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A series of benzylidene linked to hydrazinecarbothioamide as tyrosinase inhibitors Synthesis, biological evaluation and structure-activity relationship

artículo científico publicado en 2020

1,2,3-Triazole-based kojic acid analogs as potent tyrosinase inhibitors: Design, synthesis and biological evaluation

scientific article published on 31 October 2018

1,2,3-Triazole-linked 5-benzylidene (thio)barbiturates as novel tyrosinase inhibitors and free-radical scavengers

artículo científico publicado en 2020

4H-benzochromene derivatives as novel tyrosinase inhibitors and radical scavengers: synthesis, biological evaluation, and molecular docking analysis

artículo científico publicado en 2020

6-Methoxy-3,4-dihydronaphthalenone Chalcone-like Derivatives as Potent Tyrosinase Inhibitors and Radical Scavengers

artículo científico publicado en 2018

A COX/5-LOX Inhibitor Licofelone Revealed Anticonvulsant Properties Through iNOS Diminution in Mice

artículo científico publicado en 2015

Design, synthesis, cytotoxicity evaluation and docking studies of 1,2,4-triazine derivatives bearing different arylidene-hydrazinyl moieties as potential mTOR inhibitors.

artículo científico publicado en 2018

Design, synthesis, in vitro and in silico studies of novel Schiff base derivatives of 2-hydroxy-4-methoxybenzamide as tyrosinase inhibitors

artículo científico publicado en 2020

Kojic acid-natural product conjugates as mushroom tyrosinase inhibitors

scientific article published on 16 June 2020

Long Chain Alkyl Esters of Hydroxycinnamic Acids as Promising Anticancer Agents: Selective Induction of Apoptosis in Cancer Cells

artículo científico publicado en 2017

Novel morpholine containing cinnamoyl amides as potent tyrosinase inhibitors

artículo científico publicado en 2019

Novel small molecule therapeutic agents for Alzheimer disease: Focusing on BACE1 and multi-target directed ligands

artículo científico publicado en 2020

One-pot synthesis of thioxo-tetrahydropyrimidine derivatives as potent β-glucuronidase inhibitor, biological evaluation, molecular docking and molecular dynamics studies

artículo científico publicado en 2020

Oxytocin is involved in the proconvulsant effects of Sildenafil: Possible role of CREB.

artículo científico publicado en 2016

Oxytocinergic system mediates the proconvulsant effects of sildenafil: The role of calcineurin

scientific article published on 14 April 2020

Phthalimide-1,2,3-triazole hybrid compounds as tyrosinase inhibitors; synthesis, biological evaluation and molecular docking analysis

Structure-Based Design, Synthesis, Biological Evaluation and Molecular Docking Study of 4-Hydroxy-N'-methylenebenzohydrazide Derivatives Acting as Tyrosinase Inhibitors as Potentiate Anti-Melanogenesis Activities

artículo científico publicado en 2019

Structure-based design, synthesis, molecular docking study and biological evaluation of 1,2,4-triazine derivatives acting as COX/15-LOX inhibitors with anti-oxidant activities

artículo científico publicado en 2016

Synthesis and cytotoxic activity of novel poly-substituted imidazo[2,1-c][1,2,4]triazin-6-amines

artículo científico publicado en 2015

Synthesis of New Benzimidazole-1,2,3-triazole Hybrids as Tyrosinase Inhibitors

artículo científico publicado en 2018

Synthesis, biological evaluation and molecular docking analysis of vaniline-benzylidenehydrazine hybrids as potent tyrosinase inhibitors

scientific article published on 07 April 2020

The Healing Effect of and Mixture in Excisional Full Thickness Skin Wounds: Stereological Study

The natural-based optimization of kojic acid conjugated to different thio-quinazolinones as potential anti-melanogenesis agents with tyrosinase inhibitory activity

scientific article published in 2021

Topical Nicotinamide Improves Tissue Regeneration in Excisional Full-Thickness Skin Wounds: A Stereological and Pathological Study

artículo científico publicado en 2015

Topical simvastatin enhances tissue regeneration in full-thickness skin wounds in rat models

artículo científico publicado en 2014

Verapamil, a Calcium-Channel Blocker, Improves the Wound Healing Process in Rats with Excisional Full-Thickness Skin Wounds Based on Stereological Parameters.

artículo científico publicado en 2016

Veratric acid derivatives containing benzylidene-hydrazine moieties as promising tyrosinase inhibitors and free radical scavengers

scientific article published on 10 April 2019