-amines.

artículo científico publicado en 2016

Functionalized N(2-oxyiminoethyl) piperazinyl quinolones as new cytotoxic agents

artículo científico publicado en 2007

Halogenated flavanones as potential apoptosis-inducing agents: synthesis and biological activity evaluation

artículo científico publicado en 2012

Hypothesis: The potential application of doxorubicin against cutaneous leishmaniasis

artículo científico publicado en 2015

Imidazo[2,1-b]thiazole derivatives as new inhibitors of 15-lipoxygenase.

artículo científico publicado en 2014

Imidazolylchromanone oxime ethers as potential anticonvulsant agents: Anticonvulsive evaluation in PTZ-kindling model of epilepsy and SAR study

artículo científico publicado en 2010

Imidazolylchromanones containing alkyl side chain as lanosterol 14α-demethylase inhibitors: synthesis, antifungal activity and docking study.

artículo científico publicado en 2013

Imidazolylchromanones containing non-benzylic oxime ethers: synthesis and molecular modeling study of new azole antifungals selective against Cryptococcus gattii

artículo científico publicado en 2014

In Vitro Activities of Novel Azole Compounds ATTAF-1 and ATTAF-2 against Fluconazole-Susceptible and -Resistant Isolates of Candida Species.

artículo científico publicado en 2016

In vitro and in vivo evaluation of kojic acid against Toxoplasma gondii in experimental models of acute toxoplasmosis

artículo científico publicado en 2019

In vitro antileishmanial activity of novel azoles (3-imidazolylflavanones) against promastigote and amastigote stages of Leishmania major

artículo científico publicado en 2016

Indole in the target-based design of anticancer agents: A versatile scaffold with diverse mechanisms.

artículo científico publicado en 2018

Indole-derived chalcones as anti-dermatophyte agents: In vitro evaluation and in silico study

scientific article published on 23 December 2019

Indolinone-based acetylcholinesterase inhibitors: synthesis, biological activity and molecular modeling.

artículo científico publicado en 2014

Induction of apoptosis through tubulin inhibition in human cancer cells by new chromene-based chalcones

artículo científico publicado en 2012

Isochaihulactone analogues: synthesis and anti-proliferative activity of novel dibenzylbutyrolactones.

artículo científico publicado en 2010

Kojic acid and its manganese and zinc complexes as potential radioprotective agents

artículo científico publicado en 2006

Kojic acid-natural product conjugates as mushroom tyrosinase inhibitors

scientific article published on 16 June 2020

Management of multi-drug resistant Helicobacter pylori infection by supplementary, complementary and alternative medicine; a review.

artículo científico publicado en 2017

Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: synthesis, in vitro antibacterial activity and in silico study.

artículo científico publicado en 2013

Modification of 7-piperazinylquinolone antibacterials to promising anticancer lead compounds: Synthesis and in vitro studies

scientific article published on 15 December 2019

Molecular Modeling and Structural Stability of Wild-Type and Mutant CYP51 from Leishmania major: In Vitro and In Silico Analysis of a Laboratory Strain.

artículo científico publicado en 2018

Multi-structure docking analysis of BACE1 crystal structures and non-peptidic ligands

artículo científico

N-(2-(Piperazin-1-yl)phenyl)arylamide Derivatives as β-Secretase (BACE1) Inhibitors: Simple Synthesis by Ugi Four-Component Reaction and Biological Evaluation

artículo científico publicado en 2015

N-Substituted piperazinyl quinolones as potential cytotoxic agents: structure-activity relationships study

artículo científico publicado en 2008

New 5-(nitroheteroaryl)-1,3,4-thiadiazols containing acyclic amines at C-2: synthesis and SAR study for their antileishmanial activity

artículo científico publicado en 2012

New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents

artículo científico publicado en 2018

New indole-based chalconoids as tubulin-targeting antiproliferative agents.

artículo científico publicado en 2017

New potent antifungal triazole alcohols containing N-benzylpiperazine carbodithioate moiety: Synthesis, in vitro evaluation and in silico study

scientific article published on 12 June 2019

New racemic annulated pyrazolo[1,2-b]phthalazines as tacrine-like AChE inhibitors with potential use in Alzheimer's disease

artículo científico publicado en 2017

New tacrine-derived AChE/BuChE inhibitors: Synthesis and biological evaluation of 5-amino-2-phenyl-4H-pyrano[2,3-b]quinoline-3-carboxylates.

artículo científico publicado en 2017

New tetracyclic tacrine analogs containing pyrano[2,3-c]pyrazole: efficient synthesis, biological assessment and docking simulation study

artículo científico publicado en 2014

New thiazole-2(3H)-thiones containing 4-(3,4,5-trimethoxyphenyl) moiety as anticancer agents

scientific article published on 15 October 2019

Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: synthesis and in vitro biological evaluation

artículo científico publicado en 2008

Novel 3-phenylcoumarin-lipoic acid conjugates as multi-functional agents for potential treatment of Alzheimer's disease

scientific article published on 02 May 2018

Novel Tc-2-arylimidazo[2,1-b]benzothiazole derivatives as SPECT imaging agents for amyloid-β plaques

scientific article published on 29 April 2019

Novel antileishmanial chalconoids: synthesis and biological activity of 1- or 3-(6-chloro-2H-chromen-3-yl)propen-1-ones.

artículo científico publicado en 2009

Novel coumarin-3-carboxamides bearing N-benzylpiperidine moiety as potent acetylcholinesterase inhibitors.

artículo científico publicado en 2013

Novel triazole alcohol antifungals derived from fluconazole: design, synthesis, and biological activity

artículo científico publicado en 2014

One-pot, four-component synthesis of novel cytotoxic agents 1-(5-aryl-1,3,4-oxadiazol-2-yl)-1-(1H-pyrrol-2-yl)methanamines

artículo científico publicado en 2014

Phthalimide-Derived N-Benzylpyridinium Halides Targeting Cholinesterases: Synthesis and Bioactivity of New Potential Anti-Alzheimer's Disease Agents.

artículo científico publicado en 2016

Polyoxygenated cinnamoylcoumarins as conformationally constrained analogs of cytotoxic diarylpentanoids: synthesis and biological activity.

artículo científico publicado en 2013

Promising antileishmanial activity of novel imidazole antifungal drug luliconazole against Leishmania major: In vitro and in silico studies

artículo científico publicado en 2018

Promising antileishmanial effectiveness of doxorubicin and Doxil against Leishmania major: An in vitro assay

artículo científico publicado en 2017

Quinoline-based imidazole-fused heterocycles as new inhibitors of 15-lipoxygenase.

artículo científico publicado en 2016

Radioprotective effects of kojic acid against mortality induced by gamma irradiation in mice.

artículo científico publicado en 2009

Recent advances of chroman-4-one derivatives: synthetic approaches and bioactivities

artículo científico publicado en 2015

Recent advances of cytotoxic chalconoids targeting tubulin polymerization: Synthesis and biological activity.

artículo científico publicado en 2016

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

artículo científico

Replacement of the methylene of dihydrochalcones with oxygen: synthesis and biological evaluation of 2-phenoxyacetophenones

artículo científico publicado en 2012

Repurposing azole antifungals into antileishmanials: Novel 3-triazolylflavanones with promising in vitro antileishmanial activity against Leishmania major

artículo científico publicado en 2018

Selective hydrogenation of 4-carboxybenzaldehyde over palladium catalysts supported with different structural organization

Selective leishmanicidal effect of 1,3,4-thiadiazole derivatives and possible mechanism of action against Leishmania species

artículo científico publicado en 2008

Stereoselective synthesis and antifungal activity of (Z)-trans-3-azolyl-2-methylchromanone oxime ethers

artículo científico publicado en 2004

Stereoselective synthesis and in vitro antifungal evaluation of (E)- and (Z)-imidazolylchromanone oxime ethers

artículo científico publicado en 2002

Stereospecific deuteration of alpha-furanosyl azomycin nucleosides: a model reaction for tritium radiolabeling

artículo científico publicado en 2008

Straightforward synthesis of thiazoline-incorporated chalconoids from phenacyl halides

artículo científico publicado en 2013

Structural features of new quinolones and relationship to antibacterial activity against Gram-positive bacteria

artículo científico publicado en 2006

Structure-activity relationship study of a series of N-substituted piperazinyl-fluoroquinolones as anti-Helicobacter pylori agents

artículo científico publicado en 2008

Synthesis and Evaluation of 2(3H)-Thiazole Thiones as Tyrosinase Inhibitors

article published in 2012

Synthesis and anti-Helicobacter pylori activity of 5-(nitroaryl)-1,3,4-thiadiazoles with certain sulfur containing alkyl side chain

artículo científico publicado en 2008

Synthesis and anti-cancer activity evaluation of new dimethoxylated chalcone and flavanone analogs

scientific article published on 08 September 2014

Synthesis and anti-cholinesterase activity of new 7-hydroxycoumarin derivatives

artículo científico publicado en 2014

Synthesis and anti-leishmanial activity of 5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-amines containing N-[(1-benzyl-1H-1,2,3-triazol-4-yl)methyl] moieties

artículo científico publicado en 2012

Synthesis and antibacterial activity of N-(5-benzylthio-1,3,4-thiadiazol-2-yl) and N-(5-benzylsulfonyl-1,3,4-thiadiazol-2-yl)piperazinyl quinolone derivatives

artículo científico publicado en 2005

Synthesis and antibacterial activity of N-[2-(5-bromothiophen-2-yl)-2-oxoethyl] and N-[(2-5-bromothiophen-2-yl)-2-oximinoethyl] derivatives of piperazinyl quinolones.

artículo científico publicado en 2005

Synthesis and antibacterial activity of N-[2-[5-(methylthio)thiophen-2-yl]-2-oxoethyl] and N-[2-[5-(methylthio)thiophen-2-yl]-2-(oxyimino)ethyl]piperazinylquinolone derivatives.

artículo científico publicado en 2006

Synthesis and antibacterial activity of N-[5-(chlorobenzylthio)-1,3,4-thiadiazol-2-yl] piperazinyl quinolone derivatives

artículo científico publicado en 2007

Synthesis and antibacterial activity of levofloxacin derivatives with certain bulky residues on piperazine ring

artículo científico publicado en 2007

Synthesis and antibacterial activity of new 7-piperazinyl-quinolones containing a functionalized 2-(furan-3-yl)ethyl moiety

artículo científico publicado en 2007

Synthesis and antibacterial activity of new N-[2-(thiophen-3-yl)ethyl] piperazinyl quinolones

artículo científico publicado en 2007

Synthesis and antibacterial activity of new fluoroquinolones containing a substituted N-(phenethyl)piperazine moiety

artículo científico publicado en 2006

Synthesis and antibacterial activity of nitroaryl thiadiazole-gatifloxacin hybrids.

artículo científico publicado en 2008

Synthesis and antibacterial activity of nitroaryl thiadiazole-levofloxacin hybrids

artículo científico publicado en 2006

Synthesis and antibacterial activity of novel levofloxacin derivatives containing a substituted thienylethyl moiety

artículo científico publicado en 2012

Synthesis and antibacterial activity of quinolone-based compounds containing a coumarin moiety

artículo científico publicado en 2008

Synthesis and anticancer activity of N-substituted 2-arylquinazolinones bearing trans-stilbene scaffold

artículo científico publicado en 2015

Synthesis and anticholinergic activity of 4-hydroxycoumarin derivatives containing substituted benzyl-1,2,3-triazole moiety.

artículo científico publicado en 2015

Synthesis and anticholinesterase activity of coumarin-3-carboxamides bearing tryptamine moiety.

artículo científico publicado en 2016

Synthesis and antifungal activity of 1-[(2-benzyloxy)phenyl]-2-(azol-1-yl)ethanone derivatives: exploring the scaffold flexibility

artículo científico publicado en 2011

Synthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles

artículo científico publicado en 2010

Synthesis and antileishmanial activity of novel 5-(5-nitrofuran-2-y1)-1,3,4-thiadiazoles with piperazinyl-linked benzamidine substituents

artículo científico publicado en 2011

Synthesis and antioxidant properties of substituted 3-benzylidene-7-alkoxychroman-4-ones

artículo científico publicado en 2007

Synthesis and biological assessment of ciprofloxacin-derived 1,3,4-thiadiazoles as anticancer agents

artículo científico publicado en 2020

Synthesis and biological evaluation of 2-phenylthiazole-4-carboxamide derivatives as anticancer agents

artículo científico publicado en 2010

Synthesis and biological evaluation of 3-(trimethoxyphenyl)-2(3H)-thiazole thiones as combretastatin analogs.

artículo científico publicado en 2013

Synthesis and biological evaluation of 4-amino-5-cinnamoylthiazoles as chalcone-like anticancer agents.

artículo científico publicado en 2018

Synthesis and biological evaluation of 5-benzylidenerhodanine-3-acetic acid derivatives as AChE and 15-LOX inhibitors

artículo científico publicado en 2015

Synthesis and biological evaluation of fluconazole analogs with triazole-modified scaffold as potent antifungal agents

artículo científico publicado en 2015

Synthesis and biological evaluation of new N-benzylpyridinium-based benzoheterocycles as potential anti-Alzheimer's agents

scientific article published on 13 November 2018

Synthesis and biological evaluation of new coumarins bearing 2,4-diaminothiazole-5-carbonyl moiety

scientific article published on 07 June 2018

Synthesis and biological evaluation of novel imidazopyrimidin-3-amines as anticancer agents

artículo científico publicado en 2016

Synthesis and biological evaluation of quinazolinone-based hydrazones with potential use in Alzheimer's disease

artículo científico publicado en 2017

Synthesis and cytotoxic activity of novel poly-substituted imidazo[2,1-c][1,2,4]triazin-6-amines

artículo científico publicado en 2015

Synthesis and cytotoxic properties of novel (E)-3-benzylidene-7-methoxychroman-4-one derivatives.

