Lista de obras -

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

artículo científico publicado en 2015

A structure-activity relationship study of the affinity of selected imidazo[1,2-a]pyridine derivatives, congeners of zolpidem, for the omega 1-subtype of the benzodiazepine receptor

artículo científico publicado en 2001

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

artículo científico publicado en 2014

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 5. Synthesis of some triazolo[4,3-b]pyridazine and pyridazino[6,1-c]triazine derivatives as potential benzodiazepine receptor ligands

artículo científico publicado el 1 de noviembre de 1996

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 6. Aromatization of some tetrahydrotriazolo[4,3-b]pyridazine derivatives with potential activity as benzodiazepine receptor ligands

artículo científico publicado el 1 de julio de 1997

Bicyclic [b]-heteroannulated pyridazine derivatives--II. Structure-activity relationships in the 6-aryltriazolo-[4,3-b]pyridazine ligands of the benzodiazepine receptor

artículo científico publicado en 1994

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

artículo científico publicado en 2015

Conformational investigation of alpha, beta-dehydropeptides. Part VI. Molecular and crystal structure of benzyloxycarbonylglycyl-(Z)-dehydrophenylalanine

artículo científico publicado en 1994

Convenient way of synthesis and crystal structure of 1-[(5-chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine, a histamine H4 receptor antagonist

Crystal and Molecular Structure of 4-[ω-(Benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a Different Pharmacological Activity

Crystallographic and spectroscopic studies of 5-arylidene-2-amino-imidazol-4-ones

artículo científico publicado en 2009

Crystallographic studies of (Z) and (E) isomers of 2-amino-5-(2-chlorobenzylidene)-1-methyl-1H-imidazol-4(5H)-one

artículo científico publicado en 2010

Design, synthesis, and anticonvulsant activity of new N-Mannich bases derived from spirosuccinimides and spirohydantoins.

artículo científico publicado en 2010

Desulfurization of 2-thiouracil nucleosides: conformational studies of 4-pyrimidinone nucleosides

artículo científico publicado en 2011

Efficient synthesis of 2'-deoxyzebularine and its α-anomer by the silyl method of N-glycosylation. Crystal structures and conformational study in solution.

artículo científico publicado en 2014

Five-membered heterocycles. Part III. Aromaticity of 1,3-imidazole in 5+n hetero-bicyclic molecules

article

Four- and five-coordinate copper(II) complexes with N-(4,4-diphenyl-5-oxo-4,5-dihydro-1H-imidazol-2-yl)glycine

artículo científico publicado en 2008

From crystallographic data to the creation of a binding model with a receptor

artículo científico publicado en 2000

Fused 2-thiohydantoin derivatives: evaluation as potential antioxidants

scientific article published on 01 April 1997

Glycine derivatives of imidazolones as potential ligands of glycine binding site of NMDA receptors. Part 1

scientific article published on 01 September 1998

Imidazo-thiazine, -diazinone and -diazepinone derivatives. Synthesis, structure and benzodiazepine receptor binding

artículo científico publicado en 2001

Imidazo[2,1-b]thiazepines: synthesis, structure and evaluation of benzodiazepine receptor binding.

artículo científico publicado en 2004

Impact of the aryl substituent kind and distance from pyrimido[2,1-f]purindiones on the adenosine receptor selectivity and antagonistic properties.

artículo científico publicado en 2003

Inhibition of cryptosporidium parvum in vitro by 9-(alkylthio)acridine derivatives

artículo científico publicado en 2000

N9-benzyl-substituted 1,3-dimethyl- and 1,3-dipropyl-pyrimido[2,1-f]purinediones: synthesis and structure-activity relationships at adenosine A1 and A2A receptors

artículo científico publicado en 2007

Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: Structure–activity relationships as adenosine A1 and A2A receptor ligands

artículo científico publicado en 2007

Quantitative analysis of structure-activity relationship in the acridine serie. Part 1: Antiparasitic 9-thioaryl-acridine derivatives

scientific article published on 01 September 2000

Quantitative analysis of structure-activity relationship in the acridine series. Part 2: Antitumor 9-thiadiazolo-acridine derivatives

scientific article published on 01 November 2000

Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors.

