Lista de obras -

A new method for distinguishing between enantiomers and racemates and assignment of enantiomeric purity by means of solid-state NMR. Examples from oxazaphosphorinanes

artículo científico publicado en 2002

Acyloxymethyl esters of isophosphoramide mustard as new anticancer prodrugs

artículo científico publicado en 2013

Analysis of the urinary excretion of ifosfamide and its N-dechloroethylated metabolites in children using 31P-NMR spectroscopy

artículo científico publicado en 2003

Classical oxazaphosphorines--metabolism and therapeutic properties--new implications

artículo científico publicado en 2013

Discovery and evaluation of efficient selenazoles with high antifungal activity against Candida spp

artículo científico publicado en 2015

Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design, one-pot tricomponent synthesis, and lipophilicity determination

scientific article published on 04 May 2019

Ifosfamide. Metabolic studies, new therapeutic approaches and new analogs

artículo científico publicado en 2006

Isophosphoramide mustard analogues as prodrugs for anticancer gene-directed enzyme-prodrug therapy (GDEPT).

artículo científico publicado en 2002

Oxazaphosphorinane drugs. New analogues, metabolic studies, and therapeutic approaches

artículo científico publicado en 2004

Phosphate prodrugs of isophosphoramide mustard.

artículo científico publicado en 2003

Role of GSTM1, GSTP1, and GSTT1 gene polymorphism in ifosfamide metabolism affecting neurotoxicity and nephrotoxicity in children

artículo científico publicado en 2005

Studies on the side-chain hydroxylation of ifosfamide and its bromo analogue

artículo científico publicado en 2002

Synthesis and Antimicrobial Activities of (4,5,6,7-Tetrahydro-1H-indazol- 2(3H)-yl)thiazole Derivatives

artículo científico publicado en 2014

Synthesis and anticonvulsant activities of novel 2-(cyclopentylmethylene)hydrazinyl-1,3-thiazoles in mouse models of seizures

artículo científico publicado en 2016

Synthesis and antimicrobial activities of novel 6-(1,3-thiazol-4-yl)-1,3-benzoxazol-2(3H)-one derivatives

artículo científico publicado en 2014

Synthesis and antitumour activity of stereoisomers of 4-hydroperoxy derivatives of ifosfamide and its bromo analogue.

artículo científico publicado en 2002

Synthesis and biological evaluation of novel 2-(1H-imidazol-2-ylmethylidene)hydrazinyl- 1,3-thiazoles as potential antimicrobial agents

artículo científico publicado en 2015

Synthesis and in vitro antiproliferative activity of thiazole-based nitrogen mustards: the hydrogen bonding interaction between model systems and nucleobases

artículo científico publicado en 2014

Synthesis of nucleoside alpha-thiotriphosphates via an oxathiaphospholane approach

artículo científico publicado en 2005

Synthesis, Antibacterial Activity, Interaction with Nucleobase and Molecular Docking Studies of 4-Formylbenzoic Acid Based Thiazoles

artículo científico publicado en 2016

Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles.

artículo científico publicado en 2016

Synthesis, antimicrobial evaluation and theoretical prediction of NMR chemical shifts of thiazole and selenazole derivatives with high antifungal activity against Candida spp

Synthesis, in vitro biological screening and molecular docking studies of novel camphor-based thiazoles.

artículo científico publicado en 2014

The Disulfide Analogues of Isophosphoramide Mustard for Anticancer Therapy

artículo científico publicado en 2014

The First Stereocontrolled Solid-Phase Synthesis of Di-, Tri-, and Tetra[adenosine (2‘,5‘) phosphorothioate]s ⬇️

artículo científico publicado el 2 de octubre de 1998

Thiazole-based nitrogen mustards: Design, synthesis, spectroscopic studies, DFT calculation, molecular docking, and antiproliferative activity against selected human cancer cell lines

artículo científico publicado en 2016

Triazene salts: Design, synthesis, ctDNA interaction, lipophilicity determination, DFT calculation, and antiproliferative activity against human cancer cell lines

