Lista de obras - Thomas L. Mindt - Dominio Público Uruguay

"Click-to-chelate": design and incorporation of triazole-containing metal-chelating systems into biomolecules of diagnostic and therapeutic interest

artículo científico publicado en 2008

"Click-to-chelate": in vitro and in vivo comparison of a 99mTc(CO)3-labeled N(tau)-histidine folate derivative with its isostructural, clicked 1,2,3-triazole analogue

artículo científico publicado en 2008

1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting.

artículo científico publicado en 2015

1,2,3-Triazoles as amide bond mimics: triazole scan yields protease-resistant peptidomimetics for tumor targeting

artículo científico publicado en 2013

1,2,3-Triazoles as amide-bond surrogates in peptidomimetics.

artículo científico publicado en 2013

A "click chemistry" approach to the efficient synthesis of multiple imaging probes derived from a single precursor

artículo científico publicado en 2009

A bombesin-shepherdin radioconjugate designed for combined extra- and intracellular targeting

artículo científico publicado en 2014

A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate

artículo científico publicado en 2009

A solid phase-assisted approach for the facile synthesis of a highly water-soluble zirconium-89 chelator for radiopharmaceutical development.

artículo científico publicado en 2017

An octadentate bifunctional chelating agent for the development of stable zirconium-89 based molecular imaging probes

artículo científico publicado en 2014

Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticals

artículo científico publicado en 2013

Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno-PET

artículo científico publicado en 2016

Convergent Synthesis of 2H-Chromenes - a Formal [3+3] Cycloaddition by a One-pot, Three-Step Cascade.

artículo científico publicado en 2011

Cu(I)-catalyzed intramolecular cyclization of alkynoic acids in aqueous media: a "click side reaction".

artículo científico publicado en 2007

Development of 68Ga- and 89Zr-Labeled Exendin-4 as Potential Radiotracers for the Imaging of Insulinomas by PET

article

Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides

artículo científico publicado en 2012

EANM guideline for the preparation of an Investigational Medicinal Product Dossier (IMPD)

artículo científico publicado en 2014

Effect of amino acid infusion on potassium serum levels in neuroendocrine tumour patients treated with targeted radiopeptide therapy

artículo científico publicado en 2011

Electrocyclic Ring Closure of the Enols of Vinyl Quinones. A2H-Chromene Synthesis

artículo científico publicado en 2001

Evaluation of a novel radiofolate in tumour-bearing mice: promising prospects for folate-based radionuclide therapy

artículo científico publicado en 2009

Expression of different neurokinin-1 receptor (NK1R) isoforms in glioblastoma multiforme: potential implications for targeted therapy

artículo científico publicado en 2014

Fluorescent gallium and indium bis(thiosemicarbazonates) and their radiolabelled analogues: synthesis, structures and cellular confocal fluorescence imaging investigations.

artículo científico publicado en 2011

Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative

artículo científico publicado en 2008

Glycated 99m Tc-Tricarbonyl-Labeled Peptide Conjugates for Tumor Targeting by "Click-to-Chelate".

artículo científico publicado en 2016

Guidance on current good radiopharmacy practice for the small-scale preparation of radiopharmaceuticals using automated modules: a European perspective

artículo científico publicado en 2014

Heterocycle Annulation of Enolizable Vinyl Quinone Imides. Dihydroquinolines and Quinolines from Thermal 6π-Electrocyclizations and Indoles from Photochemical Cyclizations

artículo científico publicado en 2002

Imaging of activated macrophages in experimental osteoarthritis using folate-targeted animal single-photon-emission computed tomography/computed tomography

artículo científico publicado en 2011

Manganese in PET imaging: Opportunities and challenges

artículo científico publicado en 2019

Metal chelating systems synthesized using the copper(I) catalyzed azide-alkyne cycloaddition.

artículo científico publicado en 2009

Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates

artículo científico publicado en 2017

Modification of different IgG1 antibodies via glutamine and lysine using bacterial and human tissue transglutaminase

artículo científico publicado en 2007

Molecular assembly of multifunctional ⁹⁹(m)Tc radiopharmaceuticals using "clickable" amino acid derivatives.

artículo científico publicado en 2010

Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions.

artículo científico publicado en 2016

Position paper on requirements for toxicological studies in the specific case of radiopharmaceuticals

article

Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy

artículo científico publicado en 2015

Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting.