artículo científico publicado en 2016

Structural and electronic conditions for anticonvulsant activity of bicyclic hydantoin derivatives

artículo científico publicado en 1995

Structure and activity studies on glycine receptor ligands. Part 5. Diphenyl imidazolin-4-one glycinamides

artículo científico publicado en 1998

Structure of an anticonvulsant N-methyl-m-bromophenylsuccinimide ⬇️

artículo científico publicado el 15 de enero de 1992

Structure-activity relationship investigations of the modulating effect of core substituents on the affinity of pyrazoloquinolinone congeners for the benzodiazepine receptor

artículo científico publicado en 1998

Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

artículo científico publicado en 1999

Structures of three N-pyridyl-2-phenylsuccinimides and structural evidence for substituent effects on anticonvulsant properties

artículo científico publicado en 1990

Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α₁-adrenoceptor antagonistic properties

artículo científico publicado en 2012

Synthesis and anticonvulsant activity of new fluorinated N-phenyl- and N-benzyl-2-azaspiro[4.4]nonane- and [4.5]decane-1,3-dione derivatives: Part III

artículo científico publicado en 2006

Synthesis and anticonvulsant properties of new N-Mannich bases derived from 3,3-diphenyl- and 3-ethyl-3-methyl-pyrrolidine-2,5-diones. Part III.

artículo científico publicado en 2012

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

artículo científico publicado en 2017

Synthesis and biological activity of tricyclic aryloimidazo-, pyrimido-, and diazepinopurinediones

artículo científico publicado en 2006

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

artículo científico publicado en 2011

Synthesis and effects on chloroquine susceptibility in Plasmodium falciparum of a series of new dihydroanthracene derivatives

artículo científico publicado en 2002

Synthesis, biological activity and molecular modelling studies of tricyclic alkylimidazo-, pyrimido- and diazepinopurinediones

artículo científico publicado en 2013

Synthesis, physicochemical and anticonvulsant properties of N-benzyl and N-aminophenyl derivatives of 2-azaspiro[4.4]nonane and [4.5]decane-1,3-dione. Part I.

artículo científico publicado en 2005

Synthesis, physicochemical and anticonvulsant properties of new N-pyridyl derivatives of 3-phenyl- and 3,3-diphenyl-succinimides

artículo científico publicado en 1999

Tricyclic oxazolo[2,3-f]purinediones: potency as adenosine receptor ligands and anticonvulsants.

artículo científico publicado en 2004

Use of molecular electrostatic potentials for analysis of anticonvulsant activities of phenylsuccinimides

scientific article published on 01 January 1993

tert-Butyl N-[(S)-3-isobutyl-2-oxooxetan-3-yl]carbamate

artículo científico publicado en 2007

tert-Butyl N-[(S)-3-isopropyl-2-oxo-oxetan-3-yl]carbamate

artículo científico publicado en 2008

Lista de obras de

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

A structure-activity relationship study of the affinity of selected imidazo[1,2-a]pyridine derivatives, congeners of zolpidem, for the omega 1-subtype of the benzodiazepine receptor

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 5. Synthesis of some triazolo[4,3-b]pyridazine and pyridazino[6,1-c]triazine derivatives as potential benzodiazepine receptor ligands

Bicyclic [b]-heteroannelated pyridazine derivatives. Part 6. Aromatization of some tetrahydrotriazolo[4,3-b]pyridazine derivatives with potential activity as benzodiazepine receptor ligands

Bicyclic [b]-heteroannulated pyridazine derivatives--II. Structure-activity relationships in the 6-aryltriazolo-[4,3-b]pyridazine ligands of the benzodiazepine receptor

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

Conformational investigation of alpha, beta-dehydropeptides. Part VI. Molecular and crystal structure of benzyloxycarbonylglycyl-(Z)-dehydrophenylalanine

Convenient way of synthesis and crystal structure of 1-[(5-chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazine, a histamine H4 receptor antagonist

Crystal and Molecular Structure of 4-[ω-(Benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a Different Pharmacological Activity

Crystallographic and spectroscopic studies of 5-arylidene-2-amino-imidazol-4-ones

Crystallographic studies of (Z) and (E) isomers of 2-amino-5-(2-chlorobenzylidene)-1-methyl-1H-imidazol-4(5H)-one

Design, synthesis, and anticonvulsant activity of new N-Mannich bases derived from spirosuccinimides and spirohydantoins.