artículo científico publicado en 2013

Synthesis and evaluation of 4-substituted coumarins as novel acetylcholinesterase inhibitors

scientific article published on 18 March 2013

Synthesis and free radical scavenging activity of coumarin derivatives containing a 2-methylbenzothiazoline motif

scientific article published on 25 August 2011

Synthesis and hypoxia selective radiosensitization potential of beta-2-FAZA and beta-3-FAZL: fluorinated azomycin beta-nucleosides

artículo científico publicado en 2009

Synthesis and in vitro anti-Helicobacter pylori activity of N-[5-(5-nitro-2-heteroaryl)-1,3,4-thiadiazol-2-yl]thiomorpholines and related compounds

artículo científico publicado en 2007

Synthesis and in vitro anti-Toxoplasma gondii activity of a new series of aryloxyacetophenone thiosemicarbazones

artículo científico publicado en 2019

Synthesis and in vitro anti-leishmanial activity of 1-[5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-yl]- and 1-[5-(5-nitrothiophen-2-yl)-1,3,4-thiadiazol-2-yl]-4-aroylpiperazines

artículo científico publicado en 2008

Synthesis and in vitro cytotoxic activity of novel chalcone-like agents

artículo científico publicado en 2013

Synthesis and in vitro leishmanicidal activity of 2-(1-methyl-5-nitro-1H-imidazol-2-yl)-5-substituted-1,3,4-thiadiazole derivatives

artículo científico publicado en 2005

Synthesis and in-vitro antibacterial activity of 5-substituted 1-methyl-4-nitro-1H-imidazoles.

artículo científico publicado en 2008

Synthesis and in-vitro cytotoxicity of poly-functionalized 4-(2-arylthiazol-4-yl)-4H-chromenes.

artículo científico publicado en 2010

Synthesis and structure-activity relationship study of benzofuran-based chalconoids bearing benzylpyridinium moiety as potent acetylcholinesterase inhibitors.

artículo científico publicado en 2015

Synthesis and structure-activity relationship study of tacrine-based pyrano[2,3-c]pyrazoles targeting AChE/BuChE and 15-LOX.

artículo científico publicado en 2016

Synthesis of 4‐Hydroxycoumarin‐Based Triazoles/Oxadiazoles as Novel Anticancer Agents

artículo científico publicado en 2022

Synthesis, biological evaluation and docking study of 3-aroyl-1-(4-sulfamoylphenyl)thiourea derivatives as 15-lipoxygenase inhibitors

artículo científico publicado en 2014

Synthesis, computational study and cytotoxicity of 4-hydroxycoumarin-derived imines/enamines

artículo científico publicado en 2020

Synthesis, in vitro antifungal activity and in silico study of 3-(1,2,4-triazol-1-yl)flavanones.

artículo científico publicado en 2013

Synthesis, in vitro antifungal evaluation and in silico study of 3-azolyl-4-chromanone phenylhydrazones.

artículo científico publicado en 2012

Synthesis, in vitro cytotoxicity and apoptosis inducing study of 2-aryl-3-nitro-2H-chromene derivatives as potent anti-breast cancer agents

artículo científico publicado en 2014

The effects of plant cover on population of pear psylla (Cacopsylla pyricola) and its predators

artículo científico publicado en 2017

The importance of triazole scaffold in the development of anticonvulsant agents

artículo científico publicado en 2016

Tropolone alkaloids from Colchicum kurdicum (Bornm.) Stef. (Colchicaceae) as the potent novel antileishmanial compounds; purification, structure elucidation, antileishmanial activities and molecular docking studies

artículo científico publicado en 2020

Ultrastructural Investigation of Leishmania major Promastigotes Treated with A New Potent Antileishmanial Azole Using Scanning Electron and Atomic Force Microscopes

artículo científico publicado en 2018

Utility of aptamers for antileishmanial drug targets: A potential hypothesis

artículo científico publicado en 2017

β-Ionone and its analogs as promising anticancer agents

artículo científico publicado en 2016

Dominio Público Uruguay está sostenido por:

Acerca de Dominio Público Uruguay

Ayuda