Lista de obras -

A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism

artículo científico publicado en 2017

A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.

artículo científico publicado en 2014

Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo).

artículo científico publicado en 2016

Correction for "Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines".

artículo científico publicado en 2016

Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues

artículo científico publicado en 2017

In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations.

artículo científico publicado en 2016

Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist

scientific article published on 02 August 2016

Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues.

artículo científico publicado en 2014

Pharmacological characterization of tachykinin tetrabranched derivatives

artículo científico publicado en 2014

Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt1]N/OFQ(1-13).

artículo científico publicado en 2016

Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic

artículo científico publicado en 2016

Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity.

artículo científico publicado en 2015

Structure activity studies of nociceptin/orphanin FQ(1-13)-NH2 derivatives modified in position 5.

artículo científico publicado en 2015

Structure- and conformation-activity studies of nociceptin/orphanin FQ receptor dimeric ligands

artículo científico publicado en 2017

Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids

artículo científico publicado en 2017

Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration

artículo científico publicado en 2015

Synthesis of mixed opioid affinity cyclic endomorphin-2 analogues with fluorinated phenylalanines

artículo científico publicado en 2015

Synthesis, biological evaluation and structural analysis of novel peripherally active morphiceptin analogs

artículo científico publicado en 2016

Lista de obras de

A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism

A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.

Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo).

Correction for "Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines".

Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues

In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations.

Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist

Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues.

Pharmacological characterization of tachykinin tetrabranched derivatives

Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt1]N/OFQ(1-13).

Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic

Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity.

Structure activity studies of nociceptin/orphanin FQ(1-13)-NH2 derivatives modified in position 5.

Structure- and conformation-activity studies of nociceptin/orphanin FQ receptor dimeric ligands

Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids

Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration

Synthesis of mixed opioid affinity cyclic endomorphin-2 analogues with fluorinated phenylalanines

Synthesis, biological evaluation and structural analysis of novel peripherally active morphiceptin analogs

Synthesis, enantiomeric separation and docking studies of spiropiperidine analogues as ligands of the nociceptin/orphanin FQ receptor