Lista de obras -

A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6

artículo científico publicado en 2021

A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases

artículo científico publicado en 2015

A potent, selective and cell-active allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3)

artículo científico publicado en 2015

Allosteric inhibitors of plasma membrane Ca2+pumps: Invention and applications of caloxins ⬇️

artículo científico publicado el 26 de marzo de 2011

Aortic smooth muscle and endothelial plasma membrane Ca2+ pump isoforms are inhibited differently by the extracellular inhibitor caloxin 1b1.

artículo científico publicado en 2006

Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors

artículo científico publicado en 2017

Author Correction: Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response

scientific article published on 26 May 2020

Ca2+-mediated ascorbate release from coronary artery endothelial cells

artículo científico publicado en 2006

Ca2+-pumps and Na2+-Ca2+-exchangers in coronary artery endothelium versus smooth muscle

artículo científico publicado en 2007

Caloxin 1b3: A novel plasma membrane Ca2+-pump isoform 1 selective inhibitor that increases cytosolic Ca2+ in endothelial cells ⬇️

artículo científico publicado el 18 de noviembre de 2010

Caloxins: a novel class of selective plasma membrane Ca2+ pump inhibitors obtained using biotechnology

artículo científico publicado en 2007

Characterization of inv(3) cell line OCI-AML-20 with stroma dependent CD34 expression

artículo científico publicado en 2018

Correction to Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening

scientific article published on 03 August 2016

Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2

artículo científico publicado en 2016

Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).

artículo científico publicado en 2017

Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2

artículo científico publicado en 2021

Discovery of a Dual PRMT5-PRMT7 Inhibitor

artículo científico publicado en 2015

Discovery of a First-in-Class Protein Arginine Methyltransferase 6 (PRMT6) Covalent Inhibitor

scientific article published on 05 May 2020

Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor

artículo científico publicado en 2016

Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening

artículo científico publicado en 2016

Discovery of a Potent, Selective, and Cell-Active Dual Inhibitor of Protein Arginine Methyltransferase 4 and Protein Arginine Methyltransferase 6.

artículo científico publicado en 2016

Discovery of a chemical probe for PRDM9

scientific article published on 17 December 2019

Erratum: The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex

artículo científico publicado en 2017

Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3

scientific article published on 08 July 2019

Functional effects of caloxin 1c2, a novel engineered selective inhibitor of plasma membrane Ca(2+)-pump isoform 4, on coronary artery.

artículo científico publicado en 2008

HAP40 orchestrates huntingtin structure for differential interaction with polyglutamine expanded exon 1

preprint

Huntingtin structure is orchestrated by HAP40 and shows a polyglutamine expansion-specific interaction with exon 1

artículo científico publicado en 2021

LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity

artículo científico publicado en 2018

PRMT5 regulates ATF4 transcript splicing and oxidative stress response

artículo científico publicado en 2022

PRMT5 regulates ATF4 transcript splicing and oxidative stress response

preprint

Phage display: concept, innovations, applications and future

artículo científico publicado en 2010

Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response

artículo científico publicado en 2020

Photoswitchable Catalysis by a Small Swinging Molecule Confined on the Surface of a Colloidal Particle

Sialidase down-regulation reduces non-HDL cholesterol, inhibits leukocyte transmigration, and attenuates atherosclerosis in ApoE knockout mice

artículo científico publicado en 2018

TP-064, a potent and selective small molecule inhibitor of PRMT4 for multiple myeloma.

artículo científico publicado en 2018

The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex

artículo científico publicado en 2017

Therapeutic Targeting of RNA Splicing Catalysis through Inhibition of Protein Arginine Methylation

artículo científico publicado en 2019

Lista de obras de

A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6

A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases

A potent, selective and cell-active allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3)

Allosteric inhibitors of plasma membrane Ca2+pumps: Invention and applications of caloxins ⬇️

Aortic smooth muscle and endothelial plasma membrane Ca2+ pump isoforms are inhibited differently by the extracellular inhibitor caloxin 1b1.

Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors

Author Correction: Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response

Ca2+-mediated ascorbate release from coronary artery endothelial cells

Ca2+-pumps and Na2+-Ca2+-exchangers in coronary artery endothelium versus smooth muscle

Caloxin 1b3: A novel plasma membrane Ca2+-pump isoform 1 selective inhibitor that increases cytosolic Ca2+ in endothelial cells ⬇️

Caloxins: a novel class of selective plasma membrane Ca2+ pump inhibitors obtained using biotechnology

Characterization of inv(3) cell line OCI-AML-20 with stroma dependent CD34 expression

Correction to Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening

Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2

Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).

Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2

Discovery of a Dual PRMT5-PRMT7 Inhibitor

Discovery of a First-in-Class Protein Arginine Methyltransferase 6 (PRMT6) Covalent Inhibitor

Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor

Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening

Discovery of a Potent, Selective, and Cell-Active Dual Inhibitor of Protein Arginine Methyltransferase 4 and Protein Arginine Methyltransferase 6.

Discovery of a chemical probe for PRDM9

Erratum: The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex

Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3

Functional effects of caloxin 1c2, a novel engineered selective inhibitor of plasma membrane Ca(2+)-pump isoform 4, on coronary artery.

HAP40 orchestrates huntingtin structure for differential interaction with polyglutamine expanded exon 1

Huntingtin structure is orchestrated by HAP40 and shows a polyglutamine expansion-specific interaction with exon 1

LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity

PRMT5 regulates ATF4 transcript splicing and oxidative stress response

PRMT5 regulates ATF4 transcript splicing and oxidative stress response

Phage display: concept, innovations, applications and future

Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response

Photoswitchable Catalysis by a Small Swinging Molecule Confined on the Surface of a Colloidal Particle

Sialidase down-regulation reduces non-HDL cholesterol, inhibits leukocyte transmigration, and attenuates atherosclerosis in ApoE knockout mice

TP-064, a potent and selective small molecule inhibitor of PRMT4 for multiple myeloma.

The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex

Therapeutic Targeting of RNA Splicing Catalysis through Inhibition of Protein Arginine Methylation