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Lista de obras de Claudia Temperini

A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases

artículo científico publicado en 2009

Carbonic anhydrase activators: kinetic and X-ray crystallographic study for the interaction of D- and L-tryptophan with the mammalian isoforms I-XIV

artículo científico publicado en 2008

Carbonic anhydrase inhibitors. Comparison of chlorthalidone and indapamide X-ray crystal structures in adducts with isozyme II: when three water molecules and the keto-enol tautomerism make the difference

artículo científico publicado en 2009

Carbonic anhydrase inhibitors. Interaction of 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide with 12 mammalian isoforms: kinetic and X-ray crystallographic studies

artículo científico publicado en 2008

Carbonic anhydrase inhibitors. Interaction of 2-N,N-dimethylamino-1,3,4-thiadiazole-5-methanesulfonamide with 12 mammalian isoforms: kinetic and X-ray crystallographic studies

artículo científico publicado en 2008

Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct

artículo científico publicado en 2008

Carbonic anhydrase inhibitors. Interaction of the antiepileptic drug sulthiame with twelve mammalian isoforms: kinetic and X-ray crystallographic studies

artículo científico publicado en 2007

Carbonic anhydrase inhibitors. X-ray crystal studies of the carbonic anhydrase II-trithiocarbonate adduct--an inhibitor mimicking the sulfonamide and urea binding to the enzyme

artículo científico publicado en 2010

Carbonic anhydrase inhibitors: the X-ray crystal structure of the adduct of N-hydroxysulfamide with isozyme II explains why this new zinc binding function is effective in the design of potent inhibitors

artículo científico publicado en 2007

Deciphering the mechanism of carbonic anhydrase inhibition with coumarins and thiocoumarins

artículo científico publicado en 2010

Dissecting the inhibition mechanism of cytosolic versus transmembrane carbonic anhydrases by ESR

artículo científico publicado en 2009

ESI mass spectrometry and X-ray diffraction studies of adducts between anticancer platinum drugs and hen egg white lysozyme

artículo científico publicado en 2007

Nitric oxide-donating carbonic anhydrase inhibitors for the treatment of open-angle glaucoma

artículo científico publicado en 2009

Non-zinc mediated inhibition of carbonic anhydrases: coumarins are a new class of suicide inhibitors

artículo científico publicado en 2009

Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I

artículo científico publicado en 2007

Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule

artículo científico publicado en 2010

Synthesis and crystallographic analysis of new sulfonamides incorporating NO-donating moieties with potent antiglaucoma action

artículo científico publicado en 2011

The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors

artículo científico publicado en 2010

The crystal structure of the complex between a disaccharide anthracycline and the DNA hexamer d(CGATCG) reveals two different binding sites involving two DNA duplexes

artículo científico publicado en 2003

The x-ray structure of the adduct between NAMI-A and carbonic anhydrase provides insights into the reactivity of this metallodrug with proteins

artículo científico publicado en 2010

Carbonic anhydrase inhibitors. Interaction of the antitumor sulfamate EMD 486019 with twelve mammalian carbonic anhydrase isoforms: Kinetic and X-ray crystallographic studies

artículo científico publicado el 1 de agosto de 2008