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Lista de obras de Mark Cushman

A structure-based model of the reaction catalyzed by lumazine synthase from Aquifex aeolicus

artículo científico publicado en 2003

Application of Sequential Palladium Catalysis for the Discovery of Janus Kinase Inhibitors in the Benzo[ c]pyrrolo[2,3- h][1,6]naphthyridin-5-one (BPN) Series

artículo científico publicado en 2018

Crystallographic Study of a Novel Subnanomolar Inhibitor Provides Insight on the Binding Interactions of Alkenyldiarylmethanes with Human Immunodeficiency Virus-1 Reverse Transcriptase

artículo científico publicado en 2009

Design and Synthesis of Chlorinated and Fluorinated 7-Azaindenoisoquinolines as Potent Cytotoxic Anticancer Agents That Inhibit Topoisomerase I.

artículo científico publicado en 2017

Design, Synthesis, and Biological Evaluation of Potent Quinoline and Pyrroloquinoline Ammosamide Analogues as Inhibitors of Quinone Reductase 2

artículo científico publicado en 2012

Design, synthesis, and biological evaluation of antiviral agents targeting flavivirus envelope proteins

artículo científico publicado en 2008

Design, synthesis, and biological evaluation of thiazoles targeting flavivirus envelope proteins

artículo científico publicado en 2011

Indenoisoquinoline Topoisomerase Inhibitors Strongly Bind and Stabilize the MYC Promoter G-Quadruplex and Downregulate MYC

scientific article published on 08 July 2019

Lumazine synthase from Candida albicans as an anti-fungal target enzyme: structural and biochemical basis for drug design

artículo científico publicado en 2007

MAIT Recognition of a Stimulatory Bacterial Antigen Bound to MR1

artículo científico publicado en 2013

Riboflavin synthase of Schizosaccharomyces pombe. Protein dynamics revealed by 19F NMR protein perturbation experiments

artículo científico publicado en 2003

Structural study and thermodynamic characterization of inhibitor binding to lumazine synthase fromBacillus anthracis

artículo científico publicado en 2010

Synthesis and Biological Evaluation of the First Triple Inhibitors of Human Topoisomerase 1, Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), and Tyrosyl-DNA Phosphodiesterase 2 (Tdp2).

artículo científico publicado en 2017

Synthesis and cancer chemopreventive activity of zapotin, a natural product from Casimiroa edulis

artículo científico publicado en 2007

Synthesis of Casimiroin and Optimization of Its Quinone Reductase 2 and Aromatase Inhibitory Activities

artículo científico publicado en 2009

The structural basis of riboflavin binding to Schizosaccharomyces pombe 6,7-dimethyl-8-ribityllumazine synthase

artículo científico publicado en 2002