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3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-alkylamides as a new class of synthetic histone deacetylase inhibitors. 1. Design, synthesis, biological evaluation, and binding mode studies performed through three different docking procedures

artículo científico publicado en 2003

3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamides as a new class of synthetic histone deacetylase inhibitors. 2. Effect of pyrrole-C2 and/or -C4 substitutions on biological activity

artículo científico publicado en 2004

3-(4-Aroyl-1-methyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides as a new class of synthetic histone deacetylase inhibitors. 3. Discovery of novel lead compounds through structure-based drug design and docking studies

artículo científico publicado en 2004

Antimalarial and antileishmanial activities of aroyl-pyrrolyl-hydroxyamides, a new class of histone deacetylase inhibitors

artículo científico publicado en 2004

GPR55: Current knowledge and future perspectives of a purported "Type-3" cannabinoid receptor

artículo científico publicado en 2010

Histone deacetylation in epigenetics: an attractive target for anticancer therapy

artículo científico publicado en 2005

In silico scaffold evaluation and solid phase approach to identify new gelatinase inhibitors

artículo científico publicado el 13 de febrero de 2012

Structural bases for substrate and inhibitor recognition by matrix metalloproteinases

scientific article published on January 2008

Thiopyrophosphoantigens: solid-phase synthesis and in vitro characterization of a new class of Vgamma9 Vdelta2 T cells activators

artículo científico publicado en 2009