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1-[(4'-Chlorophenyl) carbonyl-4-(aryl) thiosemicarbazide derivatives as potent urease inhibitors: Synthesis, in vitro and in silico studies

scientific article published on 23 May 2018

2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors

artículo científico publicado en 2015

5-Bromo-2-aryl benzimidazole derivatives as non-cytotoxic potential dual inhibitors of α-glucosidase and urease enzymes.

artículo científico publicado en 2017

Biology-oriented drug synthesis (BIODS) of 2-(2-methyl-5-nitro-1H-imidazol-1-yl)ethyl aryl ether derivatives, in vitro α-amylase inhibitory activity and in silico studies.

artículo científico publicado en 2017

Biology-oriented drug synthesis (BIODS): In vitro β-glucuronidase inhibitory and in silico studies on 2-(2-methyl-5-nitro-1H-imidazol-1-yl)ethyl aryl carboxylate derivatives.

artículo científico publicado en 2016

Carbohydrazones as new class of carbonic anhydrase inhibitors: Synthesis, kinetics, and ligand docking studies.

artículo científico publicado en 2017

Coumarin sulfonates: As potential leads for ROS inhibition

artículo científico publicado en 2016

Dihydropyrimidones: As novel class of β-glucuronidase inhibitors.

artículo científico publicado en 2016

Facile synthesis of novel substituted aryl-thiazole (SAT) analogs via one-pot multi-component reaction as potent cytotoxic agents against cancer cell lines.

artículo científico publicado en 2016

Hydrazinyl arylthiazole based pyridine scaffolds: Synthesis, structural characterization, in vitro α-glucosidase inhibitory activity, and in silico studies.

artículo científico publicado en 2017

New Hybrid Hydrazinyl Thiazole Substituted Chromones: As Potential α-Amylase Inhibitors and Radical (DPPH & ABTS) Scavengers

artículo científico publicado en 2017

Syntheses of new 3-thiazolyl coumarin derivatives, in vitro α-glucosidase inhibitory activity, and molecular modeling studies

artículo científico publicado en 2016

Synthesis and in silico studies of novel sulfonamides having oxadiazole ring: As β-glucuronidase inhibitors.

artículo científico publicado en 2017

Synthesis of 6-chloro-2-Aryl-1H-imidazo[4,5-b]pyridine derivatives: Antidiabetic, antioxidant, β-glucuronidase inhibiton and their molecular docking studies

artículo científico publicado en 2016

Synthesis, in vitro [Formula: see text]-glucosidase inhibitory activity, and in silico study of (E)-thiosemicarbazones and (E)-2-(2-(arylmethylene)hydrazinyl)-4-arylthiazole derivatives

artículo científico publicado en 2018

Synthesis, in vitro urease inhibitory activity, and molecular docking studies of thiourea and urea derivatives

artículo científico publicado en 2018

Synthesis, in vitro α-glucosidase inhibitory activity and molecular docking studies of new thiazole derivatives

artículo científico publicado en 2016

Synthesis, in vitro β-glucuronidase inhibitory activity and in silico studies of novel (E)-4-Aryl-2-(2-(pyren-1-ylmethylene)hydrazinyl)thiazoles.

artículo científico publicado en 2016

Synthesis, α-glucosidase inhibitory activity and in silico study of tris-indole hybrid scaffold with oxadiazole ring: As potential leads for the management of type-II diabetes mellitus.

artículo científico publicado en 2017

Synthesis, β-glucuronidase inhibition and molecular docking studies of hybrid bisindole-thiosemicarbazides analogs

artículo científico publicado en 2016

Thiadiazole derivatives as New Class of β-glucuronidase inhibitors.

artículo científico publicado en 2016

Xanthine oxidase inhibitory activity of nicotino/isonicotinohydrazides: A systematic approach from in vitro, in silico to in vivo studies

artículo científico publicado en 2017