artículo científico publicado en 2013

Radiolabelling of the octadentate chelators DFO* and oxoDFO* with zirconium-89 and gallium-68

scientific article published on 13 July 2020

Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates

artículo científico publicado en 2015

Synthesis and Preclinical Evaluation of Radiolabeled [103Ru]BOLD-100

artículo científico publicado en 2023

TESOTf-induced rearrangement of quinols. Efficient construction of the fully functionalized carbon skeleton of the griseusins by a divergent-reconvergent approach

artículo científico publicado en 2006

Toward the Optimization of Bombesin-Based Radiotracers for Tumor Targeting.

artículo científico publicado en 2016

“Click to Chelate”: Synthesis and Installation of Metal Chelates into Biomolecules in a Single Step

artículo científico publicado en 2006

Lista de obras de Thomas L. Mindt

"Click-to-chelate": design and incorporation of triazole-containing metal-chelating systems into biomolecules of diagnostic and therapeutic interest

"Click-to-chelate": in vitro and in vivo comparison of a 99mTc(CO)3-labeled N(tau)-histidine folate derivative with its isostructural, clicked 1,2,3-triazole analogue

1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting.

1,2,3-Triazoles as amide bond mimics: triazole scan yields protease-resistant peptidomimetics for tumor targeting

1,2,3-Triazoles as amide-bond surrogates in peptidomimetics.

A "click chemistry" approach to the efficient synthesis of multiple imaging probes derived from a single precursor

A bombesin-shepherdin radioconjugate designed for combined extra- and intracellular targeting

A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate

A solid phase-assisted approach for the facile synthesis of a highly water-soluble zirconium-89 chelator for radiopharmaceutical development.

An octadentate bifunctional chelating agent for the development of stable zirconium-89 based molecular imaging probes

Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticals

Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno-PET

Convergent Synthesis of 2H-Chromenes - a Formal [3+3] Cycloaddition by a One-pot, Three-Step Cascade.

Cu(I)-catalyzed intramolecular cyclization of alkynoic acids in aqueous media: a "click side reaction".

Development of 68Ga- and 89Zr-Labeled Exendin-4 as Potential Radiotracers for the Imaging of Insulinomas by PET

Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides

EANM guideline for the preparation of an Investigational Medicinal Product Dossier (IMPD)

Effect of amino acid infusion on potassium serum levels in neuroendocrine tumour patients treated with targeted radiopeptide therapy

Electrocyclic Ring Closure of the Enols of Vinyl Quinones. A2H-Chromene Synthesis

Evaluation of a novel radiofolate in tumour-bearing mice: promising prospects for folate-based radionuclide therapy

Expression of different neurokinin-1 receptor (NK1R) isoforms in glioblastoma multiforme: potential implications for targeted therapy

Fluorescent gallium and indium bis(thiosemicarbazonates) and their radiolabelled analogues: synthesis, structures and cellular confocal fluorescence imaging investigations.

Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative

Glycated 99m Tc-Tricarbonyl-Labeled Peptide Conjugates for Tumor Targeting by "Click-to-Chelate".

Guidance on current good radiopharmacy practice for the small-scale preparation of radiopharmaceuticals using automated modules: a European perspective

Heterocycle Annulation of Enolizable Vinyl Quinone Imides. Dihydroquinolines and Quinolines from Thermal 6π-Electrocyclizations and Indoles from Photochemical Cyclizations

Imaging of activated macrophages in experimental osteoarthritis using folate-targeted animal single-photon-emission computed tomography/computed tomography

Manganese in PET imaging: Opportunities and challenges

Metal chelating systems synthesized using the copper(I) catalyzed azide-alkyne cycloaddition.

Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates

Modification of different IgG1 antibodies via glutamine and lysine using bacterial and human tissue transglutaminase

Molecular assembly of multifunctional ⁹⁹(m)Tc radiopharmaceuticals using "clickable" amino acid derivatives.

Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions.

Position paper on requirements for toxicological studies in the specific case of radiopharmaceuticals

Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy

Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting.

Radiolabelling of the octadentate chelators DFO* and oxoDFO* with zirconium-89 and gallium-68

Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates

Synthesis and Preclinical Evaluation of Radiolabeled [103Ru]BOLD-100

TESOTf-induced rearrangement of quinols. Efficient construction of the fully functionalized carbon skeleton of the griseusins by a divergent-reconvergent approach

Toward the Optimization of Bombesin-Based Radiotracers for Tumor Targeting.

“Click to Chelate”: Synthesis and Installation of Metal Chelates into Biomolecules in a Single Step