Desulfurization of 2-thiouracil nucleosides: conformational studies of 4-pyrimidinone nucleosides

Efficient synthesis of 2'-deoxyzebularine and its α-anomer by the silyl method of N-glycosylation. Crystal structures and conformational study in solution.

Five-membered heterocycles. Part III. Aromaticity of 1,3-imidazole in 5+n hetero-bicyclic molecules

Four- and five-coordinate copper(II) complexes with N-(4,4-diphenyl-5-oxo-4,5-dihydro-1H-imidazol-2-yl)glycine

From crystallographic data to the creation of a binding model with a receptor

Fused 2-thiohydantoin derivatives: evaluation as potential antioxidants

Glycine derivatives of imidazolones as potential ligands of glycine binding site of NMDA receptors. Part 1

Imidazo-thiazine, -diazinone and -diazepinone derivatives. Synthesis, structure and benzodiazepine receptor binding

Imidazo[2,1-b]thiazepines: synthesis, structure and evaluation of benzodiazepine receptor binding.

Impact of the aryl substituent kind and distance from pyrimido[2,1-f]purindiones on the adenosine receptor selectivity and antagonistic properties.

Inhibition of cryptosporidium parvum in vitro by 9-(alkylthio)acridine derivatives

N9-benzyl-substituted 1,3-dimethyl- and 1,3-dipropyl-pyrimido[2,1-f]purinediones: synthesis and structure-activity relationships at adenosine A1 and A2A receptors

Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: Structure–activity relationships as adenosine A1 and A2A receptor ligands

Quantitative analysis of structure-activity relationship in the acridine serie. Part 1: Antiparasitic 9-thioaryl-acridine derivatives

Quantitative analysis of structure-activity relationship in the acridine series. Part 2: Antitumor 9-thiadiazolo-acridine derivatives

Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors.

Structural and electronic conditions for anticonvulsant activity of bicyclic hydantoin derivatives

Structure and activity studies on glycine receptor ligands. Part 5. Diphenyl imidazolin-4-one glycinamides

Structure of an anticonvulsant N-methyl-m-bromophenylsuccinimide ⬇️

Structure-activity relationship investigations of the modulating effect of core substituents on the affinity of pyrazoloquinolinone congeners for the benzodiazepine receptor

Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

Structures of three N-pyridyl-2-phenylsuccinimides and structural evidence for substituent effects on anticonvulsant properties

Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α₁-adrenoceptor antagonistic properties

Synthesis and anticonvulsant activity of new fluorinated N-phenyl- and N-benzyl-2-azaspiro[4.4]nonane- and [4.5]decane-1,3-dione derivatives: Part III

Synthesis and anticonvulsant properties of new N-Mannich bases derived from 3,3-diphenyl- and 3-ethyl-3-methyl-pyrrolidine-2,5-diones. Part III.

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

Synthesis and biological activity of tricyclic aryloimidazo-, pyrimido-, and diazepinopurinediones

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

Synthesis and effects on chloroquine susceptibility in Plasmodium falciparum of a series of new dihydroanthracene derivatives

Synthesis, biological activity and molecular modelling studies of tricyclic alkylimidazo-, pyrimido- and diazepinopurinediones

Synthesis, physicochemical and anticonvulsant properties of N-benzyl and N-aminophenyl derivatives of 2-azaspiro[4.4]nonane and [4.5]decane-1,3-dione. Part I.

Synthesis, physicochemical and anticonvulsant properties of new N-pyridyl derivatives of 3-phenyl- and 3,3-diphenyl-succinimides

Tricyclic oxazolo[2,3-f]purinediones: potency as adenosine receptor ligands and anticonvulsants.

Use of molecular electrostatic potentials for analysis of anticonvulsant activities of phenylsuccinimides

tert-Butyl N-[(S)-3-isobutyl-2-oxooxetan-3-yl]carbamate

tert-Butyl N-[(S)-3-isopropyl-2-oxo-oxetan-3-yl]carbamate