artículo científico publicado en 2018

Tropinone-Derived Alkaloids as Potent Anticancer Agents: Synthesis, Tyrosinase Inhibition, Mechanism of Action, DFT Calculation, and Molecular Docking Studies

artículo científico publicado en 2020

[Increased urinary excretion of the neurotoxic side-chain metabolites of ifosphamide in children with polymorphism of the glutathione S-transferases genes]

scientific article published on 01 July 2005

Lista de obras de

A new method for distinguishing between enantiomers and racemates and assignment of enantiomeric purity by means of solid-state NMR. Examples from oxazaphosphorinanes

Acyloxymethyl esters of isophosphoramide mustard as new anticancer prodrugs

Analysis of the urinary excretion of ifosfamide and its N-dechloroethylated metabolites in children using 31P-NMR spectroscopy

Classical oxazaphosphorines--metabolism and therapeutic properties--new implications

Discovery and evaluation of efficient selenazoles with high antifungal activity against Candida spp

Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design, one-pot tricomponent synthesis, and lipophilicity determination

Ifosfamide. Metabolic studies, new therapeutic approaches and new analogs

Isophosphoramide mustard analogues as prodrugs for anticancer gene-directed enzyme-prodrug therapy (GDEPT).

Oxazaphosphorinane drugs. New analogues, metabolic studies, and therapeutic approaches

Phosphate prodrugs of isophosphoramide mustard.

Role of GSTM1, GSTP1, and GSTT1 gene polymorphism in ifosfamide metabolism affecting neurotoxicity and nephrotoxicity in children

Studies on the side-chain hydroxylation of ifosfamide and its bromo analogue

Synthesis and Antimicrobial Activities of (4,5,6,7-Tetrahydro-1H-indazol- 2(3H)-yl)thiazole Derivatives

Synthesis and anticonvulsant activities of novel 2-(cyclopentylmethylene)hydrazinyl-1,3-thiazoles in mouse models of seizures

Synthesis and antimicrobial activities of novel 6-(1,3-thiazol-4-yl)-1,3-benzoxazol-2(3H)-one derivatives

Synthesis and antitumour activity of stereoisomers of 4-hydroperoxy derivatives of ifosfamide and its bromo analogue.

Synthesis and biological evaluation of novel 2-(1H-imidazol-2-ylmethylidene)hydrazinyl- 1,3-thiazoles as potential antimicrobial agents

Synthesis and in vitro antiproliferative activity of thiazole-based nitrogen mustards: the hydrogen bonding interaction between model systems and nucleobases

Synthesis of nucleoside alpha-thiotriphosphates via an oxathiaphospholane approach

Synthesis, Antibacterial Activity, Interaction with Nucleobase and Molecular Docking Studies of 4-Formylbenzoic Acid Based Thiazoles

Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles.

Synthesis, antimicrobial evaluation and theoretical prediction of NMR chemical shifts of thiazole and selenazole derivatives with high antifungal activity against Candida spp

Synthesis, in vitro biological screening and molecular docking studies of novel camphor-based thiazoles.

The Disulfide Analogues of Isophosphoramide Mustard for Anticancer Therapy

The First Stereocontrolled Solid-Phase Synthesis of Di-, Tri-, and Tetra[adenosine (2‘,5‘) phosphorothioate]s ⬇️

Thiazole-based nitrogen mustards: Design, synthesis, spectroscopic studies, DFT calculation, molecular docking, and antiproliferative activity against selected human cancer cell lines

Triazene salts: Design, synthesis, ctDNA interaction, lipophilicity determination, DFT calculation, and antiproliferative activity against human cancer cell lines

Tropinone-Derived Alkaloids as Potent Anticancer Agents: Synthesis, Tyrosinase Inhibition, Mechanism of Action, DFT Calculation, and Molecular Docking Studies

[Increased urinary excretion of the neurotoxic side-chain metabolites of ifosphamide in children with polymorphism of the glutathione S-transferases genes]