Lista de obras - Serena Massari - Dominio Público Uruguay

1,4-Benzothiazine ATP-sensitive potassium channel openers: modifications at the C-2 and C-6 positions

artículo científico publicado en 2013

2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction

artículo científico publicado en 2018

2-Phenylquinolones as inhibitors of the HIV-1 Tat-TAR interaction

artículo científico publicado en 2009

6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis

scientific article published on 10 September 2012

6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.

artículo científico publicado en 2010

A 1,8-naphthyridone derivative targets the HIV-1 Tat-mediated transcription and potently inhibits the HIV-1 replication

artículo científico publicado en 2010

A Broad Anti-influenza Hybrid Small Molecule That Potently Disrupts the Interaction of Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits

artículo científico publicado en 2015

Blocking HIV-1 replication by targeting the Tat-hijacked transcriptional machinery

artículo científico publicado en 2013

Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions

scientific article published on 06 March 2019

C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors

artículo científico publicado en 2020

Computer-aided design, synthesis and validation of 2-phenylquinazolinone fragments as CDK9 inhibitors with anti-HIV-1 Tat-mediated transcription activity.

artículo científico publicado en 2013

Design, synthesis, and evaluation of WC5 analogues as inhibitors of human cytomegalovirus Immediate-Early 2 protein, a promising target for anti-HCMV treatment

artículo científico publicado en 2013

Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a]pyrimidine derivatives

artículo científico publicado en 2017

Ethyl 1,8-naphthyridone-3-carboxylates downregulate human papillomavirus-16 E6 and E7 oncogene expression.

artículo científico publicado en 2014

Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands.

artículo científico publicado en 2014

From 6-aminoquinolone antibacterials to 6-amino-7-thiopyranopyridinylquinolone ethyl esters as inhibitors of Staphylococcus aureus multidrug efflux pumps

artículo científico publicado en 2010

From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors

article

From small to powerful: the fragments universe and its "chem-appeal".

artículo científico publicado en 2013

Inhibition of Influenza Virus Polymerase by Interfering with Its Protein-Protein Interactions

scientific article published on 12 October 2020

Inhibition of subgenomic hepatitis C virus RNA replication by acridone derivatives: identification of an NS3 helicase inhibitor

artículo científico publicado en 2009

Modulation of HIV-1-induced activation of plasmacytoid dendritic cells by 6-desfluoroquinolones

artículo científico publicado en 2013

Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors

artículo científico publicado en 2017

Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase

artículo científico publicado en 2011

Re-evolution of the 2-phenylquinolines: ligand-based design, synthesis, and biological evaluation of a potent new class of Staphylococcus aureus NorA efflux pump inhibitors to combat antimicrobial resistance

artículo científico publicado en 2013

Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues

artículo científico publicado en 2017

Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors

artículo científico publicado en 2020

Structural investigation of cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly

artículo científico publicado en 2013

Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity

artículo científico publicado en 2011

Structure-activity relationship study on anti-HIV 6-desfluoroquinolones

artículo científico publicado en 2008

Studies of anti-HIV transcription inhibitor quinolones: identification of potent N1-vinyl derivatives

artículo científico publicado en 2010

Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position

Studies on anti-HIV quinolones: New insights on the C-6 position

article

Synthesis and chromatographic enantioresolution of anti-HIV quinolone derivatives

article

The 6-Aminoquinolone WC5 inhibits different functions of the immediate-early 2 (IE2) protein of human cytomegalovirus that are essential for viral replication

artículo científico publicado en 2014

The 6-aminoquinolone WC5 inhibits human cytomegalovirus replication at an early stage by interfering with the transactivating activity of viral immediate-early 2 protein

artículo científico publicado en 2010

The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors.

artículo científico publicado en 2015

Lista de obras de Serena Massari

1,4-Benzothiazine ATP-sensitive potassium channel openers: modifications at the C-2 and C-6 positions

2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction

2-Phenylquinolones as inhibitors of the HIV-1 Tat-TAR interaction

6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis

6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.

A 1,8-naphthyridone derivative targets the HIV-1 Tat-mediated transcription and potently inhibits the HIV-1 replication

A Broad Anti-influenza Hybrid Small Molecule That Potently Disrupts the Interaction of Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits

Blocking HIV-1 replication by targeting the Tat-hijacked transcriptional machinery

Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions

C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors

Computer-aided design, synthesis and validation of 2-phenylquinazolinone fragments as CDK9 inhibitors with anti-HIV-1 Tat-mediated transcription activity.

Design, synthesis, and evaluation of WC5 analogues as inhibitors of human cytomegalovirus Immediate-Early 2 protein, a promising target for anti-HCMV treatment

Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a]pyrimidine derivatives

Ethyl 1,8-naphthyridone-3-carboxylates downregulate human papillomavirus-16 E6 and E7 oncogene expression.

Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands.

From 6-aminoquinolone antibacterials to 6-amino-7-thiopyranopyridinylquinolone ethyl esters as inhibitors of Staphylococcus aureus multidrug efflux pumps

From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors

From small to powerful: the fragments universe and its "chem-appeal".

Inhibition of Influenza Virus Polymerase by Interfering with Its Protein-Protein Interactions

Inhibition of subgenomic hepatitis C virus RNA replication by acridone derivatives: identification of an NS3 helicase inhibitor

Modulation of HIV-1-induced activation of plasmacytoid dendritic cells by 6-desfluoroquinolones

Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors

Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase

Re-evolution of the 2-phenylquinolines: ligand-based design, synthesis, and biological evaluation of a potent new class of Staphylococcus aureus NorA efflux pump inhibitors to combat antimicrobial resistance

Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues

Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors

Structural investigation of cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly

Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity

Structure-activity relationship study on anti-HIV 6-desfluoroquinolones

Studies of anti-HIV transcription inhibitor quinolones: identification of potent N1-vinyl derivatives

Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position

Studies on anti-HIV quinolones: New insights on the C-6 position

Synthesis and chromatographic enantioresolution of anti-HIV quinolone derivatives

The 6-Aminoquinolone WC5 inhibits different functions of the immediate-early 2 (IE2) protein of human cytomegalovirus that are essential for viral replication

The 6-aminoquinolone WC5 inhibits human cytomegalovirus replication at an early stage by interfering with the transactivating activity of viral immediate-early 2 protein

The